CO2022012616A2 - Compuestos de bencimidazol para el tratamiento de trastornos metabólicos - Google Patents
Compuestos de bencimidazol para el tratamiento de trastornos metabólicosInfo
- Publication number
- CO2022012616A2 CO2022012616A2 CONC2022/0012616A CO2022012616A CO2022012616A2 CO 2022012616 A2 CO2022012616 A2 CO 2022012616A2 CO 2022012616 A CO2022012616 A CO 2022012616A CO 2022012616 A2 CO2022012616 A2 CO 2022012616A2
- Authority
- CO
- Colombia
- Prior art keywords
- treatment
- metabolic disorders
- benzimidazole compounds
- formula
- prodrugs
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/26—Oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Diabetes (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Gastroenterology & Hepatology (AREA)
- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Child & Adolescent Psychology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
RESUMEN La presente invención se relaciona en forma amplia con un compuesto de bencimidazol de la Fórmula I para el tratamiento de obesidad, diabetes, enfermedad de hígado graso no alcohólico y esteatohepatitis no alcohólica: Fórmula I o sales, cristales, hidratos, prodrogas, metabolitos o solvatos del mismo farmacéuticamente aceptables.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US202063010128P | 2020-04-15 | 2020-04-15 | |
PCT/BR2021/050158 WO2021207816A1 (en) | 2020-04-15 | 2021-04-15 | Benzimidazole compound for the treatment of metabolic disorders |
Publications (1)
Publication Number | Publication Date |
---|---|
CO2022012616A2 true CO2022012616A2 (es) | 2022-10-21 |
Family
ID=78083461
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CONC2022/0012616A CO2022012616A2 (es) | 2020-04-15 | 2022-09-05 | Compuestos de bencimidazol para el tratamiento de trastornos metabólicos |
Country Status (15)
Country | Link |
---|---|
US (1) | US20230128304A1 (es) |
EP (1) | EP4136079A4 (es) |
JP (1) | JP2023522062A (es) |
KR (1) | KR20230002427A (es) |
CN (1) | CN115335363A (es) |
AR (1) | AR121842A1 (es) |
AU (1) | AU2021256476A1 (es) |
CA (1) | CA3171746A1 (es) |
CL (1) | CL2022002821A1 (es) |
CO (1) | CO2022012616A2 (es) |
EC (1) | ECSP22078679A (es) |
GB (1) | GB2609793B (es) |
MX (1) | MX2022009872A (es) |
PE (1) | PE20221568A1 (es) |
WO (1) | WO2021207816A1 (es) |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6124463A (en) * | 1998-07-02 | 2000-09-26 | Dupont Pharmaceuticals | Benzimidazoles as corticotropin release factor antagonists |
AU2003902860A0 (en) * | 2003-06-06 | 2003-06-26 | Daicel Chemical Industries, Ltd | Benzimidazole compounds |
ES2331274B1 (es) * | 2007-10-25 | 2010-10-21 | Ferrer Internacional, S.A. | Compuesto de indolina. |
CA2737694C (en) * | 2008-09-26 | 2013-07-02 | Merck Sharp & Dohme Corp. | Novel cyclic benzimidazole derivatives useful anti-diabetic agents |
BR102016024814A2 (pt) * | 2016-10-24 | 2018-05-08 | Aché Laboratórios Farmacêuticos S.A. | composto, processo de obtenção do composto, composição farmacêutica, uso do composto e método de tratamento de desordens psiquiátricas e/ou distúrbios do sono |
ES2711808B2 (es) * | 2017-11-02 | 2020-03-13 | Univ Granada | Uso de un agonista de melatonina para inducir la para inducir adipocitos beige en el tejido adiposo blanco |
-
2021
- 2021-04-14 AR ARP210100985A patent/AR121842A1/es unknown
- 2021-04-15 EP EP21788866.8A patent/EP4136079A4/en active Pending
- 2021-04-15 JP JP2022562996A patent/JP2023522062A/ja active Pending
- 2021-04-15 KR KR1020227035995A patent/KR20230002427A/ko unknown
- 2021-04-15 AU AU2021256476A patent/AU2021256476A1/en active Pending
- 2021-04-15 WO PCT/BR2021/050158 patent/WO2021207816A1/en active Search and Examination
- 2021-04-15 PE PE2022001524A patent/PE20221568A1/es unknown
- 2021-04-15 MX MX2022009872A patent/MX2022009872A/es unknown
- 2021-04-15 CN CN202180028308.5A patent/CN115335363A/zh active Pending
- 2021-04-15 GB GB2215434.8A patent/GB2609793B/en active Active
- 2021-04-15 CA CA3171746A patent/CA3171746A1/en active Pending
- 2021-04-15 US US17/915,248 patent/US20230128304A1/en active Pending
-
2022
- 2022-09-05 CO CONC2022/0012616A patent/CO2022012616A2/es unknown
- 2022-10-11 EC ECSENADI202278679A patent/ECSP22078679A/es unknown
- 2022-10-13 CL CL2022002821A patent/CL2022002821A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
EP4136079A1 (en) | 2023-02-22 |
AU2021256476A1 (en) | 2022-08-25 |
CL2022002821A1 (es) | 2023-04-10 |
MX2022009872A (es) | 2022-08-22 |
KR20230002427A (ko) | 2023-01-05 |
US20230128304A1 (en) | 2023-04-27 |
PE20221568A1 (es) | 2022-10-06 |
WO2021207816A1 (en) | 2021-10-21 |
GB2609793B (en) | 2024-05-08 |
ECSP22078679A (es) | 2022-11-30 |
AR121842A1 (es) | 2022-07-13 |
GB2609793A (en) | 2023-02-15 |
JP2023522062A (ja) | 2023-05-26 |
GB2609793A8 (en) | 2023-03-22 |
EP4136079A4 (en) | 2024-05-15 |
CN115335363A (zh) | 2022-11-11 |
CA3171746A1 (en) | 2021-10-21 |
GB202215434D0 (en) | 2022-11-30 |
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