CY1112032T1 - Χρηση της 7-τ-βουτοξυιμινομεθυλοκαμπτοθεκινης για τη θεραπεια νεοπλασματων της μητρας - Google Patents

Χρηση της 7-τ-βουτοξυιμινομεθυλοκαμπτοθεκινης για τη θεραπεια νεοπλασματων της μητρας

Info

Publication number
CY1112032T1
CY1112032T1 CY20111101092T CY111101092T CY1112032T1 CY 1112032 T1 CY1112032 T1 CY 1112032T1 CY 20111101092 T CY20111101092 T CY 20111101092T CY 111101092 T CY111101092 T CY 111101092T CY 1112032 T1 CY1112032 T1 CY 1112032T1
Authority
CY
Cyprus
Prior art keywords
treatment
butoxyminomethylcomptothekine
mathematics
domestic
butoxyiminomethylcamptothecin
Prior art date
Application number
CY20111101092T
Other languages
English (en)
Inventor
Paolo Carminati
Marco Corsi
Claudio Zanna
Franco Cavalli
Luca Gianni
Cristiana Sessa
Original Assignee
Sigma-Tau Industrie Farmaceutiche Riunite S.P.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sigma-Tau Industrie Farmaceutiche Riunite S.P.A. filed Critical Sigma-Tau Industrie Farmaceutiche Riunite S.P.A.
Publication of CY1112032T1 publication Critical patent/CY1112032T1/el

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4738Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4741Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having oxygen as a ring hetero atom, e.g. tubocuraran derivatives, noscapine, bicuculline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4738Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Η χρήση της 7-t-βουτοξυιμινομεθυλοκαμπτοθεκίνης περιγράφεται στην παρασκευή ενός φαρμάκου χρήσιμου για τη θεραπεία νεοπλασμάτων της μήτρας, συγκεκριμένα του καρκίνου του ενδομητρίου και του τραχήλου της μήτρας.
CY20111101092T 2004-06-11 2011-11-14 Χρηση της 7-τ-βουτοξυιμινομεθυλοκαμπτοθεκινης για τη θεραπεια νεοπλασματων της μητρας CY1112032T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT000288A ITRM20040288A1 (it) 2004-06-11 2004-06-11 Uso della 7-t-butossiimminometilcamptotecina per la preparazione di un medicamento per il trattamento delle neoplasie dell'utero.
EP05761294A EP1773451B1 (en) 2004-06-11 2005-06-08 Use of 7-t-butoxyiminomethylcamptothecin for treating uterine neoplasms

Publications (1)

Publication Number Publication Date
CY1112032T1 true CY1112032T1 (el) 2015-11-04

Family

ID=34979678

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20111101092T CY1112032T1 (el) 2004-06-11 2011-11-14 Χρηση της 7-τ-βουτοξυιμινομεθυλοκαμπτοθεκινης για τη θεραπεια νεοπλασματων της μητρας

Country Status (23)

Country Link
US (1) US7700613B2 (el)
EP (1) EP1773451B1 (el)
JP (2) JP2008501785A (el)
KR (1) KR101221640B1 (el)
CN (2) CN1953784A (el)
AR (1) AR049220A1 (el)
AT (1) ATE521351T1 (el)
AU (1) AU2005251573B2 (el)
BR (1) BRPI0511931A (el)
CA (1) CA2565213C (el)
CY (1) CY1112032T1 (el)
DK (1) DK1773451T3 (el)
ES (1) ES2372056T3 (el)
HK (1) HK1205951A1 (el)
HR (1) HRP20110718T1 (el)
IT (1) ITRM20040288A1 (el)
MX (1) MXPA06014162A (el)
PL (1) PL1773451T3 (el)
PT (1) PT1773451E (el)
RS (1) RS52038B (el)
SI (1) SI1773451T1 (el)
TW (1) TWI351283B (el)
WO (1) WO2005120643A2 (el)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1915134A2 (en) * 2005-08-10 2008-04-30 Novartis AG Formulations for 7-(t-butoxy)iminomethyl camptothecin
CA2676986A1 (en) * 2007-02-01 2008-08-07 Sigma-Tau Industrie Farmaceutiche Riunite S.P.A. Pharmaceutical composition comprising a campothecin derivative

