CY1121174T1 - 4-IMIDAZOPYRIDAZIN-1-YL-BENZAMIDS AND 4-IMIDAZOTRIAZIN-1-YL-BENZAMIDS AS BTC INhibitors - Google Patents

4-IMIDAZOPYRIDAZIN-1-YL-BENZAMIDS AND 4-IMIDAZOTRIAZIN-1-YL-BENZAMIDS AS BTC INhibitors

Info

Publication number
CY1121174T1
CY1121174T1 CY20191100084T CY191100084T CY1121174T1 CY 1121174 T1 CY1121174 T1 CY 1121174T1 CY 20191100084 T CY20191100084 T CY 20191100084T CY 191100084 T CY191100084 T CY 191100084T CY 1121174 T1 CY1121174 T1 CY 1121174T1
Authority
CY
Cyprus
Prior art keywords
benzamids
imidazotriazin
imidazopyridazin
btc
inhibitors
Prior art date
Application number
CY20191100084T
Other languages
Greek (el)
Inventor
Tjeerd A. Barf
Christiaan Gerardus Johannes Maria Jans
de Adrianus Petrus Antonius MAN
Arthur A. Oubrie
Hans C.A. Raaijmakers
Johannes Bernardus Maria Rewinkel
Jan-Gerard Sterrenburg
Jacobus C.H.M. Wijkmans
Original Assignee
Merck Sharp & Dohme B.V.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP12733505.7A external-priority patent/EP2734522B1/en
Application filed by Merck Sharp & Dohme B.V. filed Critical Merck Sharp & Dohme B.V.
Publication of CY1121174T1 publication Critical patent/CY1121174T1/en

Links

Classifications

    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Abstract

Η παρούσα εφεύρεση σχετίζεται με ενώσεις 6-5μελούς συντηγμένου δακτυλίου πυριδίνης σύμφωνα με τον τύπο (I), ή ένα φαρμακευτικά αποδεκτό άλας αυτών, ή με φαρμακευτικές συνθέσεις που περιέχουν αυτές τις ενώσεις και με τη χρήση τους στη θεραπεία. Ειδικότερα, η παρούσα εφεύρεση σχετίζεται με τη χρήση ενώσεων 6-5 μελούς συντηγμένου δακτυλίου πυριδίνης σύμφωνα με τον τύπο I στη θεραπεία προκαλούμενων από Τυροσινική Κινάση του Βruton (Btk) διαταραχών.The present invention relates to compounds of 6-5 membered fused pyridine rings according to formula (I), or a pharmaceutically acceptable salt thereof, or to pharmaceutical compositions containing these compounds and for use in therapy. More particularly, the present invention relates to the use of compounds of 6-5 membered fused pyridine ring according to formula I in the treatment of Bruton Tyrosine Kinase (Btk) disorders.

CY20191100084T 2011-07-19 2019-01-22 4-IMIDAZOPYRIDAZIN-1-YL-BENZAMIDS AND 4-IMIDAZOTRIAZIN-1-YL-BENZAMIDS AS BTC INhibitors CY1121174T1 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201161509397P 2011-07-19 2011-07-19
EP11174578 2011-07-19
EP12733505.7A EP2734522B1 (en) 2011-07-19 2012-07-11 4-imidazopyridazin-1-yl-benzamides and 4-imidazotriazin-1-yl-benzamides as btk-inhibitors
PCT/EP2012/063552 WO2013010868A1 (en) 2011-07-19 2012-07-11 4 - imidazopyridazin- 1 -yl-benzamides and 4 - imidazotriazin- 1 - yl - benzamides as btk- inhibitors

Publications (1)

Publication Number Publication Date
CY1121174T1 true CY1121174T1 (en) 2020-05-29

Family

ID=67956153

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20191100084T CY1121174T1 (en) 2011-07-19 2019-01-22 4-IMIDAZOPYRIDAZIN-1-YL-BENZAMIDS AND 4-IMIDAZOTRIAZIN-1-YL-BENZAMIDS AS BTC INhibitors

Country Status (8)

Country Link
CY (1) CY1121174T1 (en)
LT (2) LT3689878T (en)
ME (1) ME03310B (en)
NI (1) NI201400004A (en)
NL (1) NL301097I2 (en)
NO (1) NO2021016I1 (en)
PT (1) PT2734522T (en)
TR (1) TR201901013T4 (en)

Also Published As

Publication number Publication date
NI201400004A (en) 2014-10-10
PT2734522T (en) 2019-02-04
LT3689878T (en) 2021-11-25
NL301097I1 (en) 2021-03-24
LTPA2021004I1 (en) 2021-04-12
NO2021016I1 (en) 2021-04-09
LTC2734522I2 (en) 2022-09-26
ME03310B (en) 2019-10-20
TR201901013T4 (en) 2019-02-21
NL301097I2 (en) 2021-04-12

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