CY1121174T1 - 4-IMIDAZOPYRIDAZIN-1-YL-BENZAMIDS AND 4-IMIDAZOTRIAZIN-1-YL-BENZAMIDS AS BTC INhibitors - Google Patents
4-IMIDAZOPYRIDAZIN-1-YL-BENZAMIDS AND 4-IMIDAZOTRIAZIN-1-YL-BENZAMIDS AS BTC INhibitorsInfo
- Publication number
- CY1121174T1 CY1121174T1 CY20191100084T CY191100084T CY1121174T1 CY 1121174 T1 CY1121174 T1 CY 1121174T1 CY 20191100084 T CY20191100084 T CY 20191100084T CY 191100084 T CY191100084 T CY 191100084T CY 1121174 T1 CY1121174 T1 CY 1121174T1
- Authority
- CY
- Cyprus
- Prior art keywords
- benzamids
- imidazotriazin
- imidazopyridazin
- btc
- inhibitors
- Prior art date
Links
Classifications
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Abstract
Η παρούσα εφεύρεση σχετίζεται με ενώσεις 6-5μελούς συντηγμένου δακτυλίου πυριδίνης σύμφωνα με τον τύπο (I), ή ένα φαρμακευτικά αποδεκτό άλας αυτών, ή με φαρμακευτικές συνθέσεις που περιέχουν αυτές τις ενώσεις και με τη χρήση τους στη θεραπεία. Ειδικότερα, η παρούσα εφεύρεση σχετίζεται με τη χρήση ενώσεων 6-5 μελούς συντηγμένου δακτυλίου πυριδίνης σύμφωνα με τον τύπο I στη θεραπεία προκαλούμενων από Τυροσινική Κινάση του Βruton (Btk) διαταραχών.The present invention relates to compounds of 6-5 membered fused pyridine rings according to formula (I), or a pharmaceutically acceptable salt thereof, or to pharmaceutical compositions containing these compounds and for use in therapy. More particularly, the present invention relates to the use of compounds of 6-5 membered fused pyridine ring according to formula I in the treatment of Bruton Tyrosine Kinase (Btk) disorders.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201161509397P | 2011-07-19 | 2011-07-19 | |
EP11174578 | 2011-07-19 | ||
EP12733505.7A EP2734522B1 (en) | 2011-07-19 | 2012-07-11 | 4-imidazopyridazin-1-yl-benzamides and 4-imidazotriazin-1-yl-benzamides as btk-inhibitors |
PCT/EP2012/063552 WO2013010868A1 (en) | 2011-07-19 | 2012-07-11 | 4 - imidazopyridazin- 1 -yl-benzamides and 4 - imidazotriazin- 1 - yl - benzamides as btk- inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1121174T1 true CY1121174T1 (en) | 2020-05-29 |
Family
ID=67956153
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20191100084T CY1121174T1 (en) | 2011-07-19 | 2019-01-22 | 4-IMIDAZOPYRIDAZIN-1-YL-BENZAMIDS AND 4-IMIDAZOTRIAZIN-1-YL-BENZAMIDS AS BTC INhibitors |
Country Status (8)
Country | Link |
---|---|
CY (1) | CY1121174T1 (en) |
LT (2) | LT3689878T (en) |
ME (1) | ME03310B (en) |
NI (1) | NI201400004A (en) |
NL (1) | NL301097I2 (en) |
NO (1) | NO2021016I1 (en) |
PT (1) | PT2734522T (en) |
TR (1) | TR201901013T4 (en) |
-
2012
- 2012-07-11 LT LTEP19215783.2T patent/LT3689878T/en unknown
- 2012-07-11 ME MEP-2019-4A patent/ME03310B/en unknown
- 2012-07-11 TR TR2019/01013T patent/TR201901013T4/en unknown
- 2012-07-11 PT PT12733505T patent/PT2734522T/en unknown
-
2014
- 2014-01-17 NI NI201400004A patent/NI201400004A/en unknown
-
2019
- 2019-01-22 CY CY20191100084T patent/CY1121174T1/en unknown
-
2021
- 2021-03-22 NL NL301097C patent/NL301097I2/en unknown
- 2021-03-24 LT LTPA2021004C patent/LTC2734522I2/en unknown
- 2021-04-09 NO NO2021016C patent/NO2021016I1/en unknown
Also Published As
Publication number | Publication date |
---|---|
NI201400004A (en) | 2014-10-10 |
PT2734522T (en) | 2019-02-04 |
LT3689878T (en) | 2021-11-25 |
NL301097I1 (en) | 2021-03-24 |
LTPA2021004I1 (en) | 2021-04-12 |
NO2021016I1 (en) | 2021-04-09 |
LTC2734522I2 (en) | 2022-09-26 |
ME03310B (en) | 2019-10-20 |
TR201901013T4 (en) | 2019-02-21 |
NL301097I2 (en) | 2021-04-12 |
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