CN107469054A - 一种可有效治疗消化性溃疡的内服药物及其制备方法 - Google Patents
一种可有效治疗消化性溃疡的内服药物及其制备方法 Download PDFInfo
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Abstract
本发明属于中药制剂领域,目的是根据中医治疗消化性溃疡的认识机理而提供一种可有效治疗消化性溃疡的内服药物,所述药物的各个组分及其质量份比如下:丹参90~180g、白芷50~160g、白术80~160g、党参150~280g、砂仁30~70g、干姜30~100g、玄参90~160g、肿节风90~350g、芡实90~160g、肉桂50~45g、人参30~100g、枳实30~100g、海螵蛸(炒黄)100~360g、木香15~70g、山楂30~120g、陈皮30~120g、蒲公英150~550g、苦杏仁45~90g、厚朴30~120g、青皮30~120g、蒲黄50~100g、地榆90~160g、血余炭50~100g、地骨皮90~160g、茜草60~100g、三七30~100g、延胡索(醋制)80~160g、甘草30~120g,本发明提供的药物是一个很好的中药组方。
Description
技术领域
本发明属于中药制剂领域,具体涉及一种可有效治疗消化性溃疡的内服药物,特别是供消化性溃疡患者使用的内服药物及其制备方法的领域。
背景技术
据相关资料显示:消化性溃疡主要指发生于胃和十二指肠的慢性溃疡,是一多发病、常见病。溃疡的形成有各种因素,其中酸性胃液对黏膜的消化作用是溃疡形成的基本因素,因此得名。酸性胃液接触的任何部位,如食管下段、胃肠吻合术后吻合口、空肠以及具有异位胃黏膜的Meckel憩室,绝大多数的溃疡发生于十二指肠和胃,故又称胃、十二指肠溃疡。
临床表现:
A.消化性溃疡疼痛特点
(a)长期性由于溃疡发生后可自行愈合,但每于愈合后又好复发,故常有上腹疼痛长期反复发作的特点。整个病程平均6~7年,有的可长达一、二十年,甚至更长。
(b)周期性上腹疼痛呈反复周期性发作,乃为此种溃疡的特征之一,尤以十二指肠溃疡更为突出。中上腹疼痛发作可持续几天、几周或更长,继以较长时间的缓解。全年都可发作,但以春、秋季节发作者多见。
(c)节律性溃疡疼痛与饮食之间的关系具有明显的相关性和节律性。在一天中,早晨3点至早餐的一段时间,胃酸分泌最低,故在此时间内很少发生疼痛。十二指肠溃疡的疼痛好在二餐之间发生,持续不减直至下餐进食或服制酸药物后缓解。一部分十二指肠溃疡病人,由于夜间的胃酸较高,尤其在睡前曾进餐者,可发生半夜疼痛。胃溃疡疼痛的发生较不规则,常在餐后1小时内发生,经1~2小时后逐渐缓解,直至下餐进食后再复出现上述节律。
(d)疼痛部位十二指肠溃疡的疼痛多出现于中上腹部,或在脐上方,或在脐上方偏右处;胃溃疡疼痛的位置也多在中上腹,但稍偏高处,或在剑突下和剑突下偏左处。疼痛范围约数厘米直径大小。因为空腔内脏的疼痛在体表上的定位一般不十分确切,所以,疼痛的部位也不一定准确反映溃疡所在解剖位置。
(e)疼痛性质多呈钝痛、灼痛或饥饿样痛,一般较轻而能耐受,持续性剧痛提示溃疡穿透或穿孔。
(f)影响因素疼痛常因精神刺激、过度疲劳、饮食不慎、药物影响、气候变化等因素诱发或加重;可因休息、进食、服制酸药、以手按压疼痛部位、呕吐等方法而减轻或缓解。
B.消化性溃疡其他症状与体征
(a)其他症状本病除中上腹疼痛外,尚可有唾液分泌增多、烧心、反胃、嗳酸、嗳气、恶心、呕吐等其他胃肠道症状。食欲多保持正常,但偶可因食后疼痛发作而惧食,以致体重减轻。全身症状可有失眠等神经官能症的表现,或有缓脉、多汗等植物神经系统不平衡的症状。
