CU23522B7 - IMIDAZOPIRIDINE TROPAN DERIVATIVES REPLACED WITH CCR5 RECEIVER ANTAGONIST ACTIVITY FOR THE TREATMENT OF HIV AND INFLAMMATION - Google Patents

IMIDAZOPIRIDINE TROPAN DERIVATIVES REPLACED WITH CCR5 RECEIVER ANTAGONIST ACTIVITY FOR THE TREATMENT OF HIV AND INFLAMMATION

Info

Publication number
CU23522B7
CU23522B7 CU20060067A CU20060067A CU23522B7 CU 23522 B7 CU23522 B7 CU 23522B7 CU 20060067 A CU20060067 A CU 20060067A CU 20060067 A CU20060067 A CU 20060067A CU 23522 B7 CU23522 B7 CU 23522B7
Authority
CU
Cuba
Prior art keywords
treatment
hiv
imidazopiridine
inflammation
antagonist activity
Prior art date
Application number
CU20060067A
Other languages
Spanish (es)
Inventor
Paul Anthony Stupple
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Priority to CU20060067A priority Critical patent/CU23522B7/en
Publication of CU23522B7 publication Critical patent/CU23522B7/en

Links

Abstract

La presente invención proporciona compuestos de fómula (I) ESPACIO PARA FORMULA en la que R1 y R2 son como se definen anteriormente en la presente memoria. Los compuestos de la presente invención son moduladores, especialmente antagonistas, de la actividad de receptores CCR5 de quimioquinas. Los moduladores de receptor CCR5 pueden ser útiles en el tratamiento de diversas enfermedades y afecciones inflamatorias y en el tratamiento de infección por VIH y retrovirus genéticamente relacionados.The present invention provides compounds of formula (I) SPACE FOR FORMULA in which R1 and R2 are as defined hereinbefore. The compounds of the present invention are modulators, especially antagonists, of the activity of chemokine CCR5 receptors. CCR5 receptor modulators can be useful in the treatment of various inflammatory diseases and conditions and in the treatment of HIV infection and genetically related retroviruses.

CU20060067A 2006-03-22 2006-03-22 IMIDAZOPIRIDINE TROPAN DERIVATIVES REPLACED WITH CCR5 RECEIVER ANTAGONIST ACTIVITY FOR THE TREATMENT OF HIV AND INFLAMMATION CU23522B7 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CU20060067A CU23522B7 (en) 2006-03-22 2006-03-22 IMIDAZOPIRIDINE TROPAN DERIVATIVES REPLACED WITH CCR5 RECEIVER ANTAGONIST ACTIVITY FOR THE TREATMENT OF HIV AND INFLAMMATION

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CU20060067A CU23522B7 (en) 2006-03-22 2006-03-22 IMIDAZOPIRIDINE TROPAN DERIVATIVES REPLACED WITH CCR5 RECEIVER ANTAGONIST ACTIVITY FOR THE TREATMENT OF HIV AND INFLAMMATION

Publications (1)

Publication Number Publication Date
CU23522B7 true CU23522B7 (en) 2010-05-19

Family

ID=42633306

Family Applications (1)

Application Number Title Priority Date Filing Date
CU20060067A CU23522B7 (en) 2006-03-22 2006-03-22 IMIDAZOPIRIDINE TROPAN DERIVATIVES REPLACED WITH CCR5 RECEIVER ANTAGONIST ACTIVITY FOR THE TREATMENT OF HIV AND INFLAMMATION

Country Status (1)

Country Link
CU (1) CU23522B7 (en)

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Legal Events

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FG Grant of patent
FD Lapse (for not paying fees)