CO6270213A2 - Composiciones farmaceuticas que comprenden acido montelukast y un unhibidor depde-4 o un corticoesteroide inhalado para administracion por inhalacion - Google Patents

Composiciones farmaceuticas que comprenden acido montelukast y un unhibidor depde-4 o un corticoesteroide inhalado para administracion por inhalacion

Info

Publication number
CO6270213A2
CO6270213A2 CO10047531A CO10047531A CO6270213A2 CO 6270213 A2 CO6270213 A2 CO 6270213A2 CO 10047531 A CO10047531 A CO 10047531A CO 10047531 A CO10047531 A CO 10047531A CO 6270213 A2 CO6270213 A2 CO 6270213A2
Authority
CO
Colombia
Prior art keywords
preparation
inhaled
unhibitor
depde
corticoesteroid
Prior art date
Application number
CO10047531A
Other languages
English (en)
Inventor
Roch Thibert
Original Assignee
Merck Frosst Canada Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Frosst Canada Ltd filed Critical Merck Frosst Canada Ltd
Publication of CO6270213A2 publication Critical patent/CO6270213A2/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

1.- Una preparacion medicinal que comprende acido montelukast y un segundo agente activo seleccionado de un inhibidor de PDE-4 y un corticoesteroide inhalado como una preparacion combinada para la administracion por inhalacion. 2.- Una preparacion de la Reivindicacion 1 en la que dicho segundo agente activo es un Compuesto X que tiene la formula:3.- Una preparacion de la Reivindicacion 1 en la que dicho segundo agente activo es mometasona furoato. 4.- Una preparacion de la Reivindicacion 1 adaptada para usar en un inhalador de polvo seco o un inhalador de dosis medida.5.- Una preparacion de la Reivindicacion 2 adaptada para usar en un inhalador de polvo seco o en un inhalador de dosis medida. 6.- Una preparacion de la Reivindicacion 3 adaptada para usar en un inhalador de polvo seco o en un inhalador de dosis medida. 7.- Un inhalador de polvo seco que contiene la preparacion medicinal de la Reivindicacion 1. 8.- Un inhalador de dosis medida que contiene la preparacion medicinal de la Reivindicacion 1.
CO10047531A 2007-10-25 2010-04-22 Composiciones farmaceuticas que comprenden acido montelukast y un unhibidor depde-4 o un corticoesteroide inhalado para administracion por inhalacion CO6270213A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US32707P 2007-10-25 2007-10-25

Publications (1)

Publication Number Publication Date
CO6270213A2 true CO6270213A2 (es) 2011-04-20

Family

ID=40579006

Family Applications (1)

Application Number Title Priority Date Filing Date
CO10047531A CO6270213A2 (es) 2007-10-25 2010-04-22 Composiciones farmaceuticas que comprenden acido montelukast y un unhibidor depde-4 o un corticoesteroide inhalado para administracion por inhalacion

Country Status (19)

Country Link
US (1) US20100210611A1 (es)
EP (1) EP2211863A4 (es)
JP (1) JP2011500731A (es)
KR (1) KR20100072295A (es)
CN (1) CN101909626A (es)
AU (1) AU2008316283A1 (es)
CA (1) CA2701956A1 (es)
CO (1) CO6270213A2 (es)
CR (1) CR11439A (es)
DO (1) DOP2010000122A (es)
GT (1) GT201000107A (es)
IL (1) IL205182A0 (es)
MA (1) MA33705B1 (es)
MX (1) MX2010004529A (es)
NI (1) NI201000069A (es)
NZ (1) NZ584876A (es)
RU (1) RU2470639C2 (es)
WO (1) WO2009052624A1 (es)
ZA (1) ZA201002562B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2012168907A1 (en) 2011-06-10 2012-12-13 Glenmark Pharmaceuticals Sa Pharmaceutical composition comprising revamilast and montelukast or zafirlukast
WO2014012954A1 (en) 2012-07-18 2014-01-23 Takeda Gmbh Treatment of partly controlled or uncontrolled severe asthma
WO2015110394A1 (en) 2014-01-22 2015-07-30 Takeda Gmbh Treatment of partly controlled or uncontrolled severe asthma with a pde4 inhibitor (and in combination with a leukotriene modifier)
CN108267531B (zh) * 2016-12-31 2022-01-11 天津金耀集团有限公司 一种环索奈德有关物质hplc测定方法
IT201900014178A1 (it) * 2019-08-06 2021-02-06 Genetic S P A Esteri del montelukast e loro formulazioni farmaceutiche

