CS212218B2 - Method of producing the new steroids of the pregnane series substituted in the position 17 - Google Patents
Method of producing the new steroids of the pregnane series substituted in the position 17 Download PDFInfo
- Publication number
- CS212218B2 CS212218B2 CS79567A CS56779A CS212218B2 CS 212218 B2 CS212218 B2 CS 212218B2 CS 79567 A CS79567 A CS 79567A CS 56779 A CS56779 A CS 56779A CS 212218 B2 CS212218 B2 CS 212218B2
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- formula
- group
- alpha
- hydroxy
- mixture
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
- C07J5/0046—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa
- C07J5/0053—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa not substituted in position 16
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
- C07J5/0046—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa
- C07J5/0061—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa substituted in position 16
- C07J5/0069—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa substituted in position 16 by a saturated or unsaturated hydrocarbon group
- C07J5/0076—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa substituted in position 16 by a saturated or unsaturated hydrocarbon group by an alkyl group
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J7/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
- C07J7/0005—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21
- C07J7/001—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group
- C07J7/004—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group substituted in position 17 alfa
- C07J7/0045—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group substituted in position 17 alfa not substituted in position 16
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B60—VEHICLES IN GENERAL
- B60W—CONJOINT CONTROL OF VEHICLE SUB-UNITS OF DIFFERENT TYPE OR DIFFERENT FUNCTION; CONTROL SYSTEMS SPECIALLY ADAPTED FOR HYBRID VEHICLES; ROAD VEHICLE DRIVE CONTROL SYSTEMS FOR PURPOSES NOT RELATED TO THE CONTROL OF A PARTICULAR SUB-UNIT
- B60W2510/00—Input parameters relating to a particular sub-units
- B60W2510/10—Change speed gearings
- B60W2510/107—Temperature
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B60—VEHICLES IN GENERAL
- B60W—CONJOINT CONTROL OF VEHICLE SUB-UNITS OF DIFFERENT TYPE OR DIFFERENT FUNCTION; CONTROL SYSTEMS SPECIALLY ADAPTED FOR HYBRID VEHICLES; ROAD VEHICLE DRIVE CONTROL SYSTEMS FOR PURPOSES NOT RELATED TO THE CONTROL OF A PARTICULAR SUB-UNIT
- B60W2720/00—Output or target parameters relating to overall vehicle dynamics
- B60W2720/10—Longitudinal speed
- B60W2720/106—Longitudinal acceleration
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Rheumatology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Pain & Pain Management (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19782803660 DE2803660A1 (de) | 1978-01-25 | 1978-01-25 | Neue in 17-position substituierte steroide der pregnanreihe, ihre herstellung und verwendung |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CS212218B2 true CS212218B2 (en) | 1982-03-26 |
Family
ID=6030585
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CS79567A CS212218B2 (en) | 1978-01-25 | 1979-01-25 | Method of producing the new steroids of the pregnane series substituted in the position 17 |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US4224320A (da) |
| EP (1) | EP0003519A1 (da) |
| JP (1) | JPS54145649A (da) |
| AT (1) | AT371824B (da) |
| AU (1) | AU529413B2 (da) |
| CA (1) | CA1139743A (da) |
| CS (1) | CS212218B2 (da) |
| DD (2) | DD150223A5 (da) |
| DE (1) | DE2803660A1 (da) |
| DK (1) | DK28679A (da) |
| ES (1) | ES477161A1 (da) |
| GB (1) | GB2013685A (da) |
| GR (1) | GR73667B (da) |