(b)体征溃疡发作期,中上腹部可有局限性压痛,程度不重,其压痛部位多与溃疡的位置基本相符。
那么,就如何找到一种可有效治疗消化性溃疡的中药组合物,是本领域技术人员亟待要解决的问题。
发明内容
随着我国中医中药学的不断发展,在治疗消化性溃疡上,人们逐渐意识到了中医治疗消化性溃疡的优点,且在治疗过程中疗效好、见效快、毒副作用小等优势,针对现有西医治疗消化性溃疡的现状,本发明的目的是在于提供一种可有效治疗消化性溃疡的内服药物,以解决消化性溃疡患者早日恢复健康的问题。该药物是以常见的中药为原料,通过选择合理的药物及其质量份比,可有效治疗上述消化性溃疡。
为达到上述发明的目的,本发明所采用的技术方案为:提供一种可有效治疗消化性溃疡的内服药物及其制备方法,其特征在于,所述药物的各个组分及其质量份比如下所示:
丹参90~180g、白芷50~160g、白术80~160g、党参150~280g、砂仁30~70g、干姜30~100g、玄参90~160g、肿节风90~350g、芡实90~160g、肉桂50~45g、人参30~100g、枳实30~100g、海螵蛸(炒黄)100~360g、木香15~70g、山楂30~120g、陈皮30~120g、蒲公英150~550g、苦杏仁45~90g、厚朴30~120g、青皮30~120g、蒲黄50~100g、地榆90~160g、血余炭50~100g、地骨皮90~160g、茜草60~100g、三七30~100g、延胡索(醋制)80~160g、甘草30~120g,辅料:微粉硅胶、微晶纤维素和淀粉适量。
一种可有效治疗消化性溃疡的内服药物及其制备方法,其特征在于,所述药物的各个组分及其质量份比如下所示:
丹参100~150g、白芷58~130g、白术90~130g、党参180~250g、砂仁38~60g、干姜38~90g、玄参100~130g、肿节风100~320g、芡实100~130g、肉桂58~42g、人参38~90g、枳实38~90g、海螵蛸(炒黄)115~320g、木香18~60g、山楂38~105g、陈皮35~105g、蒲公英180~480g、苦杏仁50~80g、厚朴38~105g、青皮38~105g、蒲黄58~90g、地榆100~130g、血余炭58~90g、地骨皮100~130g、茜草70~90g、三七38~90g、延胡索(醋制)90~130g、甘草38~105g,辅料:微粉硅胶、微晶纤维素和淀粉适量。
一种可有效治疗消化性溃疡的内服药物及其制备方法,其特征在于,所述药物的各个组分及其质量份比如下所示:
丹参130g、白芷115g、白术115g、党参220g、砂仁52g、干姜80g、玄参115g、肿节风260g、芡实115g、肉桂36g、人参80g、枳实80g、海螵蛸(炒黄)260g、木香52g、山楂95g、陈皮95g、蒲公英420g、苦杏仁70g、厚朴95g、青皮95g、蒲黄80g、地榆115g、血余炭80g、地骨皮115g、茜草80g、三七80g、延胡索(醋制)115g、甘草95g,辅料:微粉硅胶、微晶纤维素和淀粉适量。
一种可有效治疗消化性溃疡的内服药物及其制备方法,其特征在于,所述方法包括如下步骤制备而成:
A、除丹参、党参、玄参、人参和三七(研磨成细粉)外,将上述其它原料中药拣去杂质和粉尘后,按照质量份比共粉碎成(30~50目)颗粒状包煎;
B、①将包好的原料中药放入冷开水中浸泡60min,然后再将浸泡好的药物放入砂锅内,加入原料中药重量7~8 倍的冷开水进行第一次武火煎煮,待煎煮到18min时,转文火熬制120min,滤取药液;②药渣中再次加入原料中药重量6~7 倍的冷开水进行第二次武火煎煮,待煎煮到15min时,转文火熬制110min,滤取药液;③将两次药液混合浓缩成相对密度为1.08 的清膏,然后干燥、研末和消毒后备用;
