CN101824005A - 一种非布索坦的新晶型q及其制备方法 - Google Patents
一种非布索坦的新晶型q及其制备方法 Download PDFInfo
- Publication number
- CN101824005A CN101824005A CN 201010157944 CN201010157944A CN101824005A CN 101824005 A CN101824005 A CN 101824005A CN 201010157944 CN201010157944 CN 201010157944 CN 201010157944 A CN201010157944 A CN 201010157944A CN 101824005 A CN101824005 A CN 101824005A
- Authority
- CN
- China
- Prior art keywords
- febuxostat
- crystal form
- preparation
- crystal
- solvent
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Images
Abstract
Description
Claims (6)
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CN2010101579441A CN101824005B (zh) | 2010-04-27 | 2010-04-27 | 一种非布索坦的晶型q及其制备方法 |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CN2010101579441A CN101824005B (zh) | 2010-04-27 | 2010-04-27 | 一种非布索坦的晶型q及其制备方法 |
Publications (2)
Publication Number | Publication Date |
---|---|
CN101824005A true CN101824005A (zh) | 2010-09-08 |
CN101824005B CN101824005B (zh) | 2012-06-27 |
Family
ID=42688195
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CN2010101579441A Expired - Fee Related CN101824005B (zh) | 2010-04-27 | 2010-04-27 | 一种非布索坦的晶型q及其制备方法 |
Country Status (1)
Country | Link |
---|---|
CN (1) | CN101824005B (zh) |
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2016091230A1 (en) | 2014-12-12 | 2016-06-16 | Zentiva, K.S. | Formulations containing a solid solution of febuxostat |
CN107540630A (zh) * | 2016-06-29 | 2018-01-05 | 康普药业股份有限公司 | 一种非布司他化合物及制备方法 |
Citations (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1999065885A1 (en) * | 1998-06-19 | 1999-12-23 | Teijin Limited | Polymorphic modifications of 2-(3-cyano-4-isobutyloxyphenyl)-4-methyl-5-thiazole-carboxylic acid and processes for the preparation thereof |
WO2003082279A1 (fr) * | 2002-03-28 | 2003-10-09 | Teijin Limited | Preparation solide contenant une forme monocristalline |
CN1970547A (zh) * | 2006-12-07 | 2007-05-30 | 重庆医药工业研究院有限责任公司 | 非布司他的新晶型及其制备方法 |
CN101085761A (zh) * | 2007-06-29 | 2007-12-12 | 上海华拓医药科技发展股份有限公司 | 非布他特微晶及其组合物 |
CN101139325A (zh) * | 2006-09-07 | 2008-03-12 | 上海医药工业研究院 | 2-(3-氰基-4-异丁氧基苯基)-4-甲基-5-噻唑甲酸晶型及其制备方法 |
CN101386605A (zh) * | 2008-10-23 | 2009-03-18 | 中国科学院上海药物研究所 | 非布司他新型晶体及其制备方法 |
CN101671315A (zh) * | 2009-08-19 | 2010-03-17 | 何广卫 | 非布索坦的新晶型及其制备方法 |
CN101671314A (zh) * | 2009-09-17 | 2010-03-17 | 中国药科大学 | 一种非布索坦的晶型体及制备方法 |
CN101684107A (zh) * | 2008-09-26 | 2010-03-31 | 上海优拓医药科技有限公司 | 非布索坦的新晶型及其制备方法 |
-
2010
- 2010-04-27 CN CN2010101579441A patent/CN101824005B/zh not_active Expired - Fee Related
Patent Citations (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1999065885A1 (en) * | 1998-06-19 | 1999-12-23 | Teijin Limited | Polymorphic modifications of 2-(3-cyano-4-isobutyloxyphenyl)-4-methyl-5-thiazole-carboxylic acid and processes for the preparation thereof |
CN1275126A (zh) * | 1998-06-19 | 2000-11-29 | 帝人株式会社 | 2-(3-氰基-4-异丁氧基苯基)-4-甲基-5-噻唑甲酸的多晶型体及其制备方法 |
WO2003082279A1 (fr) * | 2002-03-28 | 2003-10-09 | Teijin Limited | Preparation solide contenant une forme monocristalline |
CN101139325A (zh) * | 2006-09-07 | 2008-03-12 | 上海医药工业研究院 | 2-(3-氰基-4-异丁氧基苯基)-4-甲基-5-噻唑甲酸晶型及其制备方法 |
CN1970547A (zh) * | 2006-12-07 | 2007-05-30 | 重庆医药工业研究院有限责任公司 | 非布司他的新晶型及其制备方法 |
