CN111635353A - 非晶形特考韦瑞制备 - Google Patents
非晶形特考韦瑞制备 Download PDFInfo
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- CN111635353A CN111635353A CN202010516675.7A CN202010516675A CN111635353A CN 111635353 A CN111635353 A CN 111635353A CN 202010516675 A CN202010516675 A CN 202010516675A CN 111635353 A CN111635353 A CN 111635353A
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- amorphous
- isoindol
- octahydro
- dioxo
- benzamide
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| CN107126419B (zh) * | 2016-02-26 | 2020-06-19 | 石药集团中诺药业（石家庄）有限公司 | 一种奥贝胆酸片剂及其制备方法 |
| CN112955130A (zh) * | 2018-10-30 | 2021-06-11 | 佩洛通治疗公司 | 包含取代茚满的固体分散体和药物组合物及其制备和使用方法 |
| CN115141136B (zh) * | 2021-03-31 | 2023-06-20 | 中国人民解放军军事科学院军事医学研究院 | 特考韦瑞药的共晶及其制备方法 |
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| CN103068232A (zh) * | 2010-03-23 | 2013-04-24 | 西佳科技股份有限公司 | 多晶型物形式st-246和制备方法 |
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| US6596771B2 (en) | 2001-01-12 | 2003-07-22 | Schering Corporation | Drugs for treating viral infections |
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| US8642577B2 (en) * | 2005-04-08 | 2014-02-04 | Chimerix, Inc. | Compounds, compositions and methods for the treatment of poxvirus infections |
| JP2010526848A (ja) * | 2007-05-11 | 2010-08-05 | エフ．ホフマン−ラ ロシュ アーゲー | 難溶性薬物用の医薬組成物 |
| BR112012031516A2 (pt) * | 2010-06-09 | 2016-11-08 | Abbott Lab | dispersões sólidas contendo inibidores de quinase |
| GB201103837D0 (en) * | 2011-03-07 | 2011-04-20 | Oxagen Ltd | Amorphous (5-Fluoro-2-Methyl-3-Quinolin-2-Ylmethyl-Indol-1-Yl)-acetic acid |
| US8591944B2 (en) * | 2011-03-08 | 2013-11-26 | Zalicus Pharmaceuticals Ltd. | Solid dispersion formulations and methods of use thereof |
| WO2013056108A2 (en) * | 2011-10-14 | 2013-04-18 | Array Biopharma Inc. | Solid dispersion |
| JP2013103899A (ja) * | 2011-11-11 | 2013-05-30 | Fuji Chem Ind Co Ltd | 難溶性薬物の新規な固体分散体 |
| WO2015009566A1 (en) | 2013-07-19 | 2015-01-22 | Siga Technologies, Inc. | Amorphous tecovirimat preparation |
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| CN103068232A (zh) * | 2010-03-23 | 2013-04-24 | 西佳科技股份有限公司 | 多晶型物形式st-246和制备方法 |
| CN102406617A (zh) * | 2011-11-30 | 2012-04-11 | 中国人民解放军军事医学科学院生物工程研究所 | 一种替韦立马干混悬剂及其制备方法 |
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| DOUGLAS W GROSENBACH等: "Development of the small-molecule antiviral ST-246 as a smallpox therapeutic", 《FUTURE VIROLOGY》, vol. 6, no. 5, pages 653 - 671, XP055232795, DOI: 10.2217/fvl.11.27 * |
| 陆彬: "药物新剂型与新技术 第2版", 人民卫生出版社, pages: 3 - 5 * |
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