CN101854908B - 用于化妆品和其他应用的c-19甾族化合物 - Google Patents

用于化妆品和其他应用的c-19甾族化合物 Download PDF

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Publication number
CN101854908B
CN101854908B CN2008801158388A CN200880115838A CN101854908B CN 101854908 B CN101854908 B CN 101854908B CN 2008801158388 A CN2008801158388 A CN 2008801158388A CN 200880115838 A CN200880115838 A CN 200880115838A CN 101854908 B CN101854908 B CN 101854908B
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CN
China
Prior art keywords
skin
hydrogen
hair
glands
dht
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
CN2008801158388A
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English (en)
Chinese (zh)
Other versions
CN101854908A (zh
Inventor
马丁·温迪施
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Atai Nin Ltd
Original Assignee
Erlacos GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erlacos GmbH filed Critical Erlacos GmbH
Publication of CN101854908A publication Critical patent/CN101854908A/zh
Application granted granted Critical
Publication of CN101854908B publication Critical patent/CN101854908B/zh
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/63—Steroids; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/14—Drugs for dermatological disorders for baldness or alopecia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q15/00—Anti-perspirants or body deodorants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00—Preparations for care of the skin
    • A61Q19/06—Preparations for care of the skin for countering cellulitis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00—Preparations for care of the skin
    • A61Q19/08—Anti-ageing preparations
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q7/00—Preparations for affecting hair growth
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q7/00—Preparations for affecting hair growth
    • A61Q7/02—Preparations for inhibiting or slowing hair growth
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1617—Organic compounds, e.g. phospholipids, fats
    • A61K9/1623—Sugars or sugar alcohols, e.g. lactose; Derivatives thereof; Homeopathic globules
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Dermatology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Birds (AREA)
  • Gerontology & Geriatric Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Cosmetics (AREA)
CN2008801158388A 2007-11-13 2008-11-12 用于化妆品和其他应用的c-19甾族化合物 Expired - Fee Related CN101854908B (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US288207P 2007-11-13 2007-11-13
US61/002,882 2007-11-13
EP07022015.7 2007-11-13
EP07022015.7A EP2060261B1 (en) 2007-11-13 2007-11-13 C-19 steroids for cosmetic uses
PCT/EP2008/009540 WO2009062682A1 (en) 2007-11-13 2008-11-12 C-19 steroids for cosmetic and further uses

Publications (2)

Publication Number Publication Date
CN101854908A CN101854908A (zh) 2010-10-06
CN101854908B true CN101854908B (zh) 2013-03-06

Family

ID=39198683

Family Applications (1)

Application Number Title Priority Date Filing Date
CN2008801158388A Expired - Fee Related CN101854908B (zh) 2007-11-13 2008-11-12 用于化妆品和其他应用的c-19甾族化合物

Country Status (10)

Country Link
US (1) US8258123B2 (enExample)
EP (2) EP2060261B1 (enExample)
JP (1) JP2011503129A (enExample)
KR (2) KR20100087005A (enExample)
CN (1) CN101854908B (enExample)
AU (1) AU2008323198B2 (enExample)
CA (1) CA2705529C (enExample)
DK (1) DK2060261T3 (enExample)
ES (1) ES2574933T3 (enExample)
WO (1) WO2009062682A1 (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2060300B1 (en) * 2007-11-13 2015-04-15 Curadis GmbH C-19 steroids for therapeutic uses
US11850451B2 (en) 2011-01-31 2023-12-26 Lucolas-M.D. Ltd. Cosmetic compositions and methods for improving skin conditions
JP5872806B2 (ja) * 2011-07-07 2016-03-01 花王株式会社 Ｍｆａｐ−４産生促進剤
EP2574329A1 (en) 2011-09-28 2013-04-03 ErlaCos GmbH Deodorant comprising dimethyl isosorbide
JP5980512B2 (ja) * 2012-01-30 2016-08-31 学校法人東日本学園 体臭抑制剤
JP6145181B2 (ja) * 2016-01-14 2017-06-07 花王株式会社 Ｍｆａｐ−４産生促進剤
MX383946B (es) * 2016-08-03 2025-03-14 Colgate Palmolive Co Agente activo y método para reducir el mal olor.
FR3094229B1 (fr) 2019-03-28 2021-11-12 Roquette Freres Composition topique pour le traitement des mauvaises odeurs corporelles, notamment l’halitose

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1992007586A1 (en) * 1990-10-31 1992-05-14 Beecham Group Plc Topical composition with retinoid penetration enhancer
WO2006084312A1 (en) * 2005-02-09 2006-08-17 Acrux Dds Pty Ltd Method of promoting hair growth

