CL2021000618A1 - Compuesto que contiene oxadiazol y composición farmacéutica que contiene el mismo - Google Patents
Compuesto que contiene oxadiazol y composición farmacéutica que contiene el mismoInfo
- Publication number
- CL2021000618A1 CL2021000618A1 CL2021000618A CL2021000618A CL2021000618A1 CL 2021000618 A1 CL2021000618 A1 CL 2021000618A1 CL 2021000618 A CL2021000618 A CL 2021000618A CL 2021000618 A CL2021000618 A CL 2021000618A CL 2021000618 A1 CL2021000618 A1 CL 2021000618A1
- Authority
- CL
- Chile
- Prior art keywords
- same
- pharmaceutical composition
- oxadiazole
- composition containing
- compound
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 2
- WCPAKWJPBJAGKN-UHFFFAOYSA-N oxadiazole Chemical compound C1=CON=N1 WCPAKWJPBJAGKN-UHFFFAOYSA-N 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 150000003839 salts Chemical class 0.000 abstract 2
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 206010015037 epilepsy Diseases 0.000 abstract 1
- 210000000653 nervous system Anatomy 0.000 abstract 1
- -1 oxadiazole compound Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
- C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
- C07D271/10—1,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4245—Oxadiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
- C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
- C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
Se describe en la presente invención un compuesto de oxadiazol y sales farmacéuticamente útiles del mismo. El compuesto y sales farmacéuticamente útiles del mismo son especialmente adecuadas para el tratamiento de enfermedades del sistema nervioso tal como epilepsia.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
KR20180113956 | 2018-09-21 |
Publications (1)
Publication Number | Publication Date |
---|---|
CL2021000618A1 true CL2021000618A1 (es) | 2021-08-06 |
Family
ID=69887571
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CL2021000618A CL2021000618A1 (es) | 2018-09-21 | 2021-03-12 | Compuesto que contiene oxadiazol y composición farmacéutica que contiene el mismo |
Country Status (16)
Country | Link |
---|---|
US (4) | US11053208B2 (es) |
EP (1) | EP3854788A4 (es) |
JP (1) | JP7430175B2 (es) |
KR (1) | KR102827846B1 (es) |
CN (1) | CN113272285B (es) |
AR (1) | AR118413A1 (es) |
AU (1) | AU2019341357B2 (es) |
BR (1) | BR112021005269A2 (es) |
CA (1) | CA3112700A1 (es) |
CL (1) | CL2021000618A1 (es) |
IL (1) | IL281553B2 (es) |
MX (1) | MX2021003204A (es) |
MY (1) | MY206736A (es) |
TW (1) | TWI826531B (es) |
WO (1) | WO2020060299A1 (es) |
ZA (1) | ZA202101520B (es) |
Family Cites Families (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US21121A (en) | 1858-08-10 | Appabattjs for purifying gas | ||
IE49823B1 (en) | 1979-06-01 | 1985-12-25 | Wellcome Found | 1,2,4-triazine derivatives,process for preparing such compounds and pharmaceutical compositions containing them |
GB8412357D0 (en) | 1984-05-15 | 1984-06-20 | Ucb Sa | Pharmaceutical composition |
KR0162036B1 (ko) | 1996-05-31 | 1998-12-01 | 추호석 | 스택커 크래인의 모터 제어장치 및 방법 |
JP2003524595A (ja) | 1998-07-08 | 2003-08-19 | モナシュ ユニバーシティ | 薬 剤 |