C、①按照传统制备中药胶囊剂的方法,将A 和B中研磨好的细末过筛后,加入适量的微粉硅胶、微晶纤维素和淀粉混合均匀,然后制备成胶囊(其胶囊锁合后总长度为23.3mm,药粉容量0.4~0.5g/粒),②继而抛光、消毒,分装密封即可。
一种可有效治疗消化性溃疡的内服药物及其制备方法,其特征在于,所述服用方法为:将制备好的胶囊剂药物以每日三次服用,早中晚各服一次,给药量2.5g(5粒)/次,饭后温开水送服。30天为一个疗程,服药3~6个疗程,消化性溃疡症状明显好转或痊愈,已随访一年余,未再见复发。
本发明组方中的各原料中药在中国药典、中国辞典以及其中华本草中均有详细的记载。本发明选用其中最常见的中药为原料,充分发挥各组分的药理功效:
丹参,性味:苦、微寒,具有祛瘀止痛、活血通经、清心除烦之功效,用于治疗月经不调、经闭痛经、症瘕积聚、胸腹刺痛、热痹疼痛、疮疡肿痛、心烦不眠、肝脾肿大、心绞痛;
白芷,性味:性温、味辛、气芳香、微苦,具有祛风湿、活血排脓、生肌止痛之功效,用于治疗头痛、牙痛、鼻渊、肠风痔漏、赤白带下、痈疽疮疡、皮肤瘙痒;
白术,性味:味苦、甘、性温,具有健脾益气、燥湿利水、止汗、安胎之功效,用于治疗脾气虚弱、神疲乏力、食少少腹胀、大便溏薄、水饮内停、小便不利、水肿、痰饮眩晕、温痹酸痛、气虚自汗、胎动不安等症;
党参,性味:味甘、性平,具有健脾补肺、益气生津之功效,用于治疗脾胃虚弱、食少便溏、四肢乏力、肺虚喘咳、气短自汗、气微两亏等症;
砂仁,性味:味辛、性温,具有化湿开胃、行气宽中温脾止泻安胎之功效,用于治疗湿阻气滞、脘腹胀满、不思饮食、恶心呕吐、腹痛泄泻妊娠恶阻、胎动不安;
干姜,性味:辛、热,具有温中散寒、回阳通脉、燥湿消痰之功效,用于治疗脘腹冷痛、呕吐泄泻、肢冷脉微、痰饮喘咳;
玄参,性味:甘、苦、咸、微寒,具有凉血滋阴、泻火解毒之功效,用于治疗热病伤阴、舌绛烦渴、温毒发斑、津伤便秘、骨蒸劳嗽、目赤、咽痛、瘰疠、白喉、痈肿疮毒;
肿节风,性味:苦、辛、平,具有清热凉血、活血消斑、祛风通络之功效,用于治疗血热紫斑、紫癜、风湿痹痛、跌打损伤;
芡实,性味:甘、涩、平,具有益肾固精、补脾止泻、祛湿止带之功效,用于治疗梦遗滑精、遗尿尿频、脾虚久泻、白浊、带下等病症;
肉桂,性味:辛、甘,大热,具有补火助阳、引火归源、散寒止痛、活血通经之功效,用于治疗阳痿、宫冷、腰膝冷痛、肾虚作喘、阳虚眩晕、目赤咽痛、心腹冷痛、虚寒吐泻、寒疝、奔豚、经闭、痛经等症;
人参,性味:甘、微苦、平,具有大补元气、复脉固脱、补脾益肺、生津、安神之功效,用于治疗体虚欲脱、肢冷脉微、脾虚食少、肺虚喘咳、津伤口渴、内热消渴、久病虚羸、惊悸失眠、阳痿宫冷、心力衰竭、心原性休克;
枳实,性味:苦、辛、酸、温,具有破气消积、化痰散痞之功效,用于治疗积滞内停、痞满胀痛、泻痢后重、大便不通、痰滞气阻胸痹、结胸、胃下垂、脱肛、子宫脱垂;
海螵蛸(炒黄),性味:味咸、涩、性温,具有收敛止血、固精止带、制酸止痛、收湿敛疮之功效,用于治疗吐血、呕血、崩漏、便血、衄血、创伤出血、肾虚遗精滑精、赤白带下、胃痛嘈杂、嗳气泛酸、湿疹溃疡;
木香,性味:辛、苦、温,具有行气止痛、健脾消食之功效,用于治疗胸脘胀痛、泻痢后重、食积不消、不思饮食,煨木香实肠止泻,用于泄泻腹痛;
山楂,性味:酸甘、微温、无毒,具有消食积、化滞瘀之功效,用于治疗饮食积滞、脘腹胀痛、泄泻痢疾、血瘀痛经、闭经、产后腹痛、恶露不尽;
