NI201400004A - 4 - IMIDAZOPYRIDAZIN - 1 - IL - BENZAMIDES AND 4 - IMIDAZOTRIAZIN - 1 - IL - BENZAMIDES AS BTK INHIBITORS - Google Patents

4 - IMIDAZOPYRIDAZIN - 1 - IL - BENZAMIDES AND 4 - IMIDAZOTRIAZIN - 1 - IL - BENZAMIDES AS BTK INHIBITORS

Info

Publication number
NI201400004A
NI201400004A NI201400004A NI201400004A NI201400004A NI 201400004 A NI201400004 A NI 201400004A NI 201400004 A NI201400004 A NI 201400004A NI 201400004 A NI201400004 A NI 201400004A NI 201400004 A NI201400004 A NI 201400004A
Authority
NI
Nicaragua
Prior art keywords
benzamides
imidazotriazin
imidazopyridazin
btk inhibitors
formula
Prior art date
Application number
NI201400004A
Other languages
Spanish (es)
Inventor
A Barf Tjeerd
Gerardus Johannes Maria Jans Christiaan
Adrianus Petrus Antonius Man De
A Oubrie Arthur
C A Raaijmakers Hans
Bernardus Maria Rewinkel Johannes
C H M Wijkmans Jacobus
Sterrenburg Jan-Gerard
Original Assignee
Merck Sharp & Dohme
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Sharp & Dohme filed Critical Merck Sharp & Dohme
Publication of NI201400004A publication Critical patent/NI201400004A/en

Links

Classifications

    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Abstract

La presente invención se refiere a compuestos de anillos de piridina fusionados de 5-6 miembros según la fórmula I o una sal farmacéuticamente aceptable de los mismos o a composiciones farmacéuticas que comprenden estos compuestos y a su uso en terapia. En particular, la presente invención se refiere al uso de compuestos de anillos de piridina fusionados de 5-6 miembros según la fórmula I en el tratamiento de trastornos mediados por tirosina cinasa de Bruton (BK).The present invention relates to 5-6 membered fused pyridine ring compounds according to formula I or a pharmaceutically acceptable salt thereof or to pharmaceutical compositions comprising these compounds and their use in therapy. In particular, the present invention relates to the use of 5-6 membered fused pyridine ring compounds according to formula I in the treatment of disorders mediated by Bruton's tyrosine kinase (BK).

NI201400004A 2011-07-19 2014-01-17 4 - IMIDAZOPYRIDAZIN - 1 - IL - BENZAMIDES AND 4 - IMIDAZOTRIAZIN - 1 - IL - BENZAMIDES AS BTK INHIBITORS NI201400004A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161509397P 2011-07-19 2011-07-19
EP11174578 2011-07-19

Publications (1)

Publication Number Publication Date
NI201400004A true NI201400004A (en) 2014-10-10

Family

ID=67956153

Family Applications (1)

Application Number Title Priority Date Filing Date
NI201400004A NI201400004A (en) 2011-07-19 2014-01-17 4 - IMIDAZOPYRIDAZIN - 1 - IL - BENZAMIDES AND 4 - IMIDAZOTRIAZIN - 1 - IL - BENZAMIDES AS BTK INHIBITORS

Country Status (8)

Country Link
CY (1) CY1121174T1 (en)
LT (2) LT3689878T (en)
ME (1) ME03310B (en)
NI (1) NI201400004A (en)
NL (1) NL301097I2 (en)
NO (1) NO2021016I1 (en)
PT (1) PT2734522T (en)
TR (1) TR201901013T4 (en)

Also Published As

Publication number Publication date
NO2021016I1 (en) 2021-04-09
CY1121174T1 (en) 2020-05-29
LT3689878T (en) 2021-11-25
PT2734522T (en) 2019-02-04
LTPA2021004I1 (en) 2021-04-12
NL301097I1 (en) 2021-03-24
NL301097I2 (en) 2021-04-12
TR201901013T4 (en) 2019-02-21
ME03310B (en) 2019-10-20
LTC2734522I2 (en) 2022-09-26

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