CH458371A - Verfahren zur Herstellung von Benzodiazepinderivaten - Google Patents

Verfahren zur Herstellung von Benzodiazepinderivaten

Info

Publication number
CH458371A
CH458371A CH846664A CH846664A CH458371A CH 458371 A CH458371 A CH 458371A CH 846664 A CH846664 A CH 846664A CH 846664 A CH846664 A CH 846664A CH 458371 A CH458371 A CH 458371A
Authority
CH
Switzerland
Prior art keywords
preparation
benzodiazepine derivatives
benzodiazepine
derivatives
Prior art date
Application number
CH846664A
Other languages
English (en)
Inventor
Ian Fryer Rodney
Henryk Sternbach Leo
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of CH458371A publication Critical patent/CH458371A/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CH846664A 1963-07-10 1964-06-26 Verfahren zur Herstellung von Benzodiazepinderivaten CH458371A (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US294142A US3247187A (en) 1963-07-10 1963-07-10 Oxidation of 1, 4-benzodiazepines to 1, 4-benzodiazepin-2-ones

Publications (1)

Publication Number Publication Date
CH458371A true CH458371A (de) 1968-06-30

Family

ID=23132071

Family Applications (1)

Application Number Title Priority Date Filing Date
CH846664A CH458371A (de) 1963-07-10 1964-06-26 Verfahren zur Herstellung von Benzodiazepinderivaten

Country Status (11)

Country Link
US (1) US3247187A (de)
BE (1) BE650261A (de)
BR (1) BR6460685D0 (de)
CH (1) CH458371A (de)
DE (1) DE1445901A1 (de)
DK (1) DK120600B (de)
ES (1) ES301865A1 (de)
GB (1) GB1036577A (de)
NL (1) NL6407796A (de)
NO (1) NO117639B (de)
OA (1) OA00949A (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3361742A (en) * 1964-12-07 1968-01-02 Hoffmann La Roche 5-oxo-1h-pyrrolo-[2, 1-c][1, 4]-benzodiazepin-2-crylamides
US3405123A (en) * 1965-02-08 1968-10-08 Hoffmann La Roche Process for preparing 1, 4-benzodiazepin-2-ones

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3121076A (en) * 1964-02-11 Benzodiazepinones and processes
US3176009A (en) * 1965-03-30 Hydrolysis of l-acylated-j-acyloxy benzodiazepines

Also Published As

Publication number Publication date
DK120600B (da) 1971-06-21
NL6407796A (de) 1965-01-11
BR6460685D0 (pt) 1973-07-19
GB1036577A (en) 1966-07-20
DE1445901A1 (de) 1969-02-06
BE650261A (de) 1965-01-08
US3247187A (en) 1966-04-19
NO117639B (de) 1969-09-08
ES301865A1 (es) 1965-02-01
OA00949A (fr) 1968-03-22

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