CS196336B2 - Method of producing novel 3-substituted 1-/o-benzoylphenyl/-5-/tertiary aminomethyl/-1h-1,2,4,-triazoles - Google Patents

Method of producing novel 3-substituted 1-/o-benzoylphenyl/-5-/tertiary aminomethyl/-1h-1,2,4,-triazoles Download PDF

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Publication number
CS196336B2
CS196336B2 CS768097A CS809776A CS196336B2 CS 196336 B2 CS196336 B2 CS 196336B2 CS 768097 A CS768097 A CS 768097A CS 809776 A CS809776 A CS 809776A CS 196336 B2 CS196336 B2 CS 196336B2
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CS
Czechoslovakia
Prior art keywords
formula
carboxylic acid
acid
compounds
compound
Prior art date
Application number
CS768097A
Other languages
Czech (cs)
English (en)
Inventor
Roland Heckendorn
Rene Meier
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of CS196336B2 publication Critical patent/CS196336B2/cs

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/101,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CS768097A 1975-12-12 1976-12-10 Method of producing novel 3-substituted 1-/o-benzoylphenyl/-5-/tertiary aminomethyl/-1h-1,2,4,-triazoles CS196336B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH1614775A CH601267A5 (xx) 1975-12-12 1975-12-12

Publications (1)

Publication Number Publication Date
CS196336B2 true CS196336B2 (en) 1980-03-31

Family

ID=4414812

Family Applications (1)

Application Number Title Priority Date Filing Date
CS768097A CS196336B2 (en) 1975-12-12 1976-12-10 Method of producing novel 3-substituted 1-/o-benzoylphenyl/-5-/tertiary aminomethyl/-1h-1,2,4,-triazoles

Country Status (21)

Country Link
JP (1) JPS5273871A (xx)
AT (1) AT351022B (xx)
AU (1) AU510423B2 (xx)
BE (1) BE849266R (xx)
CA (1) CA1081236A (xx)
CH (1) CH601267A5 (xx)
CS (1) CS196336B2 (xx)
CY (1) CY1177A (xx)
DE (1) DE2655483A1 (xx)
DK (1) DK557676A (xx)
ES (4) ES454152A2 (xx)
FR (1) FR2361884A2 (xx)
GB (1) GB1563735A (xx)
HK (1) HK13183A (xx)
HU (1) HU171999B (xx)
IE (1) IE44688B1 (xx)
MY (1) MY8400090A (xx)
NL (1) NL7613786A (xx)
SE (1) SE431332B (xx)
SG (1) SG1783G (xx)
ZA (1) ZA767380B (xx)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3709898A (en) * 1971-02-09 1973-01-09 Upjohn Co Process for the production of triazolobenzodiazepines and intermediates
FR2285125A1 (fr) * 1974-09-17 1976-04-16 Takeda Chemical Industries Ltd Derives de 1,2,4-triazole

Also Published As

Publication number Publication date
FR2361884A2 (fr) 1978-03-17
FR2361884B2 (xx) 1979-10-05
AU510423B2 (en) 1980-06-26
AU2047076A (en) 1978-06-15
CA1081236A (en) 1980-07-08
GB1563735A (en) 1980-03-26
SE7613918L (sv) 1977-06-13
BE849266R (fr) 1977-06-10
DE2655483A1 (de) 1977-06-16
ZA767380B (en) 1977-11-30
IE44688L (en) 1977-06-12
ES454152A2 (es) 1978-03-16
HK13183A (en) 1983-04-22
SG1783G (en) 1983-09-16
CY1177A (en) 1983-06-10
SE431332B (sv) 1984-01-30
NL7613786A (nl) 1977-06-14
HU171999B (hu) 1978-05-28
JPS616825B2 (xx) 1986-03-01
CH601267A5 (xx) 1978-06-30
IE44688B1 (en) 1982-02-24
ATA914076A (de) 1978-12-15
ES454151A2 (es) 1978-04-01
MY8400090A (en) 1984-12-31
ES454150A2 (es) 1977-12-16
ES454153A2 (es) 1978-04-01
JPS5273871A (en) 1977-06-21
AT351022B (de) 1979-07-10
DK557676A (da) 1977-06-13

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