CR20120395A - Uso farmacéutico de compuestos multicíclicos como agentes anti-síndrome de inmunodeficiencia adquirida - Google Patents

Uso farmacéutico de compuestos multicíclicos como agentes anti-síndrome de inmunodeficiencia adquirida

Info

Publication number
CR20120395A
CR20120395A CR20120395A CR20120395A CR20120395A CR 20120395 A CR20120395 A CR 20120395A CR 20120395 A CR20120395 A CR 20120395A CR 20120395 A CR20120395 A CR 20120395A CR 20120395 A CR20120395 A CR 20120395A
Authority
CR
Costa Rica
Prior art keywords
multicycle
immunodeficiency
acquired
compounds
pharmaceutical use
Prior art date
Application number
CR20120395A
Other languages
English (en)
Inventor
Joao Batista Calixto
Claudio Paulino Chaves
Luiz Francisco Pianowski
Original Assignee
Amazonia Fitomedicamentos Ltda
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Amazonia Fitomedicamentos Ltda filed Critical Amazonia Fitomedicamentos Ltda
Publication of CR20120395A publication Critical patent/CR20120395A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • A61K31/23Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin of acids having a carboxyl group bound to a chain of seven or more carbon atoms
    • A61K31/232Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin of acids having a carboxyl group bound to a chain of seven or more carbon atoms having three or more double bonds, e.g. etretinate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/575Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/47Euphorbiaceae (Spurge family), e.g. Ricinus (castorbean)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Natural Medicines & Medicinal Plants (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Emergency Medicine (AREA)
  • Botany (AREA)
  • Medical Informatics (AREA)
  • Biotechnology (AREA)
  • Alternative & Traditional Medicine (AREA)
  • Microbiology (AREA)
  • Mycology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Virology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Molecular Biology (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
CR20120395A 2010-01-15 2012-07-24 Uso farmacéutico de compuestos multicíclicos como agentes anti-síndrome de inmunodeficiencia adquirida CR20120395A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/IB2010/050198 WO2011086423A1 (en) 2010-01-15 2010-01-15 Pharmaceutical use of multicyclic compounds as anti-aids agents

Publications (1)

Publication Number Publication Date
CR20120395A true CR20120395A (es) 2012-08-30

Family

ID=42735537

Family Applications (1)

Application Number Title Priority Date Filing Date
CR20120395A CR20120395A (es) 2010-01-15 2012-07-24 Uso farmacéutico de compuestos multicíclicos como agentes anti-síndrome de inmunodeficiencia adquirida

Country Status (13)

Country Link
US (1) US20120289487A1 (es)
EP (1) EP2523663A1 (es)
JP (1) JP2013517262A (es)
KR (1) KR20120112707A (es)
CN (1) CN102711750A (es)
AU (1) AU2010342326A1 (es)
BR (1) BR112012017211A2 (es)
CA (1) CA2787236A1 (es)
CR (1) CR20120395A (es)
MX (1) MX2012008253A (es)
RU (1) RU2012134786A (es)
SG (1) SG182413A1 (es)
WO (1) WO2011086423A1 (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2013225633B2 (en) * 2012-03-02 2017-11-23 Amazonia Fitomedicamentos Ltda. Ingenol derivatives in the reactivation of latent HIV
CN108524448B (zh) * 2017-03-02 2019-10-18 新疆维吾尔自治区药物研究所 一种大戟二烯醇抗白内障眼用制剂及其制备方法和用途
CN109021051A (zh) * 2017-06-12 2018-12-18 盛世泰科生物医药技术(苏州)有限公司 四环三萜类化合物的晶型及其用途
CN109912419A (zh) * 2017-12-13 2019-06-21 复旦大学 巨大戟烷型二萜及其在制备抗艾滋病毒药物中的用途

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006007676A1 (en) * 2004-07-21 2006-01-26 Amazônia Fitomedicamentos Ltda. Combination of active fractions from the plants euphorbia tirucalli l and ficos carica l. and method of treating cancer and aids
US20090142421A1 (en) 2005-06-28 2009-06-04 Amazonia Fitomedicamentos Ltda. Active fraction of a polar solvent extract from the latex of euphorbiaceae plants

Also Published As

Publication number Publication date
JP2013517262A (ja) 2013-05-16
MX2012008253A (es) 2012-08-15
AU2010342326A1 (en) 2012-08-09
US20120289487A1 (en) 2012-11-15
SG182413A1 (en) 2012-08-30
CN102711750A (zh) 2012-10-03
RU2012134786A (ru) 2014-02-20
CA2787236A1 (en) 2011-07-21
BR112012017211A2 (pt) 2019-09-24
KR20120112707A (ko) 2012-10-11
EP2523663A1 (en) 2012-11-21
WO2011086423A1 (en) 2011-07-21

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