CO2022017377A2 - Mezclas y composiciones que comprenden 5-fluoro-4-imino-3- metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de las mismas - Google Patents

Mezclas y composiciones que comprenden 5-fluoro-4-imino-3- metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de las mismas

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Publication number
CO2022017377A2
CO2022017377A2 CONC2022/0017377A CO2022017377A CO2022017377A2 CO 2022017377 A2 CO2022017377 A2 CO 2022017377A2 CO 2022017377 A CO2022017377 A CO 2022017377A CO 2022017377 A2 CO2022017377 A2 CO 2022017377A2
Authority
CO
Colombia
Prior art keywords
compound
formula
mixtures
effective amount
compositions
Prior art date
Application number
CONC2022/0017377A
Other languages
English (en)
Inventor
Jenny Lerner Yardeni
James Sloan
Original Assignee
Adama Makhteshim Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adama Makhteshim Ltd filed Critical Adama Makhteshim Ltd
Publication of CO2022017377A2 publication Critical patent/CO2022017377A2/es

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Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A01N25/22—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests containing ingredients stabilising the active ingredients
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/69—Benzenesulfonamido-pyrimidines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A01N25/02—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests containing liquids as carriers, diluents or solvents
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A01N25/02—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests containing liquids as carriers, diluents or solvents
    • A01N25/04—Dispersions, emulsions, suspoemulsions, suspension concentrates or gels
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A01N25/12—Powders or granules
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A01N25/30—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests characterised by the surfactants
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A01N25/32—Ingredients for reducing the noxious effect of the active substances to organisms other than pests, e.g. toxicity reducing compositions, self-destructing compositions
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P3/00—Fungicides

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Environmental Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Toxicology (AREA)
  • Microbiology (AREA)
  • Mycology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Dispersion Chemistry (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Composición líquida estable que comprende: (a) una cantidad fungicidamente eficaz de un compuesto de Fórmula I, y (b) un vehículo líquido, en el que: (i) la composición comprende (a) una sustancia fungicidamente eficaz y sustancialmente pura cantidad del compuesto de Fórmula I o una cantidad eficaz como fungicida de una mezcla que contiene el compuesto de Fórmula I, donde 95% o más en peso de la mezcla es el compuesto de Fórmula I, y (b) el vehículo líquido, y / o (ii) 95% o más de la cantidad del compuesto de Fórmula I está en forma de polimorfo de Forma I, polimorfo de Forma II, Hidrato, o una mezcla de los mismos. La presente invención también proporciona mezclas y composiciones que comprenden (a) una cantidad fungicidamente eficaz de un compuesto de Fórmula I y (b) al menos un adyuvante seleccionado del grupo que consiste en: (i) poli (óxido de alquileno) alquil éter; (ii) copolímero de óxido de polialquileno de siloxano; (iii) ésteres de ácidos grasos; (iv) vinilpirrolidonas y derivados de las mismas; (v) tensioactivos a base de azúcar, (vi) ligninas, (vii) terpenos; y (viii) cualquier combinación de (i), (ii), (iii), (iv), (v), (vi) y (vii). La presente invención también proporciona métodos de uso de las mezclas y composiciones descritas en este documento y procesos para preparar las mezclas y composiciones descritas en este documento.
CONC2022/0017377A 2020-05-04 2022-12-02 Mezclas y composiciones que comprenden 5-fluoro-4-imino-3- metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de las mismas CO2022017377A2 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063019871P 2020-05-04 2020-05-04
US202063024031P 2020-05-13 2020-05-13
PCT/IB2021/053762 WO2021224802A1 (en) 2020-05-04 2021-05-04 Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof

Publications (1)

Publication Number Publication Date
CO2022017377A2 true CO2022017377A2 (es) 2022-12-20

Family

ID=75888117

Family Applications (1)

Application Number Title Priority Date Filing Date
CONC2022/0017377A CO2022017377A2 (es) 2020-05-04 2022-12-02 Mezclas y composiciones que comprenden 5-fluoro-4-imino-3- metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de las mismas

Country Status (18)

Country Link
US (1) US20230292746A1 (es)
EP (1) EP4146632A1 (es)
JP (1) JP2023523655A (es)
KR (1) KR20230069875A (es)
CN (1) CN116113623A (es)
AU (1) AU2021267206A1 (es)
BR (1) BR112022022281A2 (es)
CA (1) CA3177682A1 (es)
CL (1) CL2022003040A1 (es)
CO (1) CO2022017377A2 (es)
CR (1) CR20220610A (es)
EC (1) ECSP22091704A (es)
IL (1) IL297864A (es)
MX (1) MX2022013874A (es)
PE (1) PE20230446A1 (es)
TW (1) TW202208341A (es)
UY (1) UY39197A (es)
WO (1) WO2021224802A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2023166485A1 (en) * 2022-03-03 2023-09-07 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
WO2024028812A1 (en) 2022-08-03 2024-02-08 Adama Makhteshim Ltd. 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1h)-one for fungicide-resistant fungus

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2588742T3 (es) 2010-04-26 2016-11-04 Adama Makhteshim Ltd Derivados de N1-sulfonil-5-fluoropirimidinona N3-sustituida
AU2014373961B2 (en) 2013-12-31 2017-10-26 Adama Makhteshim Ltd. 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1H)-one and processes for their preparation
CN114794123A (zh) 2013-12-31 2022-07-29 阿达玛马克西姆股份有限公司 用防治谷类中真菌的协同杀真菌混合物
MA41272A (fr) * 2014-12-23 2017-10-31 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences
IL271950B1 (en) 2017-07-17 2024-02-01 Adama Makhteshim Ltd Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-4,3-dihydropyrimidin-2-one
CA3118729A1 (en) * 2018-11-05 2020-05-14 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof

Also Published As

Publication number Publication date
MX2022013874A (es) 2022-11-30
EP4146632A1 (en) 2023-03-15
WO2021224802A1 (en) 2021-11-11
UY39197A (es) 2021-11-30
PE20230446A1 (es) 2023-03-08
CN116113623A (zh) 2023-05-12
CR20220610A (es) 2023-01-10
US20230292746A1 (en) 2023-09-21
AU2021267206A1 (en) 2022-12-08
CA3177682A1 (en) 2021-11-11
BR112022022281A2 (pt) 2023-01-03
IL297864A (en) 2023-01-01
KR20230069875A (ko) 2023-05-19
ECSP22091704A (es) 2023-02-28
CL2022003040A1 (es) 2023-07-07
JP2023523655A (ja) 2023-06-06
TW202208341A (zh) 2022-03-01

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