CN108815076A - 一种美白护肤霜及其制备方法 - Google Patents
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Abstract
本发明公开了一种美白护肤霜及其制备方法,包括以下成分:A、油相w(%):硬脂酸4.5%,十八醇2.51%,十六醇2.5%,白油3.1%,Twenn‑60 0.5%,羊毛脂1.2%,橄榄油0.5%;B、水相:白芷提取物2.0%,甘油6.5%,三乙醇胺0.31%,芦荟浸膏1%,白果提取物1.5%,蒸馏水73.60%;C、香精0.03%,防腐剂0.25%。采用天然原料,加入有特殊作用的中草药提取物,制成水包油型的乳化产品。经初步试用,安全性好,可以消除肌肤色素,使肌肤自然、美白亮泽。
Description
技术领域
本发明属于化妆品技术领域,具体地说,一种美白护肤霜及其制备方法。
背景技术
随着社会的进步和发展,生活水平的日益提高,化妆品已愈来愈成为现代人生活中不可缺少的一部分。与此同时,人们对于化妆品的质量和性能要求也越来越高。人们希望出现一系列对人体健康无害,又具有美容保健作用的天然原料制备的护肤化妆品。天然植物类化妆品其特点为:在油水混合物中,添加各类天然植物提取营养物质的化妆品。利用中草药提取物作为美容护肤化妆品的添加剂,具有药性稳定,药力持久,对皮肤作用温和、刺激性小、安全性高、疗效显著等特点。因此,以中草药提取物作为天然物添加剂应用于化妆品中,已逐渐成为新产品开发的热点。
发明内容
本发明的目的在于提供一种美白护肤霜及其制备方法,采用天然原料,加入有特殊作用的中草药提取物,制成水包油型的乳化产品。经初步试用,安全性好,可以消除肌肤色素,使肌肤自然、美白亮泽。
其具体技术方案为:
一种美白护肤霜,包括以下成分:
A 油相 w(%)
硬脂酸4.5%,十八醇2.51%,十六醇2.5%,白油3.1%, Twenn-60 0.5%,羊毛脂1.2%,橄榄油0.5%。
B 水相
白芷提取物2.0%,甘油6.5%,三乙醇胺0.31%,芦荟浸膏1%,白果提取物(浓缩物)1.5%,蒸馏水73.60%。
C 香精0.03%,防腐剂0.25%。
本发明研制的是美白护肤化妆品。美白化妆品是指能阻碍酪氨酸酶的活性,或作用于黑色素代谢途径的各个阶段,控制、抑制黑色素生成的化妆品。酪氨酸酶普遍存在于人和动植物体内,是黑色素生物合成过程中必不可少的关键酶。酪氨酸酶的合成和催化活力的升高,使体内黑色素合成增多,导致色斑及黑色素瘤的形成。研究表明:可通过抑制酪氨酸酶活力来预防和治疗色素沉着及黑色素瘤,因此寻找有效且对人体无毒副作用的酪氨酸酶抑制剂成为研究美白化妆品配方的关键之一。本发明选出白芷、白果和芦荟三种有明显抑制黑色素转化酶活性作用的天然植物及中草药。
芦荟是百合科的肉质植物,芦荟的特征成份是芦荟大黄素及其衍生物和多种肽(酶)。包含丰富的维生素、多种氨基酸等成份,具有一系列的治疗功效和滋养皮肤的多种功效成份,对软化皮肤,收敛和防治粉刺、老年斑、雀斑、皮肤粗糙以及消炎止痒、护发、保护皮肤细嫩白洁等都有显著功效。芦荟提取物中有多种营养成份,具有营养皮肤的功能,其中多种碳水化合物、多聚糖、氨基酸是天然的保湿剂,且含有多种消除超氧化物自由基的成份,能延缓皮肤衰老和消除黄褐斑,使用安全、无毒无副作用。
