CL2023000823A1 - Métodos para tratar trastornos asociados a la vía del receptor de melanocortina 4 - Google Patents

Métodos para tratar trastornos asociados a la vía del receptor de melanocortina 4

Info

Publication number
CL2023000823A1
CL2023000823A1 CL2023000823A CL2023000823A CL2023000823A1 CL 2023000823 A1 CL2023000823 A1 CL 2023000823A1 CL 2023000823 A CL2023000823 A CL 2023000823A CL 2023000823 A CL2023000823 A CL 2023000823A CL 2023000823 A1 CL2023000823 A1 CL 2023000823A1
Authority
CL
Chile
Prior art keywords
melanocortin
methods
disorders associated
treat disorders
receptor pathway
Prior art date
Application number
CL2023000823A
Other languages
English (en)
Inventor
H T Van Der Ploeg Leonardus
Garfield Alastair
P Shah Bhavik
Original Assignee
Rhythm Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhythm Pharmaceuticals Inc filed Critical Rhythm Pharmaceuticals Inc
Publication of CL2023000823A1 publication Critical patent/CL2023000823A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Gastroenterology & Hepatology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Child & Adolescent Psychology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hematology (AREA)
  • Dermatology (AREA)
  • Organic Chemistry (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Peptides Or Proteins (AREA)
  • Medicinal Preparation (AREA)
  • Cosmetics (AREA)

Abstract

La divulgación se refiere a un método para tratar un trastorno, trastorno o condición asociados al gen agonizable de la vía MC4R, tales como obesidad o hiperfagia, en un sujeto que usa un agonista del receptor de melanocortina 4 (MC4R).
CL2023000823A 2020-09-24 2023-03-22 Métodos para tratar trastornos asociados a la vía del receptor de melanocortina 4 CL2023000823A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US202063082867P 2020-09-24 2020-09-24

Publications (1)

Publication Number Publication Date
CL2023000823A1 true CL2023000823A1 (es) 2023-09-15

Family

ID=80845850

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2023000823A CL2023000823A1 (es) 2020-09-24 2023-03-22 Métodos para tratar trastornos asociados a la vía del receptor de melanocortina 4

Country Status (13)

Country Link
US (1) US20240058414A1 (es)
EP (1) EP4216979A1 (es)
JP (1) JP2023542985A (es)
KR (1) KR20230095956A (es)
CN (1) CN116507353A (es)
AR (1) AR123603A1 (es)
AU (1) AU2021350017A1 (es)
CA (1) CA3192873A1 (es)
CL (1) CL2023000823A1 (es)
CO (1) CO2022009561A2 (es)
MX (1) MX2023003360A (es)
TW (1) TW202228760A (es)
WO (1) WO2022067086A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2024015880A2 (en) * 2022-07-12 2024-01-18 Rhythm Pharmaceuticals, Inc. Methods for treating obesity with an mc4r agonist

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8039435B2 (en) * 2005-07-08 2011-10-18 Ipsen Pharma S.A.S. Melanocortin receptor ligands
EP4029513A1 (en) * 2015-09-30 2022-07-20 Rhythm Pharmaceuticals, Inc. Melanocortin-4 receptor agonists for the treatment of disorders characterised by pomc gene hypermethylation

Also Published As

Publication number Publication date
WO2022067086A1 (en) 2022-03-31
KR20230095956A (ko) 2023-06-29
CN116507353A (zh) 2023-07-28
CA3192873A1 (en) 2022-03-31
AR123603A1 (es) 2022-12-21
CO2022009561A2 (es) 2022-07-19
TW202228760A (zh) 2022-08-01
AU2021350017A1 (en) 2023-05-04
US20240058414A1 (en) 2024-02-22
JP2023542985A (ja) 2023-10-12
MX2023003360A (es) 2023-06-23
EP4216979A1 (en) 2023-08-02

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