CO2022009561A2 - Métodos de tratamiento de los trastornos asociados a la vía del receptor de melanocortina 4 - Google Patents
Métodos de tratamiento de los trastornos asociados a la vía del receptor de melanocortina 4Info
- Publication number
- CO2022009561A2 CO2022009561A2 CONC2022/0009561A CO2022009561A CO2022009561A2 CO 2022009561 A2 CO2022009561 A2 CO 2022009561A2 CO 2022009561 A CO2022009561 A CO 2022009561A CO 2022009561 A2 CO2022009561 A2 CO 2022009561A2
- Authority
- CO
- Colombia
- Prior art keywords
- melanocortin
- treatment methods
- disorders associated
- receptor pathway
- receptor
- Prior art date
Links
- 102000001796 Melanocortin 4 receptors Human genes 0.000 title abstract 4
- 108010021436 Type 4 Melanocortin Receptor Proteins 0.000 title abstract 4
- 230000037361 pathway Effects 0.000 title abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 208000035475 disorder Diseases 0.000 abstract 2
- 206010020710 Hyperphagia Diseases 0.000 abstract 1
- 208000008589 Obesity Diseases 0.000 abstract 1
- 239000000556 agonist Substances 0.000 abstract 1
- 235000020824 obesity Nutrition 0.000 abstract 1
- 108090000623 proteins and genes Proteins 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Gastroenterology & Hepatology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Diabetes (AREA)
- Child & Adolescent Psychology (AREA)
- Obesity (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Hematology (AREA)
- Dermatology (AREA)
- Organic Chemistry (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Plant Substances (AREA)
- Peptides Or Proteins (AREA)
- Cosmetics (AREA)
- Medicinal Preparation (AREA)
Abstract
La divulgación está relacionada con un método de tratamiento de un trastorno, un desorden o una condición asociados con un gen agonizable de la vía MC4R, como la obesidad o la hiperfagia, en un sujeto usando un agonista del receptor de melanocortina-4 (MC4R).
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US202063082867P | 2020-09-24 | 2020-09-24 | |
PCT/US2021/052032 WO2022067086A1 (en) | 2020-09-24 | 2021-09-24 | Methods of treating melanocortin-4 receptor pathway-associated disorders |
Publications (1)
Publication Number | Publication Date |
---|---|
CO2022009561A2 true CO2022009561A2 (es) | 2022-07-19 |
Family
ID=80845850
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CONC2022/0009561A CO2022009561A2 (es) | 2020-09-24 | 2022-07-07 | Métodos de tratamiento de los trastornos asociados a la vía del receptor de melanocortina 4 |
Country Status (13)
Country | Link |
---|---|
US (1) | US20240058414A1 (es) |
EP (1) | EP4216979A1 (es) |
JP (1) | JP2023542985A (es) |
KR (1) | KR20230095956A (es) |
CN (1) | CN116507353A (es) |
AR (1) | AR123603A1 (es) |
AU (1) | AU2021350017A1 (es) |
CA (1) | CA3192873A1 (es) |
CL (1) | CL2023000823A1 (es) |
CO (1) | CO2022009561A2 (es) |
MX (1) | MX2023003360A (es) |
TW (1) | TW202228760A (es) |
WO (1) | WO2022067086A1 (es) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2024015880A2 (en) * | 2022-07-12 | 2024-01-18 | Rhythm Pharmaceuticals, Inc. | Methods for treating obesity with an mc4r agonist |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN101257916B (zh) * | 2005-07-08 | 2013-04-03 | 益普生制药股份有限公司 | 黑皮质素受体配体 |
CN108601816A (zh) * | 2015-09-30 | 2018-09-28 | 节奏制药公司 | 治疗黑皮质素-4受体路径相关联病症的方法 |
-
2021
- 2021-09-24 US US18/028,117 patent/US20240058414A1/en active Pending
- 2021-09-24 EP EP21873549.6A patent/EP4216979A1/en active Pending
- 2021-09-24 KR KR1020237013822A patent/KR20230095956A/ko unknown
- 2021-09-24 CN CN202180071771.8A patent/CN116507353A/zh active Pending
