CR20190527A - Parche que contiene rupatadina - Google Patents

Parche que contiene rupatadina

Info

Publication number
CR20190527A
CR20190527A CR20190527A CR20190527A CR20190527A CR 20190527 A CR20190527 A CR 20190527A CR 20190527 A CR20190527 A CR 20190527A CR 20190527 A CR20190527 A CR 20190527A CR 20190527 A CR20190527 A CR 20190527A
Authority
CR
Costa Rica
Prior art keywords
rupatadine
external patch
adhesive
acrylic adhesive
patch containing
Prior art date
Application number
CR20190527A
Other languages
English (en)
Inventor
Satoshi Kawakami
Manabu Sogabe
Original Assignee
J Uriach Y Compania S A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by J Uriach Y Compania S A filed Critical J Uriach Y Compania S A
Publication of CR20190527A publication Critical patent/CR20190527A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
    • A61K9/7061—Polyacrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12—Carboxylic acids; Salts or anhydrides thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14—Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/44—Oils, fats or waxes according to two or more groups of A61K47/02-A61K47/42; Natural or modified natural oils, fats or waxes, e.g. castor oil, polyethoxylated castor oil, montan wax, lignite, shellac, rosin, beeswax or lanolin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/04—Antipruritics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Dermatology (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Otolaryngology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Adhesives Or Adhesive Processes (AREA)

Abstract

Se proporciona un parche externo que contiene rupatadina como antihistamina de segunda generación, tiene excelentes propiedades físicas de esparadrapo, buena adhesión cuando se aplica a la piel, y buena absorción transdérmica de rupatadina como principio activo. El parche externo que contiene rupatadina usa un adhesivo acrílico como base adhesiva. Específicamente, el parche externo que contiene rupatadina usa un adhesivo acrílico como base adhesiva y además contiene un ácido orgánico que tiene de 2 a 7 átomos de carbono como agente de solubilidad, un éster de ácido graso como agente de reblandecimiento y/o un tensioactivo.
CR20190527A 2017-04-19 2018-04-18 Parche que contiene rupatadina CR20190527A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2017082559 2017-04-19
PCT/JP2018/016692 WO2018194183A1 (en) 2017-04-19 2018-04-18 Rupatadine-containing patch

Publications (1)

Publication Number Publication Date
CR20190527A true CR20190527A (es) 2020-03-17

Family

ID=63856668

Family Applications (1)

Application Number Title Priority Date Filing Date
CR20190527A CR20190527A (es) 2017-04-19 2018-04-18 Parche que contiene rupatadina

Country Status (15)

Country Link
US (1) US11179346B2 (es)
EP (1) EP3612182B1 (es)
JP (1) JP7228527B2 (es)
KR (1) KR102586423B1 (es)
CN (1) CN110740730B (es)
BR (1) BR112019021807A2 (es)
CA (1) CA3059682A1 (es)
CR (1) CR20190527A (es)
DO (1) DOP2019000270A (es)
ES (1) ES2971461T3 (es)
FI (1) FI3612182T3 (es)
NI (1) NI201900109A (es)
PL (1) PL3612182T3 (es)
TW (1) TWI825013B (es)
WO (1) WO2018194183A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4238563A1 (en) * 2020-10-29 2023-09-06 Hisamitsu Pharmaceutical Co., Inc. Ropinirole-containing patch and method for improving skin permeability of ropinirole
CN112494429B (zh) * 2020-12-29 2022-07-26 北京华氏开元医药科技有限公司 一种富马酸卢帕他定纳米乳液及其制备方法与应用

