CN108601770B - Pad4的氮杂-苯并咪唑抑制剂 - Google Patents

Pad4的氮杂-苯并咪唑抑制剂 Download PDF

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CN108601770B
CN108601770B CN201680081046.8A CN201680081046A CN108601770B CN 108601770 B CN108601770 B CN 108601770B CN 201680081046 A CN201680081046 A CN 201680081046A CN 108601770 B CN108601770 B CN 108601770B
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compound
pharmaceutically acceptable
ring
pyrrolo
pyridine
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CN108601770A (zh
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R.德夫拉伊
G.库马拉维尔
L.格利夫
A.科泰
T.克鲁尔
C.莱茨
H.泰
I.维金顿
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Padlock Therapeutics Inc
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Padlock Therapeutics Inc
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TW202140477A (zh) * 2020-02-12 2021-11-01 美商必治妥美雅史谷比公司 雜環ｐａｄ４抑制劑
MX2022013615A (es) 2020-04-30 2022-11-16 Gilead Sciences Inc Inhibidores de macrociclo de peptidilarginina deiminasas.
EP4267562A1 (en) 2020-12-22 2023-11-01 Gilead Sciences, Inc. Inhibitors of peptidylarginine deiminases
TW202233174A (zh) 2020-12-22 2022-09-01 美商基利科學股份有限公司 肽基精胺酸去亞胺酶之抑制劑
WO2025024265A1 (en) 2023-07-21 2025-01-30 Bristol-Myers Squibb Company Methods of assessing citrullination and activity of pad4 modulators
WO2025199042A1 (en) * 2024-03-18 2025-09-25 Seattle Children's Hospital D/B/A Seattle Children's Research Institute Methods for treating severe tuberculosis
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