CA962678A - 4-acetoxy-2-methyl-3-(5-methylisoxazol-3-yl-carbamoyl)-2h-1,2-benzothiazine 1,1-dioxide - Google Patents

4-acetoxy-2-methyl-3-(5-methylisoxazol-3-yl-carbamoyl)-2h-1,2-benzothiazine 1,1-dioxide

Info

Publication number
CA962678A
CA962678A CA145,331A CA145331A CA962678A CA 962678 A CA962678 A CA 962678A CA 145331 A CA145331 A CA 145331A CA 962678 A CA962678 A CA 962678A
Authority
CA
Canada
Prior art keywords
benzothiazine
methylisoxazol
acetoxy
carbamoyl
dioxide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA145,331A
Other languages
English (en)
Other versions
CA145331S (en
Inventor
John Shavel (Jr.)
Martin L. Schwartz
Harold Zinnes
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Warner Lambert Co LLC
Original Assignee
Warner Lambert Co LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co LLC filed Critical Warner Lambert Co LLC
Application granted granted Critical
Publication of CA962678A publication Critical patent/CA962678A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
CA145,331A 1971-06-22 1972-06-21 4-acetoxy-2-methyl-3-(5-methylisoxazol-3-yl-carbamoyl)-2h-1,2-benzothiazine 1,1-dioxide Expired CA962678A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US15560571A 1971-06-22 1971-06-22

Publications (1)

Publication Number Publication Date
CA962678A true CA962678A (en) 1975-02-11

Family

ID=22556087

Family Applications (1)

Application Number Title Priority Date Filing Date
CA145,331A Expired CA962678A (en) 1971-06-22 1972-06-21 4-acetoxy-2-methyl-3-(5-methylisoxazol-3-yl-carbamoyl)-2h-1,2-benzothiazine 1,1-dioxide

Country Status (6)

Country Link
US (1) US3704298A (OSRAM)
JP (1) JPS5144953B1 (OSRAM)
CA (1) CA962678A (OSRAM)
DK (1) DK131152B (OSRAM)
FR (1) FR2143146B1 (OSRAM)
GB (1) GB1340289A (OSRAM)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3787324A (en) * 1971-03-01 1974-01-22 Warner Lambert Co 4-hydroxy-3-(3-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,dioxides and process for their production
US3957772A (en) * 1975-05-21 1976-05-18 Warner-Lambert Company Process for the preparation of 4-hydroxy-3-(5-methyl-3-isoxazolylcarbamoyl)-2-methyl-2h-1,2-benzothiazine 1,1-dioxide
US4474955A (en) * 1981-06-17 1984-10-02 Vincenzo Iannella Process for preparing 4-hydroxy-2-methyl-2H-1,2-benzothiazine-3-[N-(2-pyridinyl)carboxamide]-1,1-dioxide, and its phosphoric ester
JPS60184077A (ja) * 1984-02-23 1985-09-19 フアイザー・インコーポレーテツド 抗炎症性オキシム前駆薬
US4604458A (en) * 1984-07-31 1986-08-05 The Hilton-Davis Chemical Co. 3-substituted carbonyloxy-7-disubstituted amino-10-substituted carbonylphenothiazines
US4604461A (en) * 1984-07-31 1986-08-05 The Hilton-Davis Chemical Co. 5-substituted-9-disubstituted amino-12-substituted carbonylbenzo[a]phenoxazines
US4610982A (en) * 1985-06-03 1986-09-09 Pfizer Inc. Anti-inflammatory benzo- and thieno-1,2-thiazine-3-carboxamide 1,1-dioxide derivatives, compositions, and method of use therefor
US20090221703A1 (en) 2006-07-09 2009-09-03 Chongxi Yu High penetration composition and uses thereof
US20090238763A1 (en) * 2006-07-09 2009-09-24 Chongxi Yu High penetration compositions and uses thereof
EP2084165B1 (en) * 2006-10-11 2013-06-12 Techfields Biochem Co. Ltd Positively charged water-soluble prodrugs of oxicams and related compounds with very high skin penetration rate
KR101853971B1 (ko) * 2007-06-04 2018-05-02 테크필즈 인크 매우 높은 피부 및 막 침투율을 가지는 비스테로이드성 소염제(ｎｓａｉａ) 약물전구체 및 이들의 새로운 의약적 용도
KR101946297B1 (ko) 2008-12-04 2019-02-11 충시 위 고투과력을 가진 조성물 및 이의 적용

Also Published As

Publication number Publication date
FR2143146B1 (OSRAM) 1976-03-05
JPS5144953