CN115835905A - 用于用选择性组胺h1-受体拮抗剂左卡巴斯汀及其衍生物预防和治疗近视的方法和组合物 - Google Patents
用于用选择性组胺h1-受体拮抗剂左卡巴斯汀及其衍生物预防和治疗近视的方法和组合物 Download PDFInfo
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/451—Non condensed piperidines, e.g. piperocaine having a carbocyclic group directly attached to the heterocyclic ring, e.g. glutethimide, meperidine, loperamide, phencyclidine, piminodine
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0048—Eye, e.g. artificial tears
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0048—Eye, e.g. artificial tears
- A61K9/0051—Ocular inserts, ocular implants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/10—Ophthalmic agents for accommodation disorders, e.g. myopia
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- Chemical Kinetics & Catalysis (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
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| US202063033291P | 2020-06-02 | 2020-06-02 | |
| US63/033,291 | 2020-06-02 | ||
| PCT/US2021/035344 WO2021247635A1 (fr) | 2020-06-02 | 2021-06-02 | Méthodes et compositions pour la prévention et le traitement de la myopie avec de la lévocabastine, un antagoniste sélectif du récepteur h1 de l'histamine et des dérivés de celui-ci |
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| CN115835905A true CN115835905A (zh) | 2023-03-21 |
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| KR (1) | KR20230051130A (fr) |
| CN (1) | CN115835905A (fr) |
| CA (1) | CA3181292A1 (fr) |
| IL (1) | IL298796A (fr) |
| WO (1) | WO2021247635A1 (fr) |
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| CN116270442A (zh) * | 2021-12-21 | 2023-06-23 | 浙江瑞瞳生物科技有限公司 | 一种用于矫正近距离视力的眼用制剂 |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| WO2010095478A1 (fr) * | 2009-02-20 | 2010-08-26 | 株式会社シード | Lentille de contact en hydrogel à libération prolongée de médicament et procédé de libération de médicament mettant en oeuvre une lentille de contact en hydrogel à libération prolongée de médicament |
| US9827250B2 (en) * | 2012-07-31 | 2017-11-28 | Johnson & Johnson Vision Care, Inc. | Lens incorporating myopia control optics and muscarinic agents |
| ITUB20160876A1 (it) * | 2016-02-19 | 2017-08-19 | Dambrosio Enzo Maria | Combinazione di un agente antiallergico con un antagonista muscarinico e/o un agonista dopaminergico per l'uso in prevenzione/ arresto di miopia assiale nell’uomo |
| US10945980B2 (en) * | 2016-06-21 | 2021-03-16 | The University Of Newcastle | Treatment for myopia |
| KR20200007769A (ko) * | 2017-02-21 | 2020-01-22 | 싱가포르 헬스 서비시즈 피티이 엘티디 | 아트로핀을 포함하는 근시의 발병을 방지 또는 지연하기 위한 조성물 및 방법 |
| EP3713530A4 (fr) * | 2017-11-21 | 2021-08-18 | Sydnexis, Inc. | Composition ophtalmique et dispositif d'administration associé |
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2021
- 2021-06-02 CN CN202180049465.4A patent/CN115835905A/zh active Pending
- 2021-06-02 WO PCT/US2021/035344 patent/WO2021247635A1/fr unknown
- 2021-06-02 JP JP2022574559A patent/JP2023529374A/ja active Pending
- 2021-06-02 EP EP21816939.9A patent/EP4157453A4/fr active Pending
- 2021-06-02 CA CA3181292A patent/CA3181292A1/fr active Pending
- 2021-06-02 IL IL298796A patent/IL298796A/en unknown
- 2021-06-02 KR KR1020227046225A patent/KR20230051130A/ko active Search and Examination
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| Publication number | Publication date |
|---|---|
| KR20230051130A (ko) | 2023-04-17 |
| JP2023529374A (ja) | 2023-07-10 |
| EP4157453A4 (fr) | 2024-06-19 |
| EP4157453A1 (fr) | 2023-04-05 |
| CA3181292A1 (fr) | 2021-12-09 |
| IL298796A (en) | 2023-02-01 |
| WO2021247635A1 (fr) | 2021-12-09 |
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