CN103003273A - 吡唑并吡啶激酶抑制剂 - Google Patents
吡唑并吡啶激酶抑制剂 Download PDFInfo
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Landscapes
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US29865310P | 2010-01-27 | 2010-01-27 | |
| US61/298,653 | 2010-01-27 | ||
| PCT/US2011/022536 WO2011094283A1 (en) | 2010-01-27 | 2011-01-26 | Pyrazolopyridine kinase inhibitors |
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|---|---|
| CN103003273A true CN103003273A (zh) | 2013-03-27 |
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| WO (1) | WO2011094283A1 (enExample) |
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| MX2012008642A (es) * | 2010-01-27 | 2012-11-23 | Vertex Pharma | Inhibidores de cinasas de pirazolopiridinas. |
| CN102858769A (zh) * | 2010-01-27 | 2013-01-02 | 沃泰克斯药物股份有限公司 | 吡唑并吡啶激酶抑制剂 |
| US10124001B2 (en) | 2013-09-18 | 2018-11-13 | University Of Canberra | Stem cell modulation II |
| JP2017528452A (ja) | 2014-08-25 | 2017-09-28 | ユニバーシティ・オブ・キャンベラＵｎｉｖｅｒｓｉｔｙ ｏｆ Ｃａｎｂｅｒｒａ | がん幹細胞を調節するための組成物およびその使用 |
| WO2025097025A1 (en) * | 2023-11-03 | 2025-05-08 | Evommune, Inc. | Protein kinase c (pkc) theta inhibitor compounds |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2005095400A1 (en) * | 2004-03-30 | 2005-10-13 | Vertex Pharmaceuticals Incorporated | Azaindoles useful as inhibitors of jak and other protein kinases |
| WO2009073300A1 (en) * | 2007-11-02 | 2009-06-11 | Vertex Pharmaceuticals Incorporated | [1h- pyrazolo [3, 4-b] pyridine-4-yl] -phenyle or -pyridin-2-yle derivatives as protein kinase c-theta |
| CN102159574A (zh) * | 2008-07-23 | 2011-08-17 | 沃泰克斯药物股份有限公司 | 三-环吡唑并吡啶激酶抑制剂 |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20030187026A1 (en) * | 2001-12-13 | 2003-10-02 | Qun Li | Kinase inhibitors |
| AU2005269387A1 (en) * | 2004-07-27 | 2006-02-09 | Sgx Pharmaceuticals, Inc. | Fused ring heterocycle kinase modulators |
| EP1814882A1 (en) * | 2004-11-22 | 2007-08-08 | Vertex Pharmaceuticals Incorporated | Pyrrolopyrazines and pyrazolopyrazines useful as inhibitors of protein kinases |
| NZ567133A (en) * | 2005-09-30 | 2011-07-29 | Vertex Pharma | Deazapurines useful as inhibitors of janus kinases |
| DE102006029447A1 (de) * | 2006-06-21 | 2007-12-27 | Bayer Schering Pharma Ag | Oxo-substituierte Imidazo[1,2b]pyridazine, deren Herstellung und Verwendung als Arzneimittel |
| MX2009012066A (es) * | 2007-05-09 | 2009-11-19 | Novartis Ag | Imidazopirinas sustituidas como inhibidoras de cinasa de lipido p13k. |
| JP4946728B2 (ja) | 2007-08-23 | 2012-06-06 | 三菱電機株式会社 | 電力増幅器 |
| EP2328896B1 (en) * | 2008-07-23 | 2013-10-23 | Vertex Pharmaceuticals Incorporated | Tri-cyclic pyrazolopyridine kinase inhibitors |
| US8569337B2 (en) * | 2008-07-23 | 2013-10-29 | Vertex Pharmaceuticals Incorporated | Tri-cyclic pyrazolopyridine kinase inhibitors |
| JP5542287B2 (ja) * | 2008-07-23 | 2014-07-09 | バーテックス ファーマシューティカルズ インコーポレイテッド | ピラゾロピリジンキナーゼ阻害剤 |
| KR20110039563A (ko) * | 2008-07-23 | 2011-04-19 | 버텍스 파마슈티칼스 인코포레이티드 | 피라졸로피리딘 키나제 억제제 |
| MX2012008642A (es) * | 2010-01-27 | 2012-11-23 | Vertex Pharma | Inhibidores de cinasas de pirazolopiridinas. |
| CN102858769A (zh) * | 2010-01-27 | 2013-01-02 | 沃泰克斯药物股份有限公司 | 吡唑并吡啶激酶抑制剂 |
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2011
- 2011-01-26 MX MX2012008642A patent/MX2012008642A/es active IP Right Grant
- 2011-01-26 JP JP2012551252A patent/JP2013518112A/ja not_active Withdrawn
- 2011-01-26 WO PCT/US2011/022536 patent/WO2011094283A1/en not_active Ceased
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- 2011-01-26 CA CA2787321A patent/CA2787321A1/en not_active Abandoned
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- 2011-01-26 EP EP11703771A patent/EP2528916A1/en not_active Withdrawn
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2012
- 2012-07-27 US US13/560,119 patent/US20130053395A1/en not_active Abandoned
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2005095400A1 (en) * | 2004-03-30 | 2005-10-13 | Vertex Pharmaceuticals Incorporated | Azaindoles useful as inhibitors of jak and other protein kinases |
| WO2009073300A1 (en) * | 2007-11-02 | 2009-06-11 | Vertex Pharmaceuticals Incorporated | [1h- pyrazolo [3, 4-b] pyridine-4-yl] -phenyle or -pyridin-2-yle derivatives as protein kinase c-theta |
| CN102159574A (zh) * | 2008-07-23 | 2011-08-17 | 沃泰克斯药物股份有限公司 | 三-环吡唑并吡啶激酶抑制剂 |
Also Published As
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| JP2013518112A (ja) | 2013-05-20 |
| CA2787321A1 (en) | 2011-08-04 |
| EP2528916A1 (en) | 2012-12-05 |
| US20130053395A1 (en) | 2013-02-28 |
| AU2011209644A1 (en) | 2012-08-09 |
| WO2011094283A1 (en) | 2011-08-04 |
| MX2012008642A (es) | 2012-11-23 |
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