陈皮,性味:苦、辛、温,具有理气健脾、调中、燥湿、化痰之功效,用于治疗脾胃气滞之脘腹胀满或疼痛、消化不良、湿浊阻中之胸闷腹胀、纳呆便溏、痰湿壅肺之咳嗽气喘、食少吐泻、咳嗽痰多等症;
蒲公英,性味:味苦;甘、性寒,具有清热解毒、消痈散结之功效,用于治疗乳痈、肺痈、肠痈、痄腮、疔毒疮肿、目赤肿痛、感冒发热、咳嗽、咽喉肿痛、胃火、肠炎、痢疾、肝炎、胆吓炎、尿路感染、蛇虫咬伤;
苦杏仁,性味:苦、微温,有小毒,具有降气止咳平喘、润肠通便之功效,用于治疗咳嗽气喘、胸满痰多、血虚津枯、肠燥便秘;
厚朴,性味:苦、辛、性温,具有行气消积、燥湿除满、降逆平喘之功效,用于治疗食积气滞、腹胀便秘、湿阻中焦、脘痞吐泻、痰壅气逆、胸满喘咳;
青皮,性味:苦、辛、温,具有疏肝破气、消积化滞之功效,用于治疗肝郁气滞之胁肋胀痛、乳房胀痛、乳核、乳痈、疝气疼痛、食积气滞之胃脘胀痛、以及气滞血瘀所至的癥瘕积聚、久疟癖块;
蒲黄,性味:甘、平,具有止血、化瘀、通淋之功效,用于治疗吐血、衄血、咯血、崩漏、外伤出血、经闭痛经、脘腹刺痛、跌扑肿痛、血淋涩痛;
地榆,性味:苦、酸、涩、微寒,具有凉血止血、解毒敛疮之功效,用于治疗便血、痔血、血痢、崩漏、水火烫伤、痈肿疮毒;
血余炭,性味:苦、平,具有止血、化瘀之功效,用于治疗吐血、咯血、衄血、尿血、崩漏下血、外伤出血;
地骨皮,性味:甘、寒,具有凉血除蒸、清肺降火之功效,用于治疗阴虚潮热、骨蒸盗汗、肺热咳嗽、咯血、衄血、内热消渴;
茜草,性味:苦、寒,具有凉血、止血、祛瘀、通经之功效,用于治疗吐血、衄血、崩漏、外伤出血、经闭瘀阻、关节痹痛、跌扑肿痛;
三七,性味:甘、微苦、温,具有散瘀止血、消肿定痛之功效,用于治疗咯血、吐血、衄血、便血、崩漏、外伤出血、胸腹刺痛、跌扑肿痛等症;
延胡索(醋制),性味:辛、苦、温,无毒,具有活血、散瘀、理气、止痛之功效,用于治疗心腹腰膝诸痛、月经不调、症瘕、崩中、产后血晕、恶露不尽、跌打损伤;
甘草,性味:甘、平,具有益气补中、缓急止痛、润肺止咳、泻火解毒、调和诸药之功效,用于治疗倦怠食少、肌瘦面黄、心悸气短、腹痛便溏、四肢挛急疼痛、脏躁、咳嗽气喘、咽喉肿痛、痈疮肿痛、小儿胎毒及药物、食物中毒。
本发明药物是基于中医治疗消化性溃疡的原则,从依据消化性溃疡的病理机制及药理作用认为:就消化性溃疡,本发明所提供的药物中的各原料中药药效共奏,对上述疾病有很好的效果。
具体实施方式
本发明就是针对上述消化性溃疡的治疗而提出的一种中药配方,采用该配方制备的药物药效好,见效快,是一个很好的中药组方,特别适合临床使用。下面结合本发明的具体实施方式作进一步详细的描述:
实施例1:
一种可有效治疗消化性溃疡的内服药物,其特征在于,所述药物的各个组分及其质量份比如下所示:
丹参130g、白芷115g、白术115g、党参220g、砂仁52g、干姜80g、玄参115g、肿节风260g、芡实115g、肉桂36g、人参80g、枳实80g、海螵蛸(炒黄)260g、木香52g、山楂95g、陈皮95g、蒲公英420g、苦杏仁70g、厚朴95g、青皮95g、蒲黄80g、地榆115g、血余炭80g、地骨皮115g、茜草80g、三七80g、延胡索(醋制)115g、甘草95g,辅料:微粉硅胶、微晶纤维素和淀粉适量。
实施例2:
一种可有效治疗消化性溃疡的内服药物,其特征在于,所述药物的各个组分及其质量份比如下所示:
丹参150g、白芷130g、白术130g、党参250g、砂仁60g、干姜90g、玄参130g、肿节风320g、芡实130g、肉桂42g、人参90g、枳实90g、海螵蛸(炒黄)320g、木香60g、山楂105g、陈皮105g、蒲公英480g、苦杏仁80g、厚朴105g、青皮105g、蒲黄90g、地榆130g、血余炭90g、地骨皮130g、茜草90g、三七90g、延胡索(醋制)130g、甘草105g,辅料:微粉硅胶、微晶纤维素和淀粉适量。
