CL2015001621A1 - Proceso para la formacion de tabletas de ibuprofeno de sodio dihidratado, que comprende la formacion de tabletas en una prensa a partir de gránulos. - Google Patents

Proceso para la formacion de tabletas de ibuprofeno de sodio dihidratado, que comprende la formacion de tabletas en una prensa a partir de gránulos.

Info

Publication number
CL2015001621A1
CL2015001621A1 CL2015001621A CL2015001621A CL2015001621A1 CL 2015001621 A1 CL2015001621 A1 CL 2015001621A1 CL 2015001621 A CL2015001621 A CL 2015001621A CL 2015001621 A CL2015001621 A CL 2015001621A CL 2015001621 A1 CL2015001621 A1 CL 2015001621A1
Authority
CL
Chile
Prior art keywords
tablets
formation
granules
press
sodium ibuprofen
Prior art date
Application number
CL2015001621A
Other languages
English (en)
Spanish (es)
Inventor
Latria N Boudoin
Gregory H Lambeth
Eric W Limatta
Patrick C Hu
Original Assignee
Si Group Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49841833&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2015001621(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US13/714,768 external-priority patent/US9629809B2/en
Application filed by Si Group Inc filed Critical Si Group Inc
Publication of CL2015001621A1 publication Critical patent/CL2015001621A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/192Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2095Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Inorganic Chemistry (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
CL2015001621A 2012-12-14 2015-06-11 Proceso para la formacion de tabletas de ibuprofeno de sodio dihidratado, que comprende la formacion de tabletas en una prensa a partir de gránulos. CL2015001621A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US13/714,768 US9629809B2 (en) 2008-07-21 2012-12-14 High content sodium ibuprofen granules, their preparation and their use in preparing non-effervescent solid dosage forms

Publications (1)

Publication Number Publication Date
CL2015001621A1 true CL2015001621A1 (es) 2015-08-07

Family

ID=49841833

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2015001621A CL2015001621A1 (es) 2012-12-14 2015-06-11 Proceso para la formacion de tabletas de ibuprofeno de sodio dihidratado, que comprende la formacion de tabletas en una prensa a partir de gránulos.

Country Status (9)

Country Link
EP (1) EP2931261A1 (zh)
JP (1) JP6285952B2 (zh)
CN (1) CN104884048B (zh)
BR (1) BR112015013945A8 (zh)
CA (1) CA2894272A1 (zh)
CL (1) CL2015001621A1 (zh)
HK (1) HK1210591A1 (zh)
MX (1) MX2015007571A (zh)
WO (1) WO2014093073A1 (zh)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT3675828T (pt) * 2017-08-31 2023-10-09 Novartis Ag Método de preparação de grânulos

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1293764B1 (it) * 1997-07-23 1999-03-10 Chiesi Farma Spa Composizioni farmaceutiche sotto forma di compresse effervescenti contenenti un principio attivo instabile in presenza di acqua
JP4753567B2 (ja) * 2004-11-19 2011-08-24 旭化成ケミカルズ株式会社 付着性の高い薬物を含有する錠剤の製造方法
DE102005009241A1 (de) * 2005-03-01 2006-09-07 Bayer Healthcare Ag Arzneiformen mit kontrollierter Bioverfügbarkeit
WO2010011522A1 (en) * 2008-07-21 2010-01-28 Albemarle Corporation High content sodium ibuprofen granules, their preparation and their use in preparing non-effervescent solid dosage forms
MX2020011961A (es) * 2010-03-24 2022-04-19 Jazz Pharmaceuticals Inc Formas de dosis de liberacion controlada para substancias de farmaco de alta dosis, solubles en agua e higroscopicas.

Also Published As

Publication number Publication date
JP2016508124A (ja) 2016-03-17
WO2014093073A1 (en) 2014-06-19
EP2931261A1 (en) 2015-10-21
CN104884048A (zh) 2015-09-02
HK1210591A1 (zh) 2016-04-29
JP6285952B2 (ja) 2018-02-28
CA2894272A1 (en) 2014-06-19
CN104884048B (zh) 2018-11-23
BR112015013945A8 (pt) 2019-10-08
BR112015013945A2 (pt) 2017-07-11
MX2015007571A (es) 2016-04-15

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