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2042421B1 (es) 1992-05-22 1994-08-01 Uriach & Cia Sa J Procedimiento para la obtencion de la 8-cloro-11-*1-*(5-metil-3-piridil)metil*-4-piperidiliden*-6,11-dihidro-5h-benzo*5,6*ciclohepta*1,2-b*piridina.
US9259397B2 (en) * 2000-10-23 2016-02-16 Purdue Pharma L.P. Loratadine transdermal device and methods
DE10060852A1 (de) * 2000-12-06 2002-06-20 Hexal Ag Absorptionsmittel und Kanalbildner enthaltende wirkstoffundurchlässige Deckschicht oder abziehbare Schutzschicht eines transdermalen therapeutischen Systems
CN100411692C (zh) * 2004-01-13 2008-08-20 北京康倍得医药技术开发有限公司 丙烯酸基粘合剂组合物及其药物组合物和透皮治疗系统
WO2007007863A1 (en) * 2005-07-08 2007-01-18 Senju Pharmaceutical Co., Ltd. Percutaneously absorptive ophthalmic preparation comprising olopatadine
EP2008651A1 (en) 2007-06-26 2008-12-31 Drug Delivery Solutions Limited A bioerodible patch
CN101933914A (zh) * 2009-06-29 2011-01-05 杭州赛利药物研究所有限公司 地氯雷他定贴剂及其制备方法
JP5837276B2 (ja) * 2009-09-30 2015-12-24 味の素株式会社 経口摂取用ゲル状組成物、及びその製造方法
CN102958926B (zh) 2010-06-30 2014-04-23 J·乌里亚奇·Y股份有限公司 抗组胺剂
US9566306B2 (en) * 2012-04-16 2017-02-14 Zemtsov Enterprises, Llc Formulations and methods for treatment of wounds and inflammatory skin conditions

Also Published As

Publication number Publication date
RU2019136691A3 (es) 2021-07-13
EP3612182A1 (en) 2020-02-26
EP3612182A4 (en) 2020-09-16
CN110740730A (zh) 2020-01-31
US20200121612A1 (en) 2020-04-23
KR20200006065A (ko) 2020-01-17
BR112019021807A2 (pt) 2020-05-05
FI3612182T3 (fi) 2024-02-19
JP7228527B2 (ja) 2023-02-24
EP3612182B1 (en) 2024-01-10
NI201900109A (es) 2020-01-07
TWI825013B (zh) 2023-12-11
KR102586423B1 (ko) 2023-10-11
ES2971461T3 (es) 2024-06-05
CA3059682A1 (en) 2018-10-25
JP2020524657A (ja) 2020-08-20
CN110740730B (zh) 2024-01-09
RU2019136691A (ru) 2021-05-17
TW201841638A (zh) 2018-12-01
PL3612182T3 (pl) 2024-05-13
DOP2019000270A (es) 2019-12-30
US11179346B2 (en) 2021-11-23
WO2018194183A1 (en) 2018-10-25

Similar Documents

Publication Publication Date Title
MX2017000102A (es) Calzado que tiene estructuras augeticas con propiedades controladas.
MX2016007075A (es) Formulacion adhesiva y metodos de plisado utilizando la misma.
DOP2016000339A (es) Compuestos de heteroarilo útiles como inhibidores de enzima activadora de sumo
GB2550301A (en) Antimicrobial fibers and compositions
PE20151778A1 (es) Formulacion combinada de dos compuestos antivirales
BR112016025331A2 (pt) composições antimicrobianas
MX2017009144A (es) Dimeros de benzodiazepina unidos con puentes de heteroarileno, conjugados de estos, y sus metodos de preparacion y uso.
MX366560B (es) Parche adhesivo con composicion antimicrobiana.
CL2018000070A1 (es) Modulares de diaciglicerol aciltransderasa 2 (dgta2)
MX2014011710A (es) Composiciones antimicrobianas ambientalmente preferidas.
AR084032A1 (es) Compuesto biciclico
EA201290928A1 (ru) Содержащая протеогликан совокупность микроигл
PE20150024A1 (es) Compuestos que inhiben la actividad de catecol o-metiltransferasa
MX2018009277A (es) Articulo absorbente con elemento de proteccion trasero plano.
MY181540A (en) Transdermal composition containing donepezil as active ingredient
MX2019013561A (es) Compuestos de pirrolopiridina-anilina para el tratamiento de trastornos dermicos.
NZ611920A (en) Percutaneous absorption preparation containing rivastigmine
GEP20196969B (en) New therapeutical composition containing apomorphine as active ingredient
BR112017013255A2 (pt) emplastro em gel
CR20190527A (es) Parche que contiene rupatadina
PE20170898A1 (es) Inhibidor de cinasa aurora a
BR112012015084A2 (pt) composição farmacêutica de liberação lenta de iloperidone
BR112014011066A2 (pt) artigo absorvente com elemento de estabilização
AU2016204294A1 (en) Solid State Forms Of A Quinazoline Derivative And Its Use As A BRAF Inhibitor
PE20141035A1 (es) Composiciones y metodos para tratar el cancer usando el inhibidor de pi3kbeta y el inhibidor de la via de mapk, incluidos los inhibidores de mek y raf