实施例3:
一种可有效治疗消化性溃疡的内服药物,其特征在于,所述药物的各个组分及其质量份比如下所示:
丹参180g、白芷160g、白术160g、党参280g、砂仁70g、干姜100g、玄参160g、肿节风350g、芡实160g、肉桂45g、人参100g、枳实100g、海螵蛸(炒黄)360g、木香70g、山楂120g、陈皮120g、蒲公英550g、苦杏仁90g、厚朴120g、青皮120g、蒲黄100g、地榆160g、血余炭100g、地骨皮160g、茜草100g、三七100g、延胡索(醋制)160g、甘草120g,辅料:微粉硅胶、微晶纤维素和淀粉适量。
典型病例
经临床诊断治疗消化性溃疡患者共1300例,年龄为46岁以上的705例,只有595例为46岁以下。1300例患者中痊愈的805例,有效的443例,无效的52例。总有效率达96%。
Claims (3)
1.一种可有效治疗消化性溃疡的内服药物,其特征在于,所述药物的各个组分及其质量份比如下所示:
丹参90~180g、白芷50~160g、白术80~160g、党参150~280g、砂仁30~70g、干姜30~100g、玄参90~160g、肿节风90~350g、芡实90~160g、肉桂50~45g、人参30~100g、枳实30~100g、海螵蛸(炒黄)100~360g、木香15~70g、山楂30~120g、陈皮30~120g、蒲公英150~550g、苦杏仁45~90g、厚朴30~120g、青皮30~120g、蒲黄50~100g、地榆90~160g、血余炭50~100g、地骨皮90~160g、茜草60~100g、三七30~100g、延胡索(醋制)80~160g、甘草30~120g,辅料:微粉硅胶、微晶纤维素和淀粉适量。
2.根据权利要求1所述的可有效治疗消化性溃疡的内服药物,其特征在于,所述药物的各个组分及其质量份比如下所示:
丹参100~150g、白芷58~130g、白术90~130g、党参180~250g、砂仁38~60g、干姜38~90g、玄参100~130g、肿节风100~320g、芡实100~130g、肉桂58~42g、人参38~90g、枳实38~90g、海螵蛸(炒黄)115~320g、木香18~60g、山楂38~105g、陈皮35~105g、蒲公英180~480g、苦杏仁50~80g、厚朴38~105g、青皮38~105g、蒲黄58~90g、地榆100~130g、血余炭58~90g、地骨皮100~130g、茜草70~90g、三七38~90g、延胡索(醋制)90~130g、甘草38~105g,辅料:微粉硅胶、微晶纤维素和淀粉适量。
3.根据权利要求1至2所述的可有效治疗消化性溃疡的内服药物,其特征在于,所述药物的各个组分及其质量份比如下所示:
丹参130g、白芷115g、白术115g、党参220g、砂仁52g、干姜80g、玄参115g、肿节风260g、芡实115g、肉桂36g、人参80g、枳实80g、海螵蛸(炒黄)260g、木香52g、山楂95g、陈皮95g、蒲公英420g、苦杏仁70g、厚朴95g、青皮95g、蒲黄80g、地榆115g、血余炭80g、地骨皮115g、茜草80g、三七80g、延胡索(醋制)115g、甘草95g,辅料:微粉硅胶、微晶纤维素和淀粉适量。
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