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK1251125T3 (da) * 1995-06-21 2006-04-18 Sod Conseils Rech Applic Hidtil ukendte camptothecin-analoger, fremgangsmåde til fremstilling heraf, anvendelse heraf som lægemidler og farmaceutiske præparater indeholdende disse
FR2757514B1 (fr) * 1996-12-20 1999-02-12 Sod Conseils Rech Applic Nouveaux analogues de la camptothecine, des procedes de preparation, leur application comme medicaments et les compositions pharmaceutiques les contenant
UA57757C2 (uk) * 1996-12-20 2003-07-15 Сос'Єте Де Консей Де Решерш Е Даплікасьон С'Єнтіфік (С.К.Р.А.С.) Аналоги камптотецину, спосіб їх отримання (варіанти) і фармацевтична композиція
ES2175919T3 (es) * 1999-03-09 2002-11-16 Sigma Tau Ind Farmaceuti Derivados del camptothecin con actividad antitumoral.
US7105492B2 (en) * 1999-03-09 2006-09-12 Sigma-Tau Industrie Farmaceutiche Riunite S.P.A. Camptothecin derivatives having antitumor activity
IT1306129B1 (it) * 1999-04-13 2001-05-30 Sigma Tau Ind Farmaceuti Esteri della l-carnitina o di alcanoil l-carnitine utilizzabili comelipidi cationici per l'immissione intracellulare di composti
US6352996B1 (en) * 1999-08-03 2002-03-05 The Stehlin Foundation For Cancer Research Liposomal prodrugs comprising derivatives of camptothecin and methods of treating cancer using these prodrugs
WO2003043584A2 (en) 2001-11-20 2003-05-30 University Of Kentucky Research Foundation Engineered liposomal particles containing core-loaded pro-drugs for the controlled release of camptothecins
BRPI0410648A (pt) * 2003-05-21 2006-07-04 Novartis Ag combinação de inibidores de histona desacetilase com agentes quimioterápicos

Also Published As

Publication number Publication date
CN104352496A (zh) 2015-02-18
EP1773451A2 (en) 2007-04-18
JP2008501785A (ja) 2008-01-24
KR101221640B1 (ko) 2013-01-14
AU2005251573B2 (en) 2010-04-15
US7700613B2 (en) 2010-04-20
AR049220A1 (es) 2006-07-05
ITRM20040288A1 (it) 2004-09-11
TWI351283B (en) 2011-11-01
WO2005120643A3 (en) 2006-03-30
EP1773451B1 (en) 2011-08-24
WO2005120643A8 (en) 2006-12-14
CN1953784A (zh) 2007-04-25
PL1773451T3 (pl) 2012-01-31
PT1773451E (pt) 2011-11-02
BRPI0511931A (pt) 2008-01-22
JP2014231518A (ja) 2014-12-11
DK1773451T3 (da) 2011-11-28
ATE521351T1 (de) 2011-09-15
ES2372056T3 (es) 2012-01-13
RS52038B (en) 2012-04-30
US20080020030A1 (en) 2008-01-24
SI1773451T1 (sl) 2012-01-31
AU2005251573A1 (en) 2005-12-22
CA2565213C (en) 2012-08-07
MXPA06014162A (es) 2007-03-07
KR20070030246A (ko) 2007-03-15
HK1205951A1 (en) 2015-12-31
CA2565213A1 (en) 2005-12-22
HRP20110718T1 (hr) 2011-12-31
TW200605891A (en) 2006-02-16
WO2005120643A2 (en) 2005-12-22

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