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5837699A (en) * 1994-01-27 1998-11-17 Schering Corporation Use of mometasone furoate for treating upper airway passage diseases
US20040214805A1 (en) * 1999-11-02 2004-10-28 Smithkline Beecham Corporation Method and compositions for treating pulmonary diseases
AU2002227123A1 (en) * 2000-11-07 2002-05-21 Merck And Co., Inc. Method of treatment with a combination of a pde4 inhibitor and a leukotriene antagonist
JO2311B1 (en) * 2001-08-29 2005-09-12 ميرك فروست كندا ليمتد Alkyl inhibitors Ariel phosphodiesterase-4
US20050014762A1 (en) * 2001-09-19 2005-01-20 Rolf Beume Combination
DE10237739A1 (de) * 2002-08-17 2004-02-26 Boehringer Ingelheim Pharma Gmbh & Co. Kg Inhalative Arzneimittel enthaltend ein neues Anticholinergikum in Kombination mit Corticosteroiden und Betamimetika
US7550133B2 (en) * 2002-11-26 2009-06-23 Alexza Pharmaceuticals, Inc. Respiratory drug condensation aerosols and methods of making and using them
PL1670482T5 (pl) * 2003-09-16 2022-10-03 Covis Pharma Gmbh Zastosowanie cyklezonidu w leczeniu chorób układu oddechowego
EP1678139B1 (en) * 2003-10-10 2011-08-31 Synhton B.V. Solid-state montelukast
JP4700014B2 (ja) * 2004-02-06 2011-06-15 メダ ファーマ ゲゼルシャフト ミット ベシュレンクテル ハフツング ウント コンパニー コマンディト ゲゼルシャフト 呼吸器系疾患の治療用の抗コリン作用薬及び4型ホスホジエステラーゼの組合せ剤
EP1616567A1 (en) * 2004-07-16 2006-01-18 Boehringer Ingelheim Pharma GmbH & Co.KG Medicaments for inhalation comprising PDE IV inhibitors and glycopyrrolate salts
CA2601179A1 (en) * 2005-03-16 2006-09-21 Elan Pharma International Limited Nanoparticulate leukotriene receptor antagonist/corticosteroid formulations
CA2595791C (en) * 2005-03-16 2013-10-08 Meda Pharma Gmbh & Co. Kg The combination of anticholinergics and leukotriene receptor antagonists for the treatment of respiratory diseases
JP2009509980A (ja) * 2005-09-28 2009-03-12 メルク フロスト カナダ リミテツド 篩分けされたラクトースを含むエアゾール粉末製剤

Also Published As

Publication number Publication date
NZ584876A (en) 2012-06-29
RU2470639C2 (ru) 2012-12-27
MA33705B1 (fr) 2012-11-01
CN101909626A (zh) 2010-12-08
AU2008316283A1 (en) 2009-04-30
US20100210611A1 (en) 2010-08-19
CR11439A (es) 2010-06-21
JP2011500731A (ja) 2011-01-06
KR20100072295A (ko) 2010-06-30
RU2010120806A (ru) 2011-11-27
GT201000107A (es) 2012-03-13
EP2211863A1 (en) 2010-08-04
NI201000069A (es) 2010-08-23
WO2009052624A9 (en) 2010-11-25
DOP2010000122A (es) 2010-07-15
EP2211863A4 (en) 2012-07-25
CA2701956A1 (en) 2009-04-30
ZA201002562B (en) 2011-06-29
WO2009052624A1 (en) 2009-04-30
MX2010004529A (es) 2010-05-10
IL205182A0 (en) 2010-11-30

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