CR8323A - DERIVATIVES OF TROPANO - Google Patents

DERIVATIVES OF TROPANO

Info

Publication number
CR8323A
CR8323A CR8323A CR8323A CR8323A CR 8323 A CR8323 A CR 8323A CR 8323 A CR8323 A CR 8323A CR 8323 A CR8323 A CR 8323A CR 8323 A CR8323 A CR 8323A
Authority
CR
Costa Rica
Prior art keywords
treatment
modular
conditions
inflammatory diseases
present
Prior art date
Application number
CR8323A
Other languages
Spanish (es)
Inventor
Anthony Stupple Paul
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB0323236.0A external-priority patent/GB0323236D0/en
Priority claimed from GB0325020A external-priority patent/GB0325020D0/en
Priority claimed from GB0418556A external-priority patent/GB0418556D0/en
Application filed by Pfizer filed Critical Pfizer
Publication of CR8323A publication Critical patent/CR8323A/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente invencion proporciona compuestos de formula ( I ) en la que R1 y R2 son como se definen anteriormente en la presente memoria. Los compuestos de la presente invencion son modulares, especialmente antagonistas, de la actividad de receptores CCR5 de quimioquinas. Los modulares de receptor CCR5 pueden ser utiles en el tratamiento de diversas enfermedades y afecciones inflamatorias y en el tratamiento de diversas enfermedades y afecciones inflamatorias y en el tratamiento de infeccion por VIH y retrovirus geneticamente relacionados.The present invention provides compounds of formula (I) in which R1 and R2 are as defined hereinbefore. The compounds of the present invention are modular, especially antagonists, of the activity of CCR5 chemokine receptors. The CCR5 receptor modular can be useful in the treatment of various inflammatory diseases and conditions and in the treatment of various inflammatory diseases and conditions and in the treatment of HIV infection and genetically related retroviruses.

CR8323A 2003-10-03 2006-04-03 DERIVATIVES OF TROPANO CR8323A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0323236.0A GB0323236D0 (en) 2003-10-03 2003-10-03 Chemical compounds
GB0325020A GB0325020D0 (en) 2003-10-27 2003-10-27 Chemical compounds
GB0418556A GB0418556D0 (en) 2004-08-19 2004-08-19 The treatment of pain

Publications (1)

Publication Number Publication Date
CR8323A true CR8323A (en) 2007-12-04

Family

ID=44839334

Family Applications (1)

Application Number Title Priority Date Filing Date
CR8323A CR8323A (en) 2003-10-03 2006-04-03 DERIVATIVES OF TROPANO

Country Status (1)

Country Link
CR (1) CR8323A (en)

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