CN118715213A - 用于制备n-(1-甲基环丙基)-2-(3-吡啶基)-2h-吲唑-4-甲酰胺及其中间体的方法 - Google Patents

用于制备n-(1-甲基环丙基)-2-(3-吡啶基)-2h-吲唑-4-甲酰胺及其中间体的方法 Download PDF

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Publication number
CN118715213A
CN118715213A CN202380022266.3A CN202380022266A CN118715213A CN 118715213 A CN118715213 A CN 118715213A CN 202380022266 A CN202380022266 A CN 202380022266A CN 118715213 A CN118715213 A CN 118715213A
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compound
solvent system
reaction
aspects
base
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Chinese (zh)
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A·埃尔-阿瓦
L·何
R·M·卡拉特卡尔
毛涧桦
J·米斯特里
M·帕蒂尔
C·S·斯托弗
P·韦卡利亚
J·A·赖特
T·沃格勒
D·A·克拉克
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FMC Corp
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FMC Corp
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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/26Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D307/30Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/561,2-Diazoles; Hydrogenated 1,2-diazoles
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    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
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    • C07C233/00Carboxylic acid amides
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    • C07C233/58Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of rings other than six-membered aromatic rings having the nitrogen atoms of the carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
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    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
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  • Pyridine Compounds (AREA)
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CN202380022266.3A 2022-02-17 2023-02-17 用于制备n-(1-甲基环丙基)-2-(3-吡啶基)-2h-吲唑-4-甲酰胺及其中间体的方法 Pending CN118715213A (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202263311276P 2022-02-17 2022-02-17
US63/311,276 2022-02-17
PCT/US2023/013266 WO2023158769A1 (en) 2022-02-17 2023-02-17 Processes for the preparation of n-(1- methylcyclopropyl)-2-(3 -pyridinyl)-2h- indazole-4-carboxamide and intermediates thereof

Publications (1)

Publication Number Publication Date
CN118715213A true CN118715213A (zh) 2024-09-27

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Family Applications (3)

Application Number Title Priority Date Filing Date
CN202380022266.3A Pending CN118715213A (zh) 2022-02-17 2023-02-17 用于制备n-(1-甲基环丙基)-2-(3-吡啶基)-2h-吲唑-4-甲酰胺及其中间体的方法
CN202380021091.4A Pending CN118679154A (zh) 2022-02-17 2023-02-17 N-(1-甲基环丙基)-2-(3-吡啶基)-2h-吲唑-4-甲酰胺及其中间体的制备
CN202380022264.4A Pending CN118715212A (zh) 2022-02-17 2023-02-17 N-(1-甲基环丙基)-2-(3-吡啶基)-2h-吲唑-4-甲酰胺及其中间体的制备

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CN202380021091.4A Pending CN118679154A (zh) 2022-02-17 2023-02-17 N-(1-甲基环丙基)-2-(3-吡啶基)-2h-吲唑-4-甲酰胺及其中间体的制备
CN202380022264.4A Pending CN118715212A (zh) 2022-02-17 2023-02-17 N-(1-甲基环丙基)-2-(3-吡啶基)-2h-吲唑-4-甲酰胺及其中间体的制备

Country Status (13)

Country Link
US (3) US20250154124A1 (https=)
EP (3) EP4479395A1 (https=)
JP (3) JP2025507561A (https=)
KR (3) KR20240152344A (https=)
CN (3) CN118715213A (https=)
AR (3) AR128561A1 (https=)
AU (3) AU2023221271A1 (https=)
IL (3) IL314649A (https=)
MX (3) MX2024010028A (https=)
PY (3) PY2311479A (https=)
TW (3) TW202342445A (https=)
UY (3) UY40151A (https=)
WO (3) WO2023158769A1 (https=)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI652014B (zh) 2013-09-13 2019-03-01 美商艾佛艾姆希公司 雜環取代之雙環唑殺蟲劑
CN112679467B (zh) * 2015-03-11 2024-11-01 Fmc公司 杂环取代的二环唑杀有害生物剂
BR112017019326B1 (pt) * 2015-03-12 2022-04-26 Fmc Corporation Composto, composição e método para controlar uma praga invertebrada
TWI873157B (zh) * 2019-07-11 2025-02-21 美商富曼西公司 包含吲唑之殺蟲混合物
CN111349111A (zh) * 2020-03-23 2020-06-30 安徽省逸欣铭医药科技有限公司 一种喷他佐辛前药、其制备方法及其用途

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MX2024010029A (es) 2024-08-22
UY40150A (es) 2023-09-15
IL314649A (en) 2024-09-01
WO2023158769A1 (en) 2023-08-24
UY40151A (es) 2023-09-15
JP2025507560A (ja) 2025-03-21
PY2311479A (es) 2023-10-05
KR20240152343A (ko) 2024-10-21
WO2023158771A1 (en) 2023-08-24
TW202342445A (zh) 2023-11-01
WO2023158770A1 (en) 2023-08-24
EP4479395A1 (en) 2024-12-25
EP4479393A1 (en) 2024-12-25
US20250163010A1 (en) 2025-05-22
AU2023220077A1 (en) 2024-08-22
PY2311482A (es) 2024-02-29
AR128559A1 (es) 2024-05-22
UY40152A (es) 2023-09-15
AU2023221271A1 (en) 2024-08-22
PY2311474A (es) 2023-09-14
IL314647A (en) 2024-09-01
MX2024010028A (es) 2024-08-22
MX2024010071A (es) 2024-08-20
TW202344496A (zh) 2023-11-16
JP2025507561A (ja) 2025-03-21
AR128561A1 (es) 2024-05-22
TW202342438A (zh) 2023-11-01
JP2025507562A (ja) 2025-03-21
US20250179043A1 (en) 2025-06-05
KR20240152345A (ko) 2024-10-21
AU2023222774A1 (en) 2024-08-22
US20250154124A1 (en) 2025-05-15
EP4479394A1 (en) 2024-12-25
KR20240152344A (ko) 2024-10-21
CN118715212A (zh) 2024-09-27
IL314592A (en) 2024-09-01
AR128557A1 (es) 2024-05-22
CN118679154A (zh) 2024-09-20

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