| HU (1) | HU184189B (da) |
| IE (1) | IE790135L (da) |
| IL (1) | IL56495A0 (da) |
| SU (1) | SU860708A1 (da) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2952003A1 (de) * | 1979-12-21 | 1981-07-02 | Schering Ag Berlin Und Bergkamen, 1000 Berlin | Neue kortikoid-17-thioacetale, ihre herstellung und verwendung |
| FR2552766B1 (fr) * | 1983-10-04 | 1987-06-26 | Theramex | Nouveau procede de preparation de derives de la serie du 17 a-hydroxy 19-nor progesterone |
| US4588683A (en) * | 1984-02-06 | 1986-05-13 | Eastman Kodak Company | Method of preparing 11β, 17α, 20, 21-tetrahydroxy steroids and corresponding 11β, 17α, 21-trihydroxy-20-oxo steroids |
| US4588525A (en) * | 1984-02-27 | 1986-05-13 | Molecular Biosystems, Inc. | Prodrug compounds for dermal application |
| JP2562134B2 (ja) * | 1986-09-19 | 1996-12-11 | 喜徳 喜谷 | 新規な白金−ステロイド錯体 |
| WO1994015947A1 (en) * | 1993-01-08 | 1994-07-21 | Astra Aktiebolag | Novel colon- or ileum-specific steroid derivatives |
| US5710293A (en) * | 1995-10-13 | 1998-01-20 | The Population Council, Center For Biomedical Research | Method of preparation of ester derivatives of steroids |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2924597A (en) * | 1958-04-08 | 1960-02-09 | Ormonaterapia Richter S P A | Process for the preparation of 17alpha hydroxy-progesterone, esters thereof, and intermediates therefor |
| US3187025A (en) * | 1963-06-11 | 1965-06-01 | Smith Kline French Lab | Process for preparing compound s |
| DE1543245C3 (de) * | 1965-11-26 | 1974-07-18 | Merck Patent Gmbh, 6100 Darmstadt | 16-Methy len-19-norprogesteronderivate, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Zubereitungen |
| NL6605514A (da) * | 1966-04-25 | 1967-10-26 | ||
| US3530117A (en) * | 1969-01-09 | 1970-09-22 | Merck & Co Inc | Delta**4 and delta**4,6 - 17 - hydroxy - steroidal pyrazoles of the pregnane series |
-
1978
- 1978-01-25 DE DE19782803660 patent/DE2803660A1/de not_active Withdrawn
-
1979
- 1979-01-22 EP EP79100183A patent/EP0003519A1/de not_active Withdrawn
- 1979-01-23 DK DK28679A patent/DK28679A/da not_active Application Discontinuation
- 1979-01-23 DD DD79220688A patent/DD150223A5/de unknown
- 1979-01-23 DD DD79210600A patent/DD141524A5/de unknown
- 1979-01-24 AT AT0050379A patent/AT371824B/de not_active IP Right Cessation
- 1979-01-24 GB GB7902501A patent/GB2013685A/en not_active Withdrawn
- 1979-01-24 GR GR58174A patent/GR73667B/el unknown
- 1979-01-24 HU HU79SCHE670A patent/HU184189B/hu unknown
- 1979-01-25 CA CA000320261A patent/CA1139743A/en not_active Expired
- 1979-01-25 AU AU43665/79A patent/AU529413B2/en not_active Ceased
- 1979-01-25 SU SU792718151A patent/SU860708A1/ru active
- 1979-01-25 IL IL56495A patent/IL56495A0/xx unknown
- 1979-01-25 ES ES477161A patent/ES477161A1/es not_active Expired
- 1979-01-25 US US06/006,692 patent/US4224320A/en not_active Expired - Lifetime
- 1979-01-25 JP JP660279A patent/JPS54145649A/ja active Pending
- 1979-01-25 CS CS79567A patent/CS212218B2/cs unknown
- 1979-01-30 IE IE790135A patent/IE790135L/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| HU184189B (en) | 1984-07-30 |
| DD150223A5 (de) | 1981-08-19 |
| DE2803660A1 (de) | 1979-07-26 |
| IL56495A0 (en) | 1979-03-12 |
| GB2013685A (en) | 1979-08-15 |
| AU529413B2 (en) | 1983-06-09 |
| EP0003519A1 (de) | 1979-08-22 |
| JPS54145649A (en) | 1979-11-14 |
| CA1139743A (en) | 1983-01-18 |
| SU860708A1 (ru) | 1981-08-30 |
| GR73667B (da) | 1984-03-28 |
| IE790135L (en) | 1979-07-25 |
| ES477161A1 (es) | 1979-07-01 |
| AT371824B (de) | 1983-08-10 |
| AU4366579A (en) | 1979-08-02 |
| ATA50379A (de) | 1982-12-15 |
| US4224320A (en) | 1980-09-23 |
| DD141524A5 (de) | 1980-05-07 |
| DK28679A (da) | 1979-07-26 |
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