CR9327A - Procedimiento para la preparacion de compuestos benzoxazol sustituidos - Google Patents

Procedimiento para la preparacion de compuestos benzoxazol sustituidos

Info

Publication number
CR9327A
CR9327A CR9327A CR9327A CR9327A CR 9327 A CR9327 A CR 9327A CR 9327 A CR9327 A CR 9327A CR 9327 A CR9327 A CR 9327A CR 9327 A CR9327 A CR 9327A
Authority
CR
Costa Rica
Prior art keywords
preparation
procedure
compounds
substituted benzoxazol
substituted
Prior art date
Application number
CR9327A
Other languages
English (en)
Inventor
Iera Silvio
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36593680&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CR9327(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of CR9327A publication Critical patent/CR9327A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/56Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D263/57Aryl or substituted aryl radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/18Benzimidazoles; Hydrogenated benzimidazoles with aryl radicals directly attached in position 2
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62Benzothiazoles
    • C07D277/64Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2
    • C07D277/66Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2 with aromatic rings or ring systems directly attached in position 2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

La presente invencion se relaciona con procedimientos para la preparacion de compuestos benzoxazol sustituidos, y en particular 2-(3-fluoro-4-hidroxi-fenil)-7-vinil-benzoxazol-5-ol. Los procedimientos incluyen la vinilacion de un compuesto benzoxazol sustituido que tiene una porcion sustituible apropiada.
CR9327A 2005-03-07 2007-08-17 Procedimiento para la preparacion de compuestos benzoxazol sustituidos CR9327A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US65913805P 2005-03-07 2005-03-07

Publications (1)

Publication Number Publication Date
CR9327A true CR9327A (es) 2008-01-21

Family

ID=36593680

Family Applications (1)

Application Number Title Priority Date Filing Date
CR9327A CR9327A (es) 2005-03-07 2007-08-17 Procedimiento para la preparacion de compuestos benzoxazol sustituidos

Country Status (20)

Country Link
US (1) US20060199852A1 (es)
EP (1) EP1856069A1 (es)
JP (1) JP2008531747A (es)
KR (1) KR20070111514A (es)
CN (1) CN101137627A (es)
AR (1) AR052935A1 (es)
AU (1) AU2006220735A1 (es)
BR (1) BRPI0608891A2 (es)
CA (1) CA2601973A1 (es)
CR (1) CR9327A (es)
GT (1) GT200600102A (es)
IL (1) IL185335A0 (es)
MX (1) MX2007010894A (es)
NI (1) NI200700227A (es)
NO (1) NO20074259L (es)
PE (1) PE20061068A1 (es)
RU (1) RU2007131398A (es)
SG (1) SG160353A1 (es)
TW (1) TW200643018A (es)
WO (1) WO2006096584A1 (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101128443A (zh) * 2005-03-07 2008-02-20 惠氏公司 经取代的苯并唑化合物的纯化方法
US20080146630A1 (en) * 2006-11-21 2008-06-19 Wyeth Crystal form of 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol
US20080176914A1 (en) * 2006-11-21 2008-07-24 Wyeth Crystal form of 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol
US20080139633A1 (en) * 2006-11-21 2008-06-12 Wyeth Crystal form of 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol
US20080132554A1 (en) * 2006-11-21 2008-06-05 Wyeth Crystal form of 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol
CN111954729B (zh) * 2018-01-03 2023-05-23 埃科莱布美国股份有限公司 减少水中金属腐蚀的工艺和方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2002167350A (ja) * 2000-11-30 2002-06-11 Adchemco Corp 4−第三級ブトキシスチレンの製造方法
JP2002179621A (ja) * 2000-12-08 2002-06-26 Adchemco Corp 4−アセトキシスチレンの製造方法
UA83620C2 (ru) * 2001-12-05 2008-08-11 Уайт Замещенные бензоксазолы и их аналоги как эстрогенные агенты

Also Published As

Publication number Publication date
KR20070111514A (ko) 2007-11-21
SG160353A1 (en) 2010-04-29
NO20074259L (no) 2007-09-27
EP1856069A1 (en) 2007-11-21
CN101137627A (zh) 2008-03-05
PE20061068A1 (es) 2006-12-08
WO2006096584A1 (en) 2006-09-14
GT200600102A (es) 2006-10-25
IL185335A0 (en) 2008-02-09
AR052935A1 (es) 2007-04-11
CA2601973A1 (en) 2006-09-14
BRPI0608891A2 (pt) 2012-07-31
US20060199852A1 (en) 2006-09-07
AU2006220735A1 (en) 2006-09-14
NI200700227A (es) 2008-07-03
TW200643018A (en) 2006-12-16
RU2007131398A (ru) 2009-04-20
MX2007010894A (es) 2007-12-05
JP2008531747A (ja) 2008-08-14

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal (granting procedure)