CN117120433A - 化合物、化合物的制造方法及保管方法、靶向剂的制造方法、以及组合物 - Google Patents

化合物、化合物的制造方法及保管方法、靶向剂的制造方法、以及组合物 Download PDF

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Publication number
CN117120433A
CN117120433A CN202280024610.8A CN202280024610A CN117120433A CN 117120433 A CN117120433 A CN 117120433A CN 202280024610 A CN202280024610 A CN 202280024610A CN 117120433 A CN117120433 A CN 117120433A
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CN
China
Prior art keywords
compound
reaction
ligand
acid
eluent
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Pending
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CN202280024610.8A
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English (en)
Chinese (zh)
Inventor
渡边友理惠
大泽沙优里
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Nihon Medi Physics Co Ltd
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Nihon Medi Physics Co Ltd
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Application filed by Nihon Medi Physics Co Ltd filed Critical Nihon Medi Physics Co Ltd
Publication of CN117120433A publication Critical patent/CN117120433A/zh
Pending legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B59/00—Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
    • C07B59/002—Heterocyclic compounds
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01D—SEPARATION
    • B01D15/00—Separating processes involving the treatment of liquids with solid sorbents; Apparatus therefor
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01D—SEPARATION
    • B01D15/00—Separating processes involving the treatment of liquids with solid sorbents; Apparatus therefor
    • B01D15/08—Selective adsorption, e.g. chromatography
    • B01D15/42—Selective adsorption, e.g. chromatography characterised by the development mode, e.g. by displacement or by elution
    • B01D15/424—Elution mode
    • B01D15/426—Specific type of solvent
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/05—Isotopically modified compounds, e.g. labelled

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CN202280024610.8A 2021-03-26 2022-03-25 化合物、化合物的制造方法及保管方法、靶向剂的制造方法、以及组合物 Pending CN117120433A (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2021-053783 2021-03-26
JP2021053783 2021-03-26
PCT/JP2022/014681 WO2022203082A1 (ja) 2021-03-26 2022-03-25 化合物、化合物の製造方法及び保管方法、ターゲッティング剤の製造方法、並びに組成物

Publications (1)

Publication Number Publication Date
CN117120433A true CN117120433A (zh) 2023-11-24

Family

ID=83397494

Family Applications (1)

Application Number Title Priority Date Filing Date
CN202280024610.8A Pending CN117120433A (zh) 2021-03-26 2022-03-25 化合物、化合物的制造方法及保管方法、靶向剂的制造方法、以及组合物

Country Status (5)

Country Link
US (1) US20240166631A1 (https=)
EP (1) EP4317152A4 (https=)
JP (2) JPWO2022203082A1 (https=)
CN (1) CN117120433A (https=)
WO (1) WO2022203082A1 (https=)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112020012099A2 (pt) * 2017-12-18 2020-11-17 Janssen Biotech, Inc. radiomarcação de polipeptídeos
BR112021022237A2 (pt) * 2019-05-10 2022-03-29 Janssen Biotech Inc Queladores macrocíclicos e métodos de uso dos mesmos

Also Published As

Publication number Publication date
EP4317152A4 (en) 2025-03-26
EP4317152A1 (en) 2024-02-07
JP2026012349A (ja) 2026-01-23
WO2022203082A1 (ja) 2022-09-29
JPWO2022203082A1 (https=) 2022-09-29
US20240166631A1 (en) 2024-05-23

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