CH524621A - Verfahren zur Herstellung von Benzodiazepin-Derivaten - Google Patents

Verfahren zur Herstellung von Benzodiazepin-Derivaten

Info

Publication number
CH524621A
CH524621A CH892271A CH892271A CH524621A CH 524621 A CH524621 A CH 524621A CH 892271 A CH892271 A CH 892271A CH 892271 A CH892271 A CH 892271A CH 524621 A CH524621 A CH 524621A
Authority
CH
Switzerland
Prior art keywords
preparation
benzodiazepine derivatives
benzodiazepine
derivatives
Prior art date
Application number
CH892271A
Other languages
English (en)
Inventor
Ian Fryer Rodney
Henryk Sternbach Leo
Valentine Earley James
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of CH524621A publication Critical patent/CH524621A/de

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CH892271A 1967-07-03 1968-06-26 Verfahren zur Herstellung von Benzodiazepin-Derivaten CH524621A (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US65065167A 1967-07-03 1967-07-03
US65065267A 1967-07-03 1967-07-03

Publications (1)

Publication Number Publication Date
CH524621A true CH524621A (de) 1972-06-30

Family

ID=27095915

Family Applications (3)

Application Number Title Priority Date Filing Date
CH892271A CH524621A (de) 1967-07-03 1968-06-26 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH952368A CH512475A (de) 1967-07-03 1968-06-26 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH892371A CH526558A (de) 1967-07-03 1968-06-26 Verfahren zur Herstellung von Benzodiazepin-Derivaten

Family Applications After (2)

Application Number Title Priority Date Filing Date
CH952368A CH512475A (de) 1967-07-03 1968-06-26 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH892371A CH526558A (de) 1967-07-03 1968-06-26 Verfahren zur Herstellung von Benzodiazepin-Derivaten

Country Status (11)

Country Link
US (1) US3523939A (de)
BE (1) BE717478A (de)
CA (1) CA952106A (de)
CH (3) CH524621A (de)
DE (1) DE1770778A1 (de)
FR (2) FR1586872A (de)
GB (2) GB1205996A (de)
IE (1) IE32217B1 (de)
IL (2) IL30282A (de)
NL (1) NL6809403A (de)
SE (1) SE358167B (de)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS4837280B1 (de) * 1969-03-08 1973-11-09
US3723414A (en) * 1970-02-13 1973-03-27 Schering Corp 1-polyfluoroalkyl benzodiazepines
AT333284B (de) * 1971-12-09 1976-11-10 Degussa Verfahren zur herstellung von neuen 6-aza-3h-1,4-benzodiazepinen, deren optischen isomeren und deren salzen
US4089953A (en) * 1973-06-20 1978-05-16 Ddsa Pharmaceuticals 1,5-Benzodiazocines
US4056525A (en) * 1975-06-02 1977-11-01 American Home Products Corporation 2,3-dialkoxy-3h-1,4-benzodiazepines
KR20100017766A (ko) * 2007-05-10 2010-02-16 에이엠알 테크놀로지, 인크. 아릴- 및 헤테로아릴-치환된 테트라히드로벤조-1,4-디아제핀 및 노르에피네프린, 도파민 및 세로토닌의 재흡수를 차단하기 위한 이의 용도
AR084070A1 (es) 2010-12-02 2013-04-17 Constellation Pharmaceuticals Inc Inhibidores del bromodominio y usos de los mismos
WO2012075456A1 (en) 2010-12-02 2012-06-07 Constellation Pharmaceuticals Bromodomain inhibitors and uses thereof
EP2705039B1 (de) 2011-05-04 2017-07-26 Constellation Pharmaceuticals, Inc. Bromodomainhemmer und ihre verwendung
EP2721031B1 (de) 2011-06-17 2016-01-20 Constellation Pharmaceuticals, Inc. Bromodomainhemmer und ihre verwendungen
TWI602820B (zh) 2012-06-06 2017-10-21 星宿藥物公司 溴域抑制劑及其用途
WO2013184878A1 (en) 2012-06-06 2013-12-12 Constellation Pharmaceuticals, Inc. Benzo [b] isoxazoloazepine bromodomain inhibitors and uses thereof
US9969747B2 (en) 2014-06-20 2018-05-15 Constellation Pharmaceuticals, Inc. Crystalline forms of 2-((4S)-6-(4-chlorophenyl)-1-methyl-4H-benzo[C]isoxazolo[4,5-e]azepin-4-yl)acetamide

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2893992A (en) * 1959-07-07 I ii i i
US3109843A (en) * 1963-11-05 Process for preparing
US3371085A (en) * 1959-12-10 1968-02-27 Hoffmann La Roche 5-aryl-3h-1,4-benzodiazepin-2(1h)-ones
GB1052144A (de) * 1964-02-11

Also Published As

Publication number Publication date
CH526558A (de) 1972-08-15
US3523939A (en) 1970-08-11
BE717478A (de) 1969-01-02
GB1205995A (en) 1970-09-23
IE32217L (en) 1969-01-03
IL30282A (en) 1972-11-28
FR1586872A (de) 1970-03-06
CA952106A (en) 1974-07-30
IE32217B1 (en) 1973-05-16
FR8488M (de) 1973-07-27
NL6809403A (de) 1969-01-07
IL38208A (en) 1973-04-30
GB1205996A (en) 1970-09-23
IL30282A0 (en) 1968-09-26
CH512475A (de) 1971-09-15
DE1770778A1 (de) 1972-02-17
SE358167B (de) 1973-07-23

Similar Documents

Publication Publication Date Title
CH510669A (de) Verfahren zur Herstellung von Isochinuclidin-Derivaten
CH541580A (de) Verfahren zur Herstellung von Bis-thioureidobenzol-derivaten
CH529145A (de) Verfahren zur Herstellung von 1-Aminoalkylbenzodiazepinderivaten
CH526558A (de) Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH543514A (de) Verfahren zur Herstellung von Morphinanderivaten
CH518301A (de) Verfahren zur Herstellung von Dibenzothiazepin-Derivaten
CH498846A (de) Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH473133A (de) Verfahren zur Herstellung von Benzodiazepin-Derivaten
AT273953B (de) Verfahren zur Herstellung von v-Triazolyl-cumarinderivaten
CH524620A (de) Verfahren zur Herstellung von Benzodiazepinderivaten
AT280295B (de) Verfahren zur Herstellung von Benzodiazepinderivaten
CH537394A (de) Verfahren zur Herstellung von Benzodiazepinen
CH511864A (de) Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH478812A (de) Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH517752A (de) Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH493539A (de) Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH490401A (de) Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH461517A (de) Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH460791A (de) Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH507233A (de) Verfahren zur Herstellung von Kalamycinderivaten
CH492723A (de) Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH526556A (de) Verfahren zur Herstellung von Benzodiazepinderivaten
CH497441A (de) Verfahren zur Herstellung von Dibenzazepinderivaten
CH491938A (de) Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH484164A (de) Verfahren zur Herstellung von Benzodiazepin-Derivaten

Legal Events

Date Code Title Description
PL Patent ceased