白果仁就是银杏干燥成熟的种子,其味甘、苦、涩,具有敛肺定喘、止带浊、缩小便的功效。常用于痰多喘咳,带下白浊,遗尿、尿频等疾病的治疗。其富含的白果酸在体外可抑制一些皮肤真菌。所以,外用可治头面手足多种碍容性皮肤病,并可延缓皮肤衰老,防止皮肤粗糙,可令肌肤柔嫩光滑,白皙娇美。在身体状态不好时,本发明的内分泌就容易紊乱、失调,这时体内的氧自由基过多,但是过氧化物歧化酶(SOD)不足,导致过多的氧自由基与真皮层细胞产生氧化的反应,形成大量的脂褐素(过氧化脂质),造成黄褐斑或是妊娠斑。白果中所含有的黄酮成分可以阻碍色素在真皮层的形成与沉着,达到美白肌肤与防治色素斑块的作用。除了黄酮之外,白果中的锰、钼等微量元素,亦能清除氧自由基及抑制黑色素生长;白果中所含的银杏酸对酪氨酸酶具有明显的抑制作用,可抑制酪氨酸酶单酚酶和二酚酶活力,可预防和治疗色素沉着及黑色素瘤。
白芷味香色白,微温,入药始载于《神农本草经》,因具有特殊的芳香气味,所以又名香白芷。其外用为美容要药,古代美容方多用之。《日华子本草》记载其“去面皮平疵瘕”。《本草纲目》谓其有“长肌肤,调泽颜色,可作面脂”之效,面脂即当今流行的面膜。
白芷兼具美白、防晒双重效果,而且富含精油成分,有很好的抗菌及促进血液循环的作用,具有让面色红润和改善黑头粉刺的功效。
在研制化妆品配方时,本发明对传统化妆品配方也做改进,使其在滋润美白,稳定,无害等方面更加完美。本发明改变了化妆品配方中辅料的配比,减少一些粘度较大的油相成份比例,加入羊毛脂,增加甘油成份和水的含量等,可使化妆品的营养性、渗透性更好,降低油腻感,对皮肤的保湿也有改善,使用时感觉舒适。
一种本发明所述美白护肤霜的制备方法,包括以下步骤:
(1)油相制备
预备以下重量比组分:4.5%硬脂酸、2.51%十八醇、2.5%十六醇、twenn-60 0.5%、1.2%羊毛脂、3.1%白油、0.5%橄榄油。
分别将以上预备组分硬脂酸、十八醇、十六醇、twenn-60、羊毛脂、白油置于电热恒温水浴锅内,搅拌加热至80-90℃,完全熔化呈均相后,加入0.5%橄榄油,继续搅拌,保温20-30min,形成油相混合物,备用;
(2)水相制备
预备以下重量比组分:甘油6.5%、白芷提取物2.0%、三乙醇胺0.31%、白果提取物(浓缩物)1.5%、73.60%蒸馏水。
将以上预备组分甘油、白芷提取物、三乙醇胺、白果提取物(浓缩物)蒸馏水置于电热恒温水浴锅内搅拌加热至85~95℃,完全熔化呈均相后,保温20至30min,灭菌过滤后得到水相混合物;
(3)乳液制备
预备以下重量比组分:1%的芦荟浸膏、0.03%香精, 0.25%防腐剂。
80-90 ℃下缓慢将油相混合物加入到水相混合物中,边加入边搅拌,搅拌均匀后继续搅拌 40-90min,搅拌并缓慢降温至65℃时,加入芦荟浸膏,继续搅拌降温。待温度降至45℃时,加入香精,防腐剂,持续搅拌,待温度降至35℃左右时停止搅拌,静置,冷却,得到乳膏状产品,取样检验。
与现有技术相比,本发明的有益效果为:
本发明在研制化妆品配方时,经过多种配方对比,选优实验,最后确定本品以硬脂酸和三乙醇胺作为乳化剂,表面活性剂Twenn-60起到增加乳化效果的作用,添加十六醇、十八醇作为乳化助剂,白油用作润肤剂和保湿剂,羊毛脂具有软化角质皮层的特殊作用,橄榄油能柔润皮肤、对皮肤有良好的收敛和渗透性,以甘油作为保湿剂,并增加甘油成份和水的含量,可使化妆品的营养性、渗透性更好,降低油腻感,对皮肤的保湿也有改善,使用时感觉舒适。采用复合型防腐剂(以布罗波尔、尼泊金丙酯、山梨酸)来预防微生物污染。
