CH462176A - Verfahren zur Herstellung von 1-Aralkyl-4-(thiazolyl-2)-piperazinen - Google Patents

Verfahren zur Herstellung von 1-Aralkyl-4-(thiazolyl-2)-piperazinen

Info

Publication number
CH462176A
CH462176A CH233068A CH233068A CH462176A CH 462176 A CH462176 A CH 462176A CH 233068 A CH233068 A CH 233068A CH 233068 A CH233068 A CH 233068A CH 462176 A CH462176 A CH 462176A
Authority
CH
Switzerland
Prior art keywords
piperazines
thiazolyl
aralkyl
preparation
Prior art date
Application number
CH233068A
Other languages
English (en)
Inventor
Schulte Karl Dr Dipl-Chem
Koppe Volker Dr Dipl-Chem
Siegmund Dr Sommer
Ernst Dr Schorscher
Original Assignee
Merck Ag E
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Ag E filed Critical Merck Ag E
Publication of CH462176A publication Critical patent/CH462176A/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • DTEXTILES; PAPER
    • D05SEWING; EMBROIDERING; TUFTING
    • D05BSEWING
    • D05B7/00Linking machines, e.g. for joining knitted fabrics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Textile Engineering (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CH233068A 1965-02-20 1965-12-30 Verfahren zur Herstellung von 1-Aralkyl-4-(thiazolyl-2)-piperazinen CH462176A (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DEM0064244 1965-02-20

Publications (1)

Publication Number Publication Date
CH462176A true CH462176A (de) 1968-09-15

Family

ID=7311049

Family Applications (2)

Application Number Title Priority Date Filing Date
CH1811465A CH460787A (de) 1965-02-20 1965-12-30 Verfahren zur Herstellung von 1-Aralkyl-4-(thiazolyl-2)-piperazinen
CH233068A CH462176A (de) 1965-02-20 1965-12-30 Verfahren zur Herstellung von 1-Aralkyl-4-(thiazolyl-2)-piperazinen

Family Applications Before (1)

Application Number Title Priority Date Filing Date
CH1811465A CH460787A (de) 1965-02-20 1965-12-30 Verfahren zur Herstellung von 1-Aralkyl-4-(thiazolyl-2)-piperazinen

Country Status (8)

Country Link
US (1) US3489757A (de)
BE (1) BE676686A (de)
CH (2) CH460787A (de)
DE (1) DE1595923A1 (de)
ES (1) ES323305A1 (de)
FR (1) FR5175M (de)
GB (1) GB1061247A (de)
NL (1) NL6601699A (de)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH583232A5 (de) * 1973-02-02 1976-12-31 Wander Ag Dr A
US3907819A (en) * 1973-05-14 1975-09-23 Du Pont Perhalogenated thiazoles
GB1560084A (en) * 1976-12-31 1980-01-30 Science Union & Cie Disubstituted piperazines processes for their preparation and pharmaceutical mompositions containing them
OA06083A (fr) * 1977-11-09 1981-06-30 Science Union & Cie Ste Franca Nouvelles pipérazines disubstituées, leurs procédés de préparation et les compositions pharmaceutiques les renfermant.
EP0005091B1 (de) * 1978-04-13 1981-11-25 SCIENCE UNION ET Cie SOCIETE FRANCAISE DE RECHERCHE MEDICALE Monosubstituierte Piperazine, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Präparate
US4411900A (en) * 1980-01-03 1983-10-25 Fujisawa Pharmaceutical Co., Ltd. Benzhydrylpiperozinyl thiazole derivatives and pharmaceutical composition comprising the same
US4647557A (en) * 1982-12-28 1987-03-03 Gerard Moinet Novel heterocyclic derivatives bearing an amino radical, processes for their production and the pharmaceutical compositions containing them
NL8601494A (nl) * 1985-06-22 1987-01-16 Sandoz Ag Thiazolen, hun bereiding en farmaceutische preparaten die ze bevatten.
US4914112A (en) * 1986-06-03 1990-04-03 Sumitomo Pharmaceuticals Company, Limited Aminoazole derivatives and their production and use
DE3812755A1 (de) * 1988-04-16 1989-10-26 Merck Patent Gmbh Salicylsaeurederivate
FR2637596B1 (fr) * 1988-10-11 1992-09-04 Irceba Methyl-4 ((aryl-4 piperazinyl-1)-2 ethyl)-5 thiazole et ses derives, leur procede de preparation et les medicaments en contenant
ES2062940B1 (es) * 1993-03-11 1995-06-16 Vita Invest Sa Agente gastrocinetico, proceso para su preparacion y composiciones farmaceuticas que lo contengan.
TW200826936A (en) * 2006-12-01 2008-07-01 Merck Frosst Canada Ltd Azacycloalkane derivatives as inhibitors of stearoyl-coenzyme a delta-9 desaturase
MA40532A (fr) * 2014-08-28 2021-04-28 Asceneuron Sa Inhibiteurs de glycosidases
AU2017222964B2 (en) 2016-02-25 2020-01-02 Asceneuron S. A. Glycosidase inhibitors
SG11201807012QA (en) 2016-02-25 2018-09-27 Asceneuron S A Acid addition salts of piperazine derivatives
EP3419971B1 (de) * 2016-02-25 2022-04-20 Asceneuron SA Glycosidase-inhibitoren
US11261183B2 (en) 2016-02-25 2022-03-01 Asceneuron Sa Sulfoximine glycosidase inhibitors
EP3555087A1 (de) * 2016-12-16 2019-10-23 Janssen Pharmaceutica NV Monocyclische oga-inhibitor-verbindungen
MX2019010085A (es) 2017-02-24 2019-11-21 Asceneuron S A Inhibidores de la glicosidasa de sulfoximina.
US11458140B2 (en) 2017-08-24 2022-10-04 Asceneuron Sa Annulated glycosidase inhibitors
WO2019037860A1 (en) 2017-08-24 2019-02-28 Asceneuron S.A. LINEAR INHIBITORS OF GLYCOSIDASE
US12016852B2 (en) 2018-08-22 2024-06-25 Asceneuron Sa Pyrrolidine glycosidase inhibitors
WO2020039028A1 (en) 2018-08-22 2020-02-27 Asceneuron S. A. Tetrahydro-benzoazepine glycosidase inhibitors
WO2020039029A1 (en) 2018-08-22 2020-02-27 Asceneuron S. A. Spiro compounds as glycosidase inhibitors
WO2020169804A1 (en) 2019-02-22 2020-08-27 Asceneuron Sa Fused glycosidase inhibitors

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE485737A (de) * 1947-11-12
DE1595920B2 (de) * 1964-11-04 1978-08-10 Merck Patent Gmbh, 6100 Darmstadt 4-(co-Piperazinoalkyl)-pyrazole, ihre Salze und Verfahren zu ihrer Herstellung

Also Published As

Publication number Publication date
GB1061247A (en) 1967-03-08
CH460787A (de) 1968-08-15
BE676686A (de) 1966-08-18
FR5175M (de) 1967-06-19
DE1595923A1 (de) 1969-11-27
ES323305A1 (es) 1967-03-16
NL6601699A (de) 1966-08-22
US3489757A (en) 1970-01-13

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