CO5700713A2 - Una composicion farmaceutica para la prevencion y tratamiento de adiccion a nicotina en un mamifero - Google Patents

Una composicion farmaceutica para la prevencion y tratamiento de adiccion a nicotina en un mamifero

Info

Publication number
CO5700713A2
CO5700713A2 CO05113614A CO05113614A CO5700713A2 CO 5700713 A2 CO5700713 A2 CO 5700713A2 CO 05113614 A CO05113614 A CO 05113614A CO 05113614 A CO05113614 A CO 05113614A CO 5700713 A2 CO5700713 A2 CO 5700713A2
Authority
CO
Colombia
Prior art keywords
addiction
dependence
tobacco
treatment
pharmaceutical composition
Prior art date
Application number
CO05113614A
Other languages
English (en)
Inventor
Jotham W Coe
Steven Bradley Sands
Philip A Iredale
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of CO5700713A2 publication Critical patent/CO5700713A2/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/34Tobacco-abuse
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Addiction (AREA)
  • Organic Chemistry (AREA)
  • Psychiatry (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

1.- Una composición farmacéutica para tratar dependencia o adicción a nicotina, dependencia o adicción a tabaco, para reducir los síntomas de abstinencia de nicotina o para ayudar en el cese o disminución de uso de tabaco o abuso de sustancias o dependencias conductuales que comprende:(a) un agonista parcial de receptores nicotínicos o una sal farmacéuticamente aceptable del mismo;(b) un antagonista del receptor CB-1 o una sal farmacéuticamente aceptable del mismo; y (c) un vehículo farmacéuticamente aceptable;en la que los agentes activos "a" y "b" anteriores están presentes en cantidades que hacen la composición eficaz en el tratamiento de dependencia o adicción a nicotina, dependencia o adicción a tabaco, en la reducción de los síntomas de abstinencia de nicotina o en la ayuda en el cese o disminución de uso de tabaco o abuso de sustancias o dependencias conductuales.
CO05113614A 2003-05-09 2005-11-09 Una composicion farmaceutica para la prevencion y tratamiento de adiccion a nicotina en un mamifero CO5700713A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US46942903P 2003-05-09 2003-05-09

Publications (1)

Publication Number Publication Date
CO5700713A2 true CO5700713A2 (es) 2006-11-30

Family

ID=33435233

Family Applications (1)

Application Number Title Priority Date Filing Date
CO05113614A CO5700713A2 (es) 2003-05-09 2005-11-09 Una composicion farmaceutica para la prevencion y tratamiento de adiccion a nicotina en un mamifero

Country Status (13)

Country Link
US (1) US20040224963A1 (es)
EP (1) EP1624895A2 (es)
JP (1) JP2006525992A (es)
KR (1) KR20060009314A (es)
CN (1) CN1784243A (es)
AU (1) AU2004237153A1 (es)
BR (1) BRPI0410173A (es)
CA (1) CA2525225A1 (es)
CO (1) CO5700713A2 (es)
MX (1) MXPA05012088A (es)
NO (1) NO20055767L (es)
RU (1) RU2005131497A (es)
WO (1) WO2004098580A2 (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE521512C2 (sv) 2001-06-25 2003-11-11 Niconovum Ab Anordning för administrering av en substans till främre delen av en individs munhåla
EP1575901B1 (en) * 2002-12-19 2012-10-10 Merck Sharp & Dohme Corp. Substituted amides
EP1578422B1 (en) 2002-12-20 2007-04-11 NicoNovum AB A physically and chemically stable nicotine and micorcrystalline cellulose containing particulate material
US9402809B2 (en) 2006-03-16 2016-08-02 Niconovum Usa, Inc. Snuff composition

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2692575B1 (fr) * 1992-06-23 1995-06-30 Sanofi Elf Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
EP0937077B1 (en) * 1996-10-30 2006-05-17 Pfizer Inc. Pyridone-fused azabicyclic- or cytisine derivatives, their preparation and their use in addiction therapy
FR2758723B1 (fr) * 1997-01-28 1999-04-23 Sanofi Sa Utilisation des antagonistes des recepteurs aux cannabinoides centraux pour la preparation de medicaments
DK1044189T4 (en) * 1997-12-31 2015-03-30 Pfizer Prod Inc Aryl-fused fused azapolycyclic connections
CN1144787C (zh) * 1998-04-29 2004-04-07 辉瑞产品公司 芳基稠合氮杂多元环化合物
FR2804604B1 (fr) * 2000-02-09 2005-05-27 Sanofi Synthelabo Utilisation d'un antagoniste des recepteurs aux cannabinoides centraux pour la preparation de medicaments utiles pour faciliter l'arret de la consommation de tabac
TWI231757B (en) * 2001-09-21 2005-05-01 Solvay Pharm Bv 1H-Imidazole derivatives having CB1 agonistic, CB1 partial agonistic or CB1-antagonistic activity

Also Published As

Publication number Publication date
WO2004098580A2 (en) 2004-11-18
MXPA05012088A (es) 2006-02-22
EP1624895A2 (en) 2006-02-15
US20040224963A1 (en) 2004-11-11
AU2004237153A1 (en) 2004-11-18
JP2006525992A (ja) 2006-11-16
NO20055767L (no) 2005-12-05
KR20060009314A (ko) 2006-01-31
BRPI0410173A (pt) 2006-05-16
CN1784243A (zh) 2006-06-07
WO2004098580A3 (en) 2005-01-06
CA2525225A1 (en) 2004-11-18
RU2005131497A (ru) 2006-06-27

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Legal Events

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