具体实施方式
下面结合具体实施例对本发明的技术方案作进一步详细地说明。
1 原料浸出液的制备
1.1 芦荟提取物的制备
选择2~3年以上叶龄、生长状况良好的新鲜芦荟叶洗净切碎,研磨0.5 h后放入碘量瓶中,加入100mL乙醚浸泡5h进行脱色,抽滤(同收乙醚),加300mL体积分数为95%的乙醇浸泡24h后减压蒸馏,将残留的乙醚和过量的乙醇低温蒸出。并利用吸附方法除去大黄素,醌甙等苦味成份。通过低温浓缩成一定黏度的芦荟提取物。
1.2 白芷有效成分提取
取适量白芷粉碎,过40目筛,称取适量与70%乙醇按1:12(g:ml)比例加入到三角锥形瓶中,室温放置,期间多次振荡,48h后过滤,45℃水浴真空旋转蒸发浓缩,超纯水溶解收集,收集液用真空冷冻干燥机冷冻干燥成粉末,均质得白芷提取物。
1.3 白果有效成分提取
白果去除种皮,置于烘箱中烘干至恒重,经粉碎机打粉并过40 目筛,置于干燥器内备用。取适量白果粉置于250 mL的三角瓶中,加入70%乙醇溶液(料液比1:15),70 ℃下超声提取40min,将滤渣再连续提取2次,合并提取液,旋转蒸发仪浓缩,得浓缩液备用。
2 .美白护肤霜的研制工艺
2.1 原料及其规格
白果浸膏(新提取)、白油(化妆品级)、羊毛脂(化妆品级)、橄榄油(化妆品级)、三乙醇胺(分析纯)、十八醇(化学纯)、硬酯酸(一级品)、化妆品防腐剂(布罗波尔、尼泊金丙酯、山梨酸)、芦荟浸膏(新制备)、白芷提取物(新制备)、吐温(实验试剂)、十六醇(化学纯)、丙三醇(分析纯)、香精、蒸馏水。
2.2 仪器
AFR-1高剪切混合乳化机,上海艾枫机电设备厂;CS101-4型电热鼓风干燥器,重庆试验设备厂;RE-52C型旋转蒸发器,上海亚荣生化仪器厂; 西门子KK19V70TI型电冰箱;TGL-16C型高速台式离心机,上海安亭科学仪器厂;pHS-3C型精密pH计,上海雷磁仪器厂;FA1004型电子分析天平,上海金鹏分析仪器有限公司;HH·SH-2型电热恒温水浴锅,北京长安科学仪器厂;JJ-1型定时电动搅拌器,江苏省金坛市金城教学仪器厂。
2.3 配方
A 油相 w(%)
硬脂酸4.5%,十八醇2.51%,十六醇2.5%,白油3.1%, Twenn-60 0.5%,羊毛脂1.2%,橄榄油0.5%。
B 水相
白芷提取物2.0%,甘油6.5%,三乙醇胺0.31%,芦荟浸膏1%,白果提取物(浓缩物)1.5%,蒸馏水73.60%。。
C 香精0.03%,防腐剂0.25%。
在研制化妆品配方时,经过多种配方对比,选优实验,最后确定本品以硬脂酸和三乙醇胺作为乳化剂,表面活性剂Twenn-60起到增加乳化效果的作用,添加十六醇、十八醇作为乳化助剂,白油用作润肤剂和保湿剂,羊毛脂具有软化角质皮层的特殊作用,橄榄油能柔润皮肤、对皮肤有良好的收敛和渗透性,以甘油作为保湿剂,并增加甘油成份和水的含量,可使化妆品的营养性、渗透性更好,降低油腻感,对皮肤的保湿也有改善,使用时感觉舒适。采用复合型防腐剂(以布罗波尔、尼泊金丙酯、山梨酸)来预防微生物污染。
2.4 制备方法
(1)油相制备
预备以下重量比组分:4.5%硬脂酸、2.51%十八醇、2.5%十六醇、twenn-60 0.5%、1.2%羊毛脂、3.1%白油、0.5%橄榄油。
分别将以上预备组分硬脂酸、十八醇、十六醇、twenn-60、羊毛脂、白油置于电热恒温水浴锅内,搅拌加热至80-90℃,完全熔化呈均相后,加入0.5%橄榄油,继续搅拌,保温20-30min,形成油相混合物,备用;
