CY2014037I2 - C-MET MODULATORS AND METHODS OF USE - Google Patents

C-MET MODULATORS AND METHODS OF USE

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Publication number
CY2014037I2
CY2014037I2 CY2014037C CY2014037C CY2014037I2 CY 2014037 I2 CY2014037 I2 CY 2014037I2 CY 2014037 C CY2014037 C CY 2014037C CY 2014037 C CY2014037 C CY 2014037C CY 2014037 I2 CY2014037 I2 CY 2014037I2
Authority
CY
Cyprus
Prior art keywords
methods
met modulators
modulators
met
Prior art date
Application number
CY2014037C
Other languages
Greek (el)
Other versions
CY2014037I1 (en
Original Assignee
Exelixis, Inc.
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34397024&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY2014037(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Exelixis, Inc. filed Critical Exelixis, Inc.
Publication of CY2014037I1 publication Critical patent/CY2014037I1/en
Publication of CY2014037I2 publication Critical patent/CY2014037I2/en

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20—Oxygen atoms
    • C07D215/22—Oxygen atoms attached in position 2 or 4
    • C07D215/233—Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 4
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
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    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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JP2011042686A (en) 2011-03-03
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US11124482B2 (en) 2021-09-21
US20140155396A1 (en) 2014-06-05
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