CN116096371A - 含有饱和含氧杂环基的嘧啶二酮类化合物及其用途 - Google Patents
含有饱和含氧杂环基的嘧啶二酮类化合物及其用途 Download PDFInfo
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- CN116096371A CN116096371A CN202080103762.8A CN202080103762A CN116096371A CN 116096371 A CN116096371 A CN 116096371A CN 202080103762 A CN202080103762 A CN 202080103762A CN 116096371 A CN116096371 A CN 116096371A
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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Abstract
一种含有饱和含氧杂环基的嘧啶二酮类化合物及其用途，以及包含该类化合物的药物组合物，它们可以作为促性腺激素释放激素受体拮抗剂。还涉及制备这类化合物和药物组合物的方法，以及它们在预防或治疗性激素依赖性疾病，包括但不限于，前列腺癌、子宫内膜异位症、子宫肌瘤、性早熟等疾病中的用途。
Description
PCT国内申请，说明书已公开。
Claims (10)
- PCT国内申请，权利要求书已公开。
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/CN2020/119029 WO2022067566A1 (zh) | 2020-09-29 | 2020-09-29 | 含有饱和含氧杂环基的嘧啶二酮类化合物及其用途 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN116096371A true CN116096371A (zh) | 2023-05-09 |
| CN116096371A8 CN116096371A8 (zh) | 2024-05-14 |
Family
ID=80949338
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN202080103762.8A Pending CN116096371A (zh) | 2020-09-29 | 2020-09-29 | 含有饱和含氧杂环基的嘧啶二酮类化合物及其用途 |
Country Status (2)
| Country | Link |
|---|---|
| CN (1) | CN116096371A (zh) |
| WO (1) | WO2022067566A1 (zh) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2024031089A1 (en) | 2022-08-05 | 2024-02-08 | Gilead Sciences, Inc. | Sars-cov2 main protease inhibitors |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW449600B (en) * | 1994-04-19 | 2001-08-11 | Takeda Chemical Industries Ltd | Condensed-ring thiophene derivatives, their production and use |
| UY23948A1 (es) * | 1995-02-08 | 2001-10-25 | Takeda Chemical Industries Ltd | Derivados de anillos condensados de tiofeno su producción y uso. |
| WO2003064429A1 (fr) * | 2002-01-30 | 2003-08-07 | Takeda Chemical Industries, Ltd. | Thienopyrimidines, procedes de fabrication et d'utilisation correspondants |
| EP1495768A4 (en) * | 2002-04-12 | 2007-12-05 | Takeda Pharmaceutical | AGENTS FOR PREVENTING / TREATING HEAT BURSTS |
| WO2010026993A1 (ja) * | 2008-09-03 | 2010-03-11 | 武田薬品工業株式会社 | 製剤における吸収性改善方法および吸収性が改善された製剤 |
| CN109983017B (zh) * | 2017-07-28 | 2021-11-12 | 江苏恒瑞医药股份有限公司 | 一种嘧啶酮并杂芳基类衍生物的制备方法及其中间体 |
-
2020
- 2020-09-29 CN CN202080103762.8A patent/CN116096371A/zh active Pending
- 2020-09-29 WO PCT/CN2020/119029 patent/WO2022067566A1/zh active Application Filing
Also Published As
| Publication number | Publication date |
|---|---|
| WO2022067566A1 (zh) | 2022-04-07 |
| CN116096371A8 (zh) | 2024-05-14 |
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Address after: 523808 No.1, Gongye North Road, Songshanhu Park, Dongguan City, Guangdong Province Applicant after: Guangdong Dongyangguang Pharmaceutical Co.,Ltd. Address before: 523808 No.1, Gongye North Road, Songshanhu Park, Dongguan City, Guangdong Province Applicant before: SUNSHINE LAKE PHARMA Co.,Ltd. |
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Correction item: PCT international application to national stage day Correct: 2023.03.03 False: 2023.03.02 Number: 19-01 Page: The title page Volume: 39 Correction item: PCT international application to national stage day Correct: 2023.03.03 False: 2023.03.02 Number: 19-01 Volume: 39 |
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