CN107753962A - 放射性示踪剂组合物 - Google Patents
放射性示踪剂组合物 Download PDFInfo
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- CN107753962A CN107753962A CN201711237827.4A CN201711237827A CN107753962A CN 107753962 A CN107753962 A CN 107753962A CN 201711237827 A CN201711237827 A CN 201711237827A CN 107753962 A CN107753962 A CN 107753962A
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
- A61K51/0497—Organic compounds conjugates with a carrier being an organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
- A61K51/08—Peptides, e.g. proteins, carriers being peptides, polyamino acids, proteins
- A61K51/082—Peptides, e.g. proteins, carriers being peptides, polyamino acids, proteins the peptide being a RGD-containing peptide
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B59/00—Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
- C07B59/008—Peptides; Proteins
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B63/00—Purification; Separation; Stabilisation; Use of additives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/13—Labelling of peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Optics & Photonics (AREA)
- Physics & Mathematics (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Analytical Chemistry (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US42139010P | 2010-12-09 | 2010-12-09 | |
| US61/421390 | 2010-12-09 | ||
| CN2011800590925A CN103338791A (zh) | 2010-12-09 | 2011-12-09 | 放射性示踪剂组合物 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN2011800590925A Division CN103338791A (zh) | 2010-12-09 | 2011-12-09 | 放射性示踪剂组合物 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN107753962A true CN107753962A (zh) | 2018-03-06 |
Family
ID=45346469
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN201711237827.4A Pending CN107753962A (zh) | 2010-12-09 | 2011-12-09 | 放射性示踪剂组合物 |
| CN2011800590925A Pending CN103338791A (zh) | 2010-12-09 | 2011-12-09 | 放射性示踪剂组合物 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN2011800590925A Pending CN103338791A (zh) | 2010-12-09 | 2011-12-09 | 放射性示踪剂组合物 |
Country Status (7)
| Country | Link |
|---|---|
| US (2) | US9180213B2 (https=) |
| EP (1) | EP2648767B1 (https=) |
| JP (1) | JP6055417B2 (https=) |
| KR (1) | KR20130124522A (https=) |
| CN (2) | CN107753962A (https=) |
| CA (1) | CA2820387A1 (https=) |
| WO (1) | WO2012076697A1 (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB201202420D0 (en) * | 2012-02-13 | 2012-03-28 | Ge Healthcare Ltd | Radiotracer compositions |
| CN104470547B (zh) * | 2012-05-24 | 2018-01-26 | 未来化学株式会社 | 利用筒状物合成放射性药物的方法 |
| GB201221266D0 (en) * | 2012-11-27 | 2013-01-09 | Ge Healthcare Ltd | Aldehyde compositions |
| GB201314936D0 (en) | 2013-08-21 | 2013-10-02 | Ge Healthcare Ltd | Radiolabelling method |
| GB201322456D0 (en) * | 2013-12-18 | 2014-02-05 | Ge Healthcare Ltd | Radiotracer compositions and methods |
| KR102668112B1 (ko) * | 2014-12-04 | 2024-05-23 | 지이 헬쓰케어 리미티드 | 방사성 약제로부터의 아세트알데히드의 제거 방법 |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101151054A (zh) * | 2004-09-14 | 2008-03-26 | 通用电气医疗集团股份有限公司 | 放射性氟化肽 |
| WO2010079079A2 (en) * | 2008-12-17 | 2010-07-15 | General Electric Company | PDGF-Rβ BINDERS |
| WO2010114723A1 (en) * | 2009-03-30 | 2010-10-07 | Ge Healthcare Limited | Radiolabelling reagents and methods |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0305704D0 (en) | 2003-03-13 | 2003-04-16 | Amersham Plc | Radiofluorination methods |
| US7659400B2 (en) | 2003-07-31 | 2010-02-09 | Washington University | Radiolabelled benzamide analogues, their synthesis and use in diagnostic imaging |
| CA2619941C (en) | 2005-08-31 | 2014-04-01 | Immunomedics, Inc. | F-18 peptides for pre targeted positron emission tomography imaging |
| US8586595B2 (en) * | 2007-02-07 | 2013-11-19 | Purdue Research Foundation | Positron emission tomography imaging method |
| WO2009002914A2 (en) | 2007-06-25 | 2008-12-31 | Interdigital Technology Corporation | Method and apparatus for supporting inter-frequency and inter-radio access technology handover |
| EP2297070A2 (en) * | 2008-07-03 | 2011-03-23 | Bayer Schering Pharma Aktiengesellschaft | Compounds and processes for production of radiopharmaceuticals |
| EP2322500A1 (en) | 2009-11-11 | 2011-05-18 | Bayer Schering Pharma Aktiengesellschaft | Fluoro-labeled homo-glutamate derivatives and precursors thereof |
| AU2010321278B2 (en) | 2009-11-17 | 2014-08-14 | Piramal Imaging Sa | Method for production of F-18 labeled glutamic acid derivatives |
-
2011
- 2011-12-09 CA CA2820387A patent/CA2820387A1/en not_active Abandoned
- 2011-12-09 CN CN201711237827.4A patent/CN107753962A/zh active Pending
- 2011-12-09 EP EP11794725.9A patent/EP2648767B1/en active Active
- 2011-12-09 CN CN2011800590925A patent/CN103338791A/zh active Pending
- 2011-12-09 WO PCT/EP2011/072352 patent/WO2012076697A1/en not_active Ceased
- 2011-12-09 US US13/992,800 patent/US9180213B2/en active Active
- 2011-12-09 JP JP2013542563A patent/JP6055417B2/ja active Active
- 2011-12-09 KR KR1020137017594A patent/KR20130124522A/ko not_active Withdrawn
-
2015
- 2015-10-07 US US14/877,107 patent/US9987382B2/en active Active
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101151054A (zh) * | 2004-09-14 | 2008-03-26 | 通用电气医疗集团股份有限公司 | 放射性氟化肽 |
| WO2010079079A2 (en) * | 2008-12-17 | 2010-07-15 | General Electric Company | PDGF-Rβ BINDERS |
| WO2010114723A1 (en) * | 2009-03-30 | 2010-10-07 | Ge Healthcare Limited | Radiolabelling reagents and methods |
Non-Patent Citations (2)
| Title |
|---|
| THORSTEN POETHKO,ET AL: "Two-Step Methodology for High-Yield Routine Radiohalogenation of Peptides: 18F-Labeled RGD and Octreotide Analogs", 《THE JOURNAL OF NUCLEAR MEDICINE》 * |
| XUEHE LI，ET AL: "Site-Specific Labeling of Annexin V with F-18 for Apoptosis Imaging", 《BIOCONJUGATE CHEMISTRY》 * |
Also Published As
| Publication number | Publication date |
|---|---|
| JP2014500268A (ja) | 2014-01-09 |
| CN103338791A (zh) | 2013-10-02 |
| US20160022847A1 (en) | 2016-01-28 |
| JP6055417B2 (ja) | 2016-12-27 |
| US9987382B2 (en) | 2018-06-05 |
| CA2820387A1 (en) | 2012-06-14 |
| WO2012076697A1 (en) | 2012-06-14 |
| EP2648767B1 (en) | 2023-03-15 |
| US9180213B2 (en) | 2015-11-10 |
| EP2648767A1 (en) | 2013-10-16 |
| KR20130124522A (ko) | 2013-11-14 |
| US20130259804A1 (en) | 2013-10-03 |
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Application publication date: 20180306 |