CS196369B2 - Method of preparing 7-/alpha-/2,3-dihydro-2-oxo-1h-benzoimidazol-1-yl carbonylamino/arylacetamido/cephalosporins - Google Patents

Method of preparing 7-/alpha-/2,3-dihydro-2-oxo-1h-benzoimidazol-1-yl carbonylamino/arylacetamido/cephalosporins Download PDF

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Publication number
CS196369B2
CS196369B2 CS774095A CS409577A CS196369B2 CS 196369 B2 CS196369 B2 CS 196369B2 CS 774095 A CS774095 A CS 774095A CS 409577 A CS409577 A CS 409577A CS 196369 B2 CS196369 B2 CS 196369B2
Authority
CS
Czechoslovakia
Prior art keywords
formula
hydrogen
ylthiomethyl
oxo
methyl
Prior art date
Application number
CS774095A
Other languages
Czech (cs)
English (en)
Inventor
William H Lunn
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of CS196369B2 publication Critical patent/CS196369B2/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
CS774095A 1976-06-21 1977-06-21 Method of preparing 7-/alpha-/2,3-dihydro-2-oxo-1h-benzoimidazol-1-yl carbonylamino/arylacetamido/cephalosporins CS196369B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/698,431 US4061861A (en) 1976-06-21 1976-06-21 7-[α-(2,3-DIHYDRO-2-OXO-1H-benzimidazol-1-ylcarbonyl-amino)arylacetamido]cephalosporins

Publications (1)

Publication Number Publication Date
CS196369B2 true CS196369B2 (en) 1980-03-31

Family

ID=24805210

Family Applications (1)

Application Number Title Priority Date Filing Date
CS774095A CS196369B2 (en) 1976-06-21 1977-06-21 Method of preparing 7-/alpha-/2,3-dihydro-2-oxo-1h-benzoimidazol-1-yl carbonylamino/arylacetamido/cephalosporins

Country Status (22)

Country Link
US (1) US4061861A (ro)
JP (1) JPS52156897A (ro)
AR (1) AR213853A1 (ro)
AU (1) AU508432B2 (ro)
BE (1) BE855966A (ro)
CS (1) CS196369B2 (ro)
DD (1) DD131174A5 (ro)
DE (1) DE2727325A1 (ro)
DK (1) DK271377A (ro)
ES (1) ES459945A1 (ro)
FI (1) FI771902A (ro)
FR (1) FR2355848A1 (ro)
GB (1) GB1580935A (ro)
GR (1) GR70337B (ro)
IL (1) IL52143A0 (ro)
NL (1) NL7706742A (ro)
PL (1) PL106565B1 (ro)
PT (1) PT66661B (ro)
RO (1) RO71162A (ro)
SE (1) SE7707125L (ro)
YU (1) YU145577A (ro)
ZA (1) ZA772994B (ro)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4368198A (en) * 1976-03-03 1983-01-11 Sumitomo Chemical Company Limited Cephalosporins
US4302454A (en) * 1976-03-03 1981-11-24 Sumitomo Chemical Company, Limited Cephalosporins
CH641468A5 (de) * 1978-05-30 1984-02-29 Hoffmann La Roche Cephemderivate.
US4331666A (en) * 1979-05-11 1982-05-25 Farmitalia Carlo Erba S.P.A. 3-[(8-Carboxy-6-tetrazolo[1,5-b]pyridazinyl)-thiomethyl]-7-[2-(2-amino-4-thiazolyl)-2-methoxyimino-acetamido]-3-cephem-4-carboxylic acid
FR2701027B1 (fr) * 1993-02-01 1997-07-18 Warner Lambert Co Procede de synthese ameliore du 9-(beta-d-arabinofuranosyl)adenine 5'-phosphate.
US9061250B2 (en) 2009-06-26 2015-06-23 Bl Technologies, Inc. Non-braided, textile-reinforced hollow fiber membrane
US9643129B2 (en) 2011-12-22 2017-05-09 Bl Technologies, Inc. Non-braided, textile-reinforced hollow fiber membrane
PL408133A1 (pl) 2014-05-07 2015-11-09 Innowacyjne Techniki Energii Odnawialnych Spółka Z Ograniczoną Odpowiedzialnością System połączonych technologii wytwarzania i wykorzystania energii odnawialnej

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1479711A (en) * 1973-06-12 1977-07-13 Beecham Group Ltd Acylureido cephalosporins
FR2233067A1 (en) * 1973-06-12 1975-01-10 Beecham Group Ltd N-(thio)acyl carbamoyl-glycylamino-cephalosporin ic acids - as antibiotics esp. active against pseudomonas and gram neg. organisms producing cephalosporinase
DE2354219A1 (de) * 1973-10-30 1975-05-07 Bayer Ag Beta-lactam-antibiotica, ein verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel
GB1486349A (en) * 1974-11-28 1977-09-21 Bayer Ag Beta-lactam antibiotics process for their preparation and their use as medicaments

Also Published As

Publication number Publication date
AR213853A1 (es) 1979-03-30
PL106565B1 (pl) 1979-12-31
NL7706742A (nl) 1977-12-23
IL52143A0 (en) 1977-07-31
ES459945A1 (es) 1978-08-16
ZA772994B (en) 1978-12-27
RO71162A (ro) 1981-11-24
AU2542677A (en) 1978-11-30
FR2355848A1 (fr) 1978-01-20
YU145577A (en) 1982-10-31
JPS52156897A (en) 1977-12-27
DK271377A (da) 1977-12-22
PL199032A1 (pl) 1978-04-10
GR70337B (ro) 1982-09-20
PT66661A (en) 1977-07-01
GB1580935A (en) 1980-12-10
SE7707125L (sv) 1977-12-22
PT66661B (en) 1978-11-13
DE2727325A1 (de) 1977-12-29
FI771902A (ro) 1977-12-22
US4061861A (en) 1977-12-06
AU508432B2 (en) 1980-03-20
DD131174A5 (de) 1978-06-07
BE855966A (fr) 1977-12-21

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