- 2021-09-24 AU AU2021350017A patent/AU2021350017A1/en active Pending
- 2021-09-24 TW TW110135665A patent/TW202228760A/zh unknown
- 2021-09-24 JP JP2023518779A patent/JP2023542985A/ja active Pending
- 2021-09-24 AR ARP210102664A patent/AR123603A1/es unknown
- 2021-09-24 CA CA3192873A patent/CA3192873A1/en active Pending
- 2021-09-24 WO PCT/US2021/052032 patent/WO2022067086A1/en active Application Filing
- 2021-09-24 MX MX2023003360A patent/MX2023003360A/es unknown
-
2022
- 2022-07-07 CO CONC2022/0009561A patent/CO2022009561A2/es unknown
-
2023
- 2023-03-22 CL CL2023000823A patent/CL2023000823A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
AR123603A1 (es) | 2022-12-21 |
CL2023000823A1 (es) | 2023-09-15 |
WO2022067086A1 (en) | 2022-03-31 |
CA3192873A1 (en) | 2022-03-31 |
KR20230095956A (ko) | 2023-06-29 |
TW202228760A (zh) | 2022-08-01 |
EP4216979A1 (en) | 2023-08-02 |
AU2021350017A1 (en) | 2023-05-04 |
CN116507353A (zh) | 2023-07-28 |
JP2023542985A (ja) | 2023-10-12 |
US20240058414A1 (en) | 2024-02-22 |
MX2023003360A (es) | 2023-06-23 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
MX2022010425A (es) | Metodos de tratamiento de enfermedades asociadas a los receptores de estrogenos. | |
EA201992474A2 (ru) | Агонисты 5ht для лечения нарушений | |
CO2022009561A2 (es) | Métodos de tratamiento de los trastornos asociados a la vía del receptor de melanocortina 4 | |
UY37269A (es) | Agonista del receptor de glucocorticoides e inmunoconjugados del mismo | |
CO2021005231A2 (es) | Composiciones y métodos para la edición génica de lactato deshidrogenasa (ldha) | |
EA201000673A1 (ru) | СПОСОБЫ И КОМПОЗИЦИИ ДЛЯ ИЗМЕРЕНИЯ АКТИВАЦИИ Wnt И ДЛЯ ЛЕЧЕНИЯ Wnt-ОПОСРЕДОВАННЫХ РАКОВЫХ ЗАБОЛЕВАНИЙ | |
PH12017502120A1 (en) | A method and an apparatus for forming a lignin fraction, a lignin composition and its use | |
EA201792437A1 (ru) | Способы и композиции для лечения нарушений, ассоциированных со старением | |
CL2018003565A1 (es) | Anticuerpos antifactor de la coagulación xi. | |
CL2022001256A1 (es) | Métodos y composiciones para tratar un trastorno asociado con el angiotensinogeno agt | |
CO2020005417A2 (es) | Inhibidores de la quinasa p38 que reducen la expresión de dux4 y de los genes corriente abajo para el tratamiento de fshd | |
CR20160132A (es) | Composiciones y método para tratar condiciones asociadas con el complemento | |
CL2018002810A1 (es) | Anticuerpos anti-factor bb del complemento y usos de estos referencia cruzada. | |
BR112018006674A2 (pt) | método de tratamento de distúrbios associados com a via do receptor de melanocortina-4 | |
CO2021008998A2 (es) | Amidas de pirrolidina iii sustituidas | |
MX2022008320A (es) | Métodos para tratar trastornos de pénfigo. | |
CL2021001903A1 (es) | Tratamiento de la hepatotoxicidad | |
WO2018150276A3 (en) | The combination of cotinine plus antioxidant for treatment resistant depression and other neuropathological conditions | |
EA201891253A1 (ru) | Способ получения высококачественного исходного материала для процесса парового крекинга | |
CL2020002165A1 (es) | Uso de tradipitant para tratar la cinetosis. | |
WO2023086428A3 (en) | Novel modulators of the aryl hydrocarbon receptor and methods of use thereof | |
CU20200038A7 (es) | Compuestos derivados de pirazolo-pirrolo-pirimidina-diona como inhibidores de p2x3 | |
MX2023005342A (es) | Métodos para tratar padecimientos relacionados con el receptor s1p1. | |
CL2023003126A1 (es) | Métodos de identificación de pacientes con posibilidad de beneficiarse de tratamiento con inhibidor de telomerasa | |
MX2022012302A (es) | Formas polimórficas de metopimazina novedosas. |