CO6150168A2 - Combinaciones farmacologicas que comprenden benzoxazinonas para el tratamiento de enfermedades de las vias aereas - Google Patents

Combinaciones farmacologicas que comprenden benzoxazinonas para el tratamiento de enfermedades de las vias aereas

Info

Publication number
CO6150168A2
CO6150168A2 CO09016427A CO09016427A CO6150168A2 CO 6150168 A2 CO6150168 A2 CO 6150168A2 CO 09016427 A CO09016427 A CO 09016427A CO 09016427 A CO09016427 A CO 09016427A CO 6150168 A2 CO6150168 A2 CO 6150168A2
Authority
CO
Colombia
Prior art keywords
compounds
pharmacological combinations
pharmacological
benzoxazinonas
treatment
Prior art date
Application number
CO09016427A
Other languages
English (en)
Inventor
Ingo Konetzki
Thierry Bouyssou
Sabine Pestel
Andreas Schnapp
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of CO6150168A2 publication Critical patent/CO6150168A2/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/536Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with carbocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/06Antiabortive agents; Labour repressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/04Antipruritics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Cardiology (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pregnancy & Childbirth (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Hospice & Palliative Care (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

1.- Combinaciones farmacológicas que, además de uno o varios compuestos de la fórmula general 1en donde R1 y R2 son, de modo independiente entre sí, H, halógeno o alquilo C1-4 o juntos son alquileno C1-6; y R3 es H, halógeno, OH, alquilo C1-4 u O-alquilo C1-4, contienen al menos otro principio activo 2. 2.- Combinaciones farmacológicas de acuerdo con la reivindicación 1 que, además de uno o varios compuestos de la fórmula 1 contienen como otro principio activo 2 uno o varios compuestos que están seleccionados de las clases de los anticolinérgicos (2a), inhibidores de PDE IV (2b), esteroides (2c), antagonistas de LTD4 (2d) e inhibidores de EGFR (2e). 3.- Combinaciones farmacológicas de acuerdo con la reivindicación 1 ó 2, que contienen uno o varios compuestos de la fórmula general 1, en donde R1 y R2 iguales o diferentes, hidrógeno, flúor, cloro, metilo, etilo, propilo, butilo o conjuntamente -CH2-CH2-, -CH2-CH2-CH2-, -CH2-CH2-CH2-CH2- o -CH2-CH2-CH2-CH2-CH2-; hidrógeno, flúor, cloro, OH, metilo, etilo, metoxi o etoxi. 4.- Combinaciones farmacológicas de acuerdo con la reivindicación 1, 2 ó 3, que contienen uno o varios compuestos de la fórmula general 1, en donde R1 y R2 iguales o diferentes, etilo, propilo o conjuntamente -CH2-CH2-, -CH2-CH2-CH2-, -CH2-CH2-CH2-CH2- o -CH2-CH2-CH2-CH2-CH2-; R3 hidrógeno, flúor, OH, metilo o metoxi.
CO09016427A 2006-08-22 2009-02-19 Combinaciones farmacologicas que comprenden benzoxazinonas para el tratamiento de enfermedades de las vias aereas CO6150168A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP06119272 2006-08-22

Publications (1)

Publication Number Publication Date
CO6150168A2 true CO6150168A2 (es) 2010-04-20

Family

ID=38535607

Family Applications (1)

Application Number Title Priority Date Filing Date
CO09016427A CO6150168A2 (es) 2006-08-22 2009-02-19 Combinaciones farmacologicas que comprenden benzoxazinonas para el tratamiento de enfermedades de las vias aereas

Country Status (20)

Country Link
US (1) US20080051392A1 (es)
EP (1) EP2094271A2 (es)
JP (1) JP2010501521A (es)
KR (1) KR20090047539A (es)
CN (1) CN101505757A (es)
AR (1) AR062475A1 (es)
AU (1) AU2007287536A1 (es)
BR (1) BRPI0715855A2 (es)
CA (1) CA2661496A1 (es)
CO (1) CO6150168A2 (es)
EA (1) EA200900269A1 (es)
EC (1) ECSP099080A (es)
IL (1) IL197125A0 (es)
MX (1) MX2009001355A (es)
NO (1) NO20090067L (es)
PE (1) PE20081358A1 (es)
TW (1) TW200817009A (es)
UY (1) UY30552A1 (es)
WO (1) WO2008023003A1 (es)
ZA (1) ZA200810828B (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102005008921A1 (de) * 2005-02-24 2006-08-31 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Arzneimittel zur Behandlung von Atemwegserkrankungen
US7423146B2 (en) * 2005-11-09 2008-09-09 Boehringer Ingelheim International Gmbh Process for the manufacturing of pharmaceutically active 3,1-benzoxazine-2-ones
PE20080610A1 (es) * 2006-08-22 2008-07-15 Boehringer Ingelheim Int Nuevos beta-agonistas enantiomericamente puros, procedimientos para su preparacion y uso como medicamentos
EP2093219A1 (de) 2008-02-22 2009-08-26 Boehringer Ingelheim International Gmbh Kristalline, enantiomerenreine Salzform eines Betamimetikums und dessen Verwendung als Arzneimittel
WO2011061527A1 (en) 2009-11-17 2011-05-26 Astrazeneca Ab Combinations comprising a glucocorticoid receptor modulator for the treatment of respiratory diseases
GB201016912D0 (en) 2010-10-07 2010-11-24 Astrazeneca Ab Novel combination

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3026534A1 (de) * 1980-07-12 1982-03-18 C.H. Boehringer Sohn, 6507 Ingelheim 3,1-benzoxazin-2-one, ihre herstellung und verwendung
US4570630A (en) * 1983-08-03 1986-02-18 Miles Laboratories, Inc. Medicament inhalation device
US4811731A (en) * 1985-07-30 1989-03-14 Glaxo Group Limited Devices for administering medicaments to patients
WO2005013993A1 (en) * 2003-07-29 2005-02-17 Boehringer Ingelheim International Gmbh Medicaments comprising pde iv inhibitors and an anticholinergic for treating respiratory disorders
DE102004048390A1 (de) * 2004-10-01 2006-04-06 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Pulverinhalativa auf Basis modifizierter Laktosemischungen als Hilfsstoff
DE102005008921A1 (de) * 2005-02-24 2006-08-31 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Arzneimittel zur Behandlung von Atemwegserkrankungen
US7423146B2 (en) * 2005-11-09 2008-09-09 Boehringer Ingelheim International Gmbh Process for the manufacturing of pharmaceutically active 3,1-benzoxazine-2-ones

Also Published As

Publication number Publication date
AR062475A1 (es) 2008-11-12
IL197125A0 (en) 2009-11-18
CA2661496A1 (en) 2008-02-28
MX2009001355A (es) 2009-02-13
ECSP099080A (es) 2009-02-27
TW200817009A (en) 2008-04-16
EP2094271A2 (de) 2009-09-02
JP2010501521A (ja) 2010-01-21
PE20081358A1 (es) 2008-10-31
BRPI0715855A2 (pt) 2013-07-30
KR20090047539A (ko) 2009-05-12
WO2008023003A8 (de) 2008-05-22
AU2007287536A1 (en) 2008-02-28
CN101505757A (zh) 2009-08-12
UY30552A1 (es) 2008-03-31
US20080051392A1 (en) 2008-02-28
EA200900269A1 (ru) 2009-08-28
ZA200810828B (en) 2009-11-25
WO2008023003A1 (de) 2008-02-28
NO20090067L (no) 2009-03-17

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