CR9870A - Dihydrogen phosphate salt of a prostaglandin d2 recptor antagonist - Google Patents

Dihydrogen phosphate salt of a prostaglandin d2 recptor antagonist

Info

Publication number
CR9870A
CR9870A CR9870A CR9870A CR9870A CR 9870 A CR9870 A CR 9870A CR 9870 A CR9870 A CR 9870A CR 9870 A CR9870 A CR 9870A CR 9870 A CR9870 A CR 9870A
Authority
CR
Costa Rica
Prior art keywords
prostaglandin
dihydrogen phosphate
phosphate salt
receiver antagonist
antagonist
Prior art date
Application number
CR9870A
Other languages
English (en)
Inventor
Beverly Langevin
Edwuard Orton
Daniel Sherer
Original Assignee
Aventis Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Inc filed Critical Aventis Pharma Inc
Publication of CR9870A publication Critical patent/CR9870A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/04—Antipruritics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/12—Ophthalmic agents for cataracts
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/14—Decongestants or antiallergics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Rheumatology (AREA)
  • Vascular Medicine (AREA)
  • Anesthesiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
CR9870A 2005-10-13 2008-04-07 Dihydrogen phosphate salt of a prostaglandin d2 recptor antagonist CR9870A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US72629005P 2005-10-13 2005-10-13

Publications (1)

Publication Number Publication Date
CR9870A true CR9870A (es) 2008-06-18

Family

ID=37963090

Family Applications (1)

Application Number Title Priority Date Filing Date
CR9870A CR9870A (es) 2005-10-13 2008-04-07 Dihydrogen phosphate salt of a prostaglandin d2 recptor antagonist

Country Status (36)