UA78211C2 (en) | 2001-07-09 | 2007-03-15 | Ortho Mcneil Pharm Inc | Salts of fructopyranose derivatives as anticonvulsant |
AU2005271669A1 (en) * | 2004-08-03 | 2006-02-16 | Merck & Co., Inc. | 1,3-disubstituted heteroaryl NMDA/NR2B antagonists |
US7598279B2 (en) * | 2005-04-22 | 2009-10-06 | Sk Holdings Co., Ltd. | Neurotherapeutic azole compounds |
EP2051964A4 (en) * | 2006-07-28 | 2012-03-07 | Univ Connecticut | INHIBITORS OF FATTY ACID AMIDHYDROLASE |
CN102015637B (zh) | 2008-02-06 | 2014-05-21 | 第一三共株式会社 | 苯基吡咯衍生物 |
CA2785679C (en) | 2009-12-28 | 2017-12-12 | General Incorporated Association Pharma Valley Project Supporting Organization | 1,3,4-oxadiazole-2-carboxamide compound |
EP2544679B1 (en) * | 2010-03-12 | 2019-05-15 | Omeros Corporation | Pde10 inhibitors and related compositions and methods |
WO2017060488A1 (en) * | 2015-10-09 | 2017-04-13 | Almirall, S.A. | New trpa1 antagonists |
-
2019
- 2019-09-19 TW TW108133837A patent/TWI826531B/zh active
- 2019-09-20 WO PCT/KR2019/012257 patent/WO2020060299A1/ko active Application Filing
- 2019-09-20 US US16/613,659 patent/US11053208B2/en active Active
- 2019-09-20 IL IL281553A patent/IL281553B2/en unknown
- 2019-09-20 CA CA3112700A patent/CA3112700A1/en active Pending
- 2019-09-20 KR KR1020217007242A patent/KR102827846B1/ko active Active
- 2019-09-20 MX MX2021003204A patent/MX2021003204A/es unknown
- 2019-09-20 CN CN201980076515.0A patent/CN113272285B/zh active Active
- 2019-09-20 MY MYPI2021001215A patent/MY206736A/en unknown
- 2019-09-20 AU AU2019341357A patent/AU2019341357B2/en active Active
- 2019-09-20 BR BR112021005269-0A patent/BR112021005269A2/pt unknown
- 2019-09-20 AR ARP190102667A patent/AR118413A1/es unknown
- 2019-09-20 JP JP2021516367A patent/JP7430175B2/ja active Active
- 2019-09-20 EP EP19863530.2A patent/EP3854788A4/en active Pending
-
2021
- 2021-03-05 ZA ZA2021/01520A patent/ZA202101520B/en unknown
- 2021-03-12 CL CL2021000618A patent/CL2021000618A1/es unknown
- 2021-05-24 US US17/327,928 patent/US11603358B2/en active Active
-
2023
- 2023-01-18 US US18/155,924 patent/US12145914B2/en active Active
-
2024
- 2024-10-10 US US18/911,634 patent/US20250034101A1/en active Pending
Also Published As
Publication number | Publication date |
---|---|
KR20210047889A (ko) | 2021-04-30 |
JP2022503775A (ja) | 2022-01-12 |
US20220024886A1 (en) | 2022-01-27 |
US11053208B2 (en) | 2021-07-06 |
US12145914B2 (en) | 2024-11-19 |
AU2019341357B2 (en) | 2023-03-02 |
EP3854788A1 (en) | 2021-07-28 |
MX2021003204A (es) | 2021-05-27 |
TW202023547A (zh) | 2020-07-01 |
AR118413A1 (es) | 2021-10-06 |
TWI826531B (zh) | 2023-12-21 |
JP7430175B2 (ja) | 2024-02-09 |
BR112021005269A2 (pt) | 2021-06-15 |
CA3112700A1 (en) | 2020-03-26 |
US20230150955A1 (en) | 2023-05-18 |
MY206736A (en) | 2025-01-03 |
US20210115001A1 (en) | 2021-04-22 |
US20250034101A1 (en) | 2025-01-30 |
KR102827846B1 (ko) | 2025-07-01 |
WO2020060299A1 (ko) | 2020-03-26 |
CN113272285A (zh) | 2021-08-17 |
CN113272285B (zh) | 2024-06-07 |
ZA202101520B (en) | 2022-08-31 |
US11603358B2 (en) | 2023-03-14 |
AU2019341357A1 (en) | 2021-04-08 |
IL281553A (en) | 2021-05-31 |
IL281553B1 (en) | 2025-02-01 |
IL281553B2 (en) | 2025-06-01 |
EP3854788A4 (en) | 2022-06-15 |
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