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2763818A (en) * 1954-10-14 1956-09-18 Westinghouse Electric Corp Lighting arrester
US2762818A (en) 1955-05-26 1956-09-11 Searle & Co 4-hydroxytestosterone and esters thereof
ZA843232B (en) * 1983-05-03 1984-12-24 Bristol Myers Co Antiperspirant stick with low staining potential
JPS62132810A (ja) * 1985-12-05 1987-06-16 Shiseido Co Ltd 化粧料
GB8721384D0 (en) * 1987-09-11 1987-10-21 Erba Farmitalia 17-substituted andro-sta-1 4-dien-3-one derivatives
GB9021546D0 (en) 1990-10-04 1990-11-21 Beecham Group Plc Novel composition
US5486511A (en) 1993-05-25 1996-01-23 Merrell Dow Pharmaceuticals Inc. 4-amino-17β-(cyclopropyloxy)androst-4-en-3-one, 4-amino-17β-(cyclopropylamino)androst-4-en-3-one and related compounds as C17-20 lyase and 5α-reductase
DE4405898A1 (de) 1994-02-18 1995-08-24 Schering Ag Transdermale therapeutische Systeme enthaltend Sexualsteroide
DE69519582D1 (de) * 1994-09-14 2001-01-11 Univ Sheffield Kontrolle des haarwuchses
US5824326A (en) * 1997-06-27 1998-10-20 Chesebrough-Pond's Usa Co., Division Of Conopco, Inc. Activity enhancement of ferulic acid with dimethyl isosorbride in cosmetic compositions
EP1429779A2 (en) 2001-09-21 2004-06-23 Merck & Co., Inc. Androstanes as androgen receptor modulators
US6586417B1 (en) * 2002-04-22 2003-07-01 Nutrisport Pharmacal, Inc. Ester and ether derivatives of 4-hydroxy 4-androstene-3,17-dione and a method for the regulation of athletic function in humans
US20030199487A1 (en) * 2002-04-22 2003-10-23 Mr. Vince Paternoster Ester and ether derivatives of 4-hydroxytestosterone and a method for the regulation of athletic function in humans
US20030229063A1 (en) * 2002-06-05 2003-12-11 Llewellyn William Charles Use of 4-hydroxytestosterone to lower estrogen levels in humans
US20060018937A1 (en) * 2002-10-25 2006-01-26 Foamix Ltd. Steroid kit and foamable composition and uses thereof
EP1689864A2 (en) * 2003-10-21 2006-08-16 Dyad Pharmaceutical Corporation Method and compositions for treating 5alpha-reductase type 1 and type 2 dependent conditions
EP1692317A4 (en) 2003-12-12 2007-12-19 Univ Rochester Non-androgen dependent roles for androgen receptor and non-androgen related inhibitors of androgen receptor
JP4755845B2 (ja) * 2005-04-28 2011-08-24 共栄化学工業株式会社 テストステロン−５α−リダクターゼ阻害剤及びテストステロン−５α−リダクターゼ阻害剤を含有する化粧料。
EP1854465A1 (en) * 2006-05-12 2007-11-14 Alexander Tobias Teichmann Use of 4,17 beta-dihydroxyandrost-4-ene-3-one for treating cancers

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1992007586A1 (en) * 1990-10-31 1992-05-14 Beecham Group Plc Topical composition with retinoid penetration enhancer
WO2006084312A1 (en) * 2005-02-09 2006-08-17 Acrux Dds Pty Ltd Method of promoting hair growth

Also Published As

Publication number Publication date
KR20100087005A (ko) 2010-08-02
ES2574933T3 (es) 2016-06-23
KR20160036098A (ko) 2016-04-01
CA2705529A1 (en) 2009-05-22
CN101854908A (zh) 2010-10-06
JP2011503129A (ja) 2011-01-27
US8258123B2 (en) 2012-09-04
DK2060261T3 (en) 2016-06-13
EP2207523A1 (en) 2010-07-21
EP2060261B1 (en) 2016-03-09
KR101776544B1 (ko) 2017-09-07
CA2705529C (en) 2016-10-11
EP2060261A1 (en) 2009-05-20
AU2008323198A1 (en) 2009-05-22
US20100256102A1 (en) 2010-10-07
WO2009062682A1 (en) 2009-05-22
HK1148669A1 (en) 2011-09-16
AU2008323198B2 (en) 2014-03-20

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