CN101085761A (zh) * | 2007-06-29 | 2007-12-12 | 上海华拓医药科技发展股份有限公司 | 非布他特微晶及其组合物 |
CN101684107A (zh) * | 2008-09-26 | 2010-03-31 | 上海优拓医药科技有限公司 | 非布索坦的新晶型及其制备方法 |
CN101386605A (zh) * | 2008-10-23 | 2009-03-18 | 中国科学院上海药物研究所 | 非布司他新型晶体及其制备方法 |
CN101671315A (zh) * | 2009-08-19 | 2010-03-17 | 何广卫 | 非布索坦的新晶型及其制备方法 |
CN101671314A (zh) * | 2009-09-17 | 2010-03-17 | 中国药科大学 | 一种非布索坦的晶型体及制备方法 |
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2016091230A1 (en) | 2014-12-12 | 2016-06-16 | Zentiva, K.S. | Formulations containing a solid solution of febuxostat |
CN107540630A (zh) * | 2016-06-29 | 2018-01-05 | 康普药业股份有限公司 | 一种非布司他化合物及制备方法 |
Also Published As
Publication number | Publication date |
---|---|
CN101824005B (zh) | 2012-06-27 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CN101139325B (zh) | 2-(3-氰基-4-异丁氧基苯基)-4-甲基-5-噻唑甲酸晶型及其制备方法 | |
CN102827153B (zh) | 阿齐沙坦的晶型及其制备方法 | |
AU2011312042B2 (en) | Methods of making L-ornithine phenyl acetate | |
JP2006151999A5 (zh) | ||
JP2009084270A5 (zh) | ||
CA2546701A1 (en) | Crystalline ammonium salts of rosuvastatin | |
CN102421432A (zh) | L-鸟氨酸苯乙酸盐及其制备方法 | |
CN103951634B (zh) | 一种依帕司他结晶盐水合物和羟基哌啶共晶物及其制备方法和应用 | |
JP5303765B2 (ja) | 結晶性イミダゾール−5−カルボン酸誘導体 | |
CN101824005B (zh) | 一种非布索坦的晶型q及其制备方法 | |
KR20210095238A (ko) | 무정형 형태의 akt 저해성 피리미디닐 - 사이클로펜탄 화합물, 조성물 및 이들의 방법 | |
CN103965116A (zh) | 半5-氟胞嘧啶盐、其制备方法及应用 | |
CN101824007A (zh) | 一种非布索坦的新晶型m及其制备方法 | |
CN101824006A (zh) | 一种非布索坦的新晶型p及其制备方法 | |
CN103880829B (zh) | 一种阿齐沙坦晶体及其制备方法和用途 | |
CN104610195A (zh) | 沃替西汀的天冬氨酸盐或其水合物及其制备方法和用途 | |
CO5780134A1 (es) | Forma polimorfica de descetoprofeno trometamol, su preparacion y composiciones que lo contienen | |
TWI705065B (zh) | 嗎啉衍生物的鹽及其晶型、其製備方法及藥物組成物、用途 | |
CN101328138B (zh) | 甲氧苄啶的制备方法 | |
WO2011134101A1 (zh) | 一种非布索坦的新晶型n及其制备方法 | |
RU2019106531A (ru) | Кристалл соли производного хиназолина | |
CA2608087A1 (en) | Methods for synthesizing heterocyclic compounds | |
CN104292232A (zh) | 一种培美曲塞二钠的杂质a的中间体的合成方法 | |
JP2010516756A (ja) | アトルバスタチンのストロンチウム塩、及びこれを含む医薬組成物 | |
ES2356501T3 (es) | Procedimiento para la preparación de zolmitriptan. |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
C06 | Publication | ||
PB01 | Publication | ||
C10 | Entry into substantive examination | ||
SE01 | Entry into force of request for substantive examination | ||
C14 | Grant of patent or utility model | ||
GR01 | Patent grant | ||
ASS | Succession or assignment of patent right |
Owner name: ZHOU HANG Free format text: FORMER OWNER: SHANGHAI KAIMINONG PHARMACEUTICAL TECHNOLOGY CO., LTD. Effective date: 20120531 |
|
C41 | Transfer of patent application or patent right or utility model | ||
COR | Change of bibliographic data |
Free format text: CORRECT: ADDRESS; FROM: 201203 PUDONG NEW AREA, SHANGHAI TO: 210018 NANJING, JIANGSU PROVINCE |
|
TR01 | Transfer of patent right |
Effective date of registration: 20120531 Address after: 210018, Xuanwu District, Nanjing Cheng Yin Street, No. 119 Patentee after: Zhou Hang Address before: 201203 Shanghai city Pudong New Area Cailun Road Lane 720 Building No. 1 room 512 Patentee before: Cheminno (Shanghai) Co., Ltd. |
|
C17 | Cessation of patent right | ||
CF01 | Termination of patent right due to non-payment of annual fee |
Granted publication date: 20120627 Termination date: 20130427 |