(2)水相制备
预备以下重量比组分:甘油6.5%、白芷提取物2.0%、三乙醇胺0.31%、白果提取物(浓缩物)1.5%、73.60%蒸馏水。
将以上预备组分甘油、白芷提取物、三乙醇胺、白果提取物(浓缩物)蒸馏水置于电热恒温水浴锅内搅拌加热至85~95℃完全熔化呈均相后,保温20至30min,灭菌过滤后得到水相混合物;
(3)乳液制备
预备以下重量比组分:1%的芦荟浸膏、0.03%香精,0.05%布罗波尔 0.2%防腐剂。
80-90 ℃下缓慢将油相混合物加入到水相混合物中,边加入边搅拌,搅拌均匀后继续搅拌 40-90min,搅拌并缓慢降温至65℃时,加入芦荟浸膏,继续搅拌降温。待温度降至45℃时,加入香精、防腐剂,持续搅拌,待温度降至35℃左右时停止搅拌,静置,冷却,得到乳膏状产品,取样检验 。
以上所述,仅为本发明较佳的具体实施方式,本发明的保护范围不限于此,任何熟悉本技术领域的技术人员在本发明披露的技术范围内,可显而易见地得到的技术方案的简单变化或等效替换均落入本发明的保护范围内。
Claims (5)
1.一种美白护肤霜,其特征在于,包括以下成分:
A 油相
硬脂酸4.5%,十八醇2.51%,十六醇2.5%,白油3.1%, Twenn-60 0.5%,羊毛脂1.2%,橄榄油0.5%;
B 水相
白芷提取物2.0%,甘油6.5%,三乙醇胺0.31%,芦荟浸膏1%,白果提取物1.5%,蒸馏水73.60%;
C 香精0.03%,防腐剂0.25%。
2.一种权利要求1所述美白护肤霜的制备方法,其特征在于,包括以下步骤:
(1) 油相制备
预备以下重量比组分:4.5%硬脂酸、2.51%十八醇、2.5%十六醇、twenn-60 0.5%、1.2%羊毛脂、3.1%白油、0.5%橄榄油;
分别将以上预备组分硬脂酸、十八醇、十六醇、twenn-60、羊毛脂、白油置于电热恒温水浴锅内,搅拌加热至80-90℃,完全熔化呈均相后,加入0.5%橄榄油,继续搅拌,保温20-30min,形成油相混合物,备用;
(2) 水相制备
预备以下重量比组分:甘油6.5%、白芷提取物2.0%、三乙醇胺0.31%、白果提取物1.5%、73.60%蒸馏水;
将以上预备组分甘油、白芷提取物、三乙醇胺、白果提取物蒸馏水置于电热恒温水浴锅内搅拌加热至85~95℃完全熔化呈均相后,保温20至30min,灭菌过滤后得到水相混合物;
(3) 乳液制备
预备以下重量比组分:1%的芦荟浸膏、0.03%香精, 0.25%防腐剂;
80-90 ℃下缓慢将油 相混合物加入到水相混合物中,边加入边搅拌,搅拌均匀后继续搅拌 40-90min,搅拌并缓慢降温至65℃时,加入芦荟浸膏,继续搅拌降温;待温度降至45℃时,加入香精、防腐剂,持续搅拌,待温度降至35℃时停止搅拌,静置,冷却,得到乳膏状产品,取样检验。
3.根据权利要求2所述美白护肤霜的制备方法,其特征在于,所述香精为茉莉香精或玫瑰香精。
4.根据权利要求2所述美白护肤霜的制备方法,其特征在于,所述防腐剂为布罗波尔、尼泊金丙酯、山梨酸的一种或两种。
5. 根据权利要求2所述美白护肤霜的制备方法,其特征在于,所述防腐剂由布罗波尔、尼泊金丙酯、山梨酸混合而成,三者的质量比为1 : 3:1。
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