Country Link
US (1) US7642249B2 (es)
EP (1) EP1948620B1 (es)
JP (1) JP2009511591A (es)
KR (1) KR101365480B1 (es)
CN (1) CN101287714B (es)
AR (1) AR058085A1 (es)
AU (1) AU2006304187B2 (es)
BR (1) BRPI0617311A2 (es)
CA (1) CA2625563C (es)
CR (1) CR9870A (es)
DK (1) DK1948620T3 (es)
DO (2) DOP2006000220A (es)
EC (1) ECSP088362A (es)
ES (1) ES2409833T3 (es)
GT (1) GT200600457A (es)
HK (1) HK1125133A1 (es)
HN (1) HN2008000603A (es)
HR (1) HRP20130341T1 (es)
IL (1) IL190673A (es)
MA (1) MA30005B1 (es)
MY (1) MY145648A (es)
NI (1) NI200800116A (es)
NO (1) NO20082072L (es)
NZ (1) NZ567433A (es)
PE (1) PE20070791A1 (es)
PL (1) PL1948620T3 (es)
PT (1) PT1948620E (es)
RS (1) RS52799B (es)
RU (1) RU2419614C2 (es)
SI (1) SI1948620T1 (es)
TN (1) TNSN08131A1 (es)
TW (1) TW200728288A (es)
UA (1) UA93062C2 (es)
UY (1) UY29862A1 (es)
WO (1) WO2007047378A2 (es)
ZA (1) ZA200802586B (es)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GT200500284A (es) * 2004-10-15 2006-03-27 Aventis Pharma Inc Pirimidinas como antagonistas del receptor de prostaglandina d2
DOP2007000068A (es) * 2006-04-12 2007-10-31 Sanofi Aventis Us Llc Compuestos de amino-pirimidina 2,6-sustituidos-4-monosustituidos como antagonistas del receptor de prostaglandina d2
WO2007146838A2 (en) * 2006-06-09 2007-12-21 Icos Corporation Substituted phenyl acetic acids as dp-2 antagonists
ATE531699T1 (de) * 2007-06-29 2011-11-15 Sanofi Sa Verfahren zur herstellung von 2-(3-ä6-ä2-(2,4-
CN101952244B (zh) 2008-02-01 2014-11-05 潘米拉制药公司 前列腺素d2受体的n，n-二取代氨基烷基联苯拮抗剂
WO2009108720A2 (en) * 2008-02-25 2009-09-03 Amira Pharmaceuticals, Inc. Antagonists of prostaglandin d2 receptors
GB2463788B (en) * 2008-09-29 2010-12-15 Amira Pharmaceuticals Inc Heteroaryl antagonists of prostaglandin D2 receptors
WO2010039977A2 (en) 2008-10-01 2010-04-08 Amira Pharmaceuticals, Inc. Heteroaryl antagonists of prostaglandin d2 receptors
WO2010042652A2 (en) 2008-10-08 2010-04-15 Amira Pharmaceuticals, Inc. Heteroalkyl biphenyl antagonists of prostaglandin d2 receptors
US20100112606A1 (en) * 2008-10-17 2010-05-06 Michael Armstrong Measurement and analysis of leukotrienes
AR074776A1 (es) * 2008-12-18 2011-02-09 Sanofi Aventis Metodo para tratar la degeneracion macular; modulando el sistema inmunitario del paciente
JP2013500978A (ja) 2009-07-31 2013-01-10 パンミラ ファーマシューティカルズ，エルエルシー． Ｄｐ２受容体アンタゴニストの眼の医薬組成物
EP2462110A4 (en) 2009-08-05 2013-04-03 Panmira Pharmaceuticals Llc DP2 ANTAGONIST AND USES THEREOF
EP2590640A1 (en) 2010-07-08 2013-05-15 Ramot at Tel-Aviv University Ltd Use of fts and analogs to treat non-autoimmune-allergic and non-allergic inflammatory conditions
US8785467B2 (en) * 2010-09-30 2014-07-22 Merck Sharp & Dohme Corp. Alkoxy pyrimidine PDE10 inhibitors
WO2014066568A1 (en) 2012-10-24 2014-05-01 Winthrop-University Hospital Non-invasive biomarker to identify subjects at risk of preterm delivery
EP3256121B1 (en) 2015-02-13 2024-08-07 INSERM - Institut National de la Santé et de la Recherche Médicale Ptgdr-1 and/or ptgdr-2 antagonists for preventing and/or treating systemic lupus erythematosus
LT3302448T (lt) 2015-06-04 2024-02-12 Aurigene Oncology Limited Pakeisti heterociklilo dariniai kaip cdk inhibitoriai
KR20200109293A (ko) 2017-09-13 2020-09-22 프로제너티, 인크. 자간전증 바이오마커 및 관련된 시스템 및 방법
EP4070113A4 (en) 2019-12-04 2023-12-20 Biora Therapeutics, Inc. ASSESSMENT OF PREECAMPSIA USING FREE AND DISSOCIATE PLACENTAL GROWTH FACTOR ASSAYS

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2198867A1 (en) * 2001-12-07 2010-06-23 Vertex Pharmaceuticals, Inc. Pyrimidine-based compounds useful as GSK-3 inhibitors
KR100768609B1 (ko) * 2003-07-09 2007-10-18 에프. 호프만-라 로슈 아게 티오페닐아미노이미다졸린
GT200500284A (es) * 2004-10-15 2006-03-27 Aventis Pharma Inc Pirimidinas como antagonistas del receptor de prostaglandina d2

Also Published As

Publication number Publication date
NZ567433A (en) 2010-06-25
PT1948620E (pt) 2013-05-06
BRPI0617311A2 (pt) 2011-07-19
US7642249B2 (en) 2010-01-05
AR058085A1 (es) 2008-01-23
HK1125133A1 (en) 2009-07-31
RS52799B (en) 2013-10-31
MY145648A (en) 2012-03-15
SI1948620T1 (sl) 2013-05-31
PE20070791A1 (es) 2007-08-16
RU2008118491A (ru) 2009-11-20
UY29862A1 (es) 2007-05-31
US20080194600A1 (en) 2008-08-14
UA93062C2 (ru) 2011-01-10
AU2006304187A1 (en) 2007-04-26
HN2008000603A (es) 2010-11-03
JP2009511591A (ja) 2009-03-19
ES2409833T3 (es) 2013-06-28
IL190673A0 (en) 2008-11-03
ES2409833T8 (es) 2013-09-26
AU2006304187B2 (en) 2011-04-28
EP1948620A2 (en) 2008-07-30
CN101287714A (zh) 2008-10-15
DOP2006000220A (es) 2007-05-15
CN101287714B (zh) 2011-04-06
DK1948620T3 (da) 2013-06-24
CA2625563C (en) 2011-04-19
WO2007047378A3 (en) 2007-08-02
TW200728288A (en) 2007-08-01
CA2625563A1 (en) 2007-04-26
IL190673A (en) 2011-12-29
DOP2006000223A (es) 2007-05-15
ZA200802586B (en) 2009-09-30
TNSN08131A1 (en) 2009-07-14
NO20082072L (no) 2008-05-02
RU2419614C2 (ru) 2011-05-27
WO2007047378A2 (en) 2007-04-26
HRP20130341T1 (en) 2013-05-31
NI200800116A (es) 2011-12-15
MA30005B1 (fr) 2008-12-01
GT200600457A (es) 2007-04-27
PL1948620T3 (pl) 2013-08-30
KR20080057275A (ko) 2008-06-24
KR101365480B1 (ko) 2014-02-21
ECSP088362A (es) 2008-05-30
EP1948620B1 (en) 2013-03-20

Similar Documents

Publication Publication Date Title
CR9870A (es) Dihydrogen phosphate salt of a prostaglandin d2 recptor antagonist
DK1877562T3 (da) Stivelse med højt indhold af phosphat
CR10186A (es) Inhibidores de 11-beta-hsd1
ES2401192T8 (es) Deazapurinas útiles como inhibidores de janus cinasas
DE602004029953D1 (de) Schaltbare Antennenanordnung zur Abschätzung der Einfallsrichtung eines Empfangssignals
ATE449762T1 (de) Kristalline formen einer biphenylverbindung
MA28876B1 (fr) Amides bicycliques comme inhibiteurs de kinases
ATE520660T1 (de) Kristalline formen einer dimethylphenylverbindung
ATE479682T1 (de) Kristalline form einer chinolin-carboxamid- verbindung
BRPI0922880A2 (pt) compostos inibidores de quinase
BRPI0912132A2 (pt) Protease específica de prolina do penicillium chrysogenum
DE602006020758D1 (de) Längslenker einer aufhängung
BRPI0616731A2 (pt) derivados de isoquinolina como inibidores do igf-1r
PL1723157T5 (pl) Amorficzne postaci rizedronianu monosodowego
BRPI0718444A2 (pt) Inibidores de receptor de adp de plaqueta
DE602006003661D1 (de) Ampa-rezeptoren-verstärker
ITMI20061848A1 (it) Procedimento per la preparazione di composti feniltetrazolici
FI20050736A0 (fi) Reaaliaikaisen palvelun laatu
BRPI0621575A2 (pt) conjunto de peças de conexão para tubos cilindricos para brinquedos de montar em três dimensões
IL186499A0 (en) New crystalline atorvastatin hemicalcium salt polymorph form
ITMI20060716A1 (it) Dispositivo per la taratura di un trasmettitore di campo
DE602006008015D1 (de) Feste salzformen eines pyrrolsubstituierten 2-indolinons
MX2009002606A (es) Derivados de arginina con actividad antagonistica de np-1.
DE602005016615D1 (de) Kompensation der parasitären kopplung zwischen hf-ng
FR2938960B1 (fr) Procede de transmission d'une coordonnee geographique.

Legal Events

Date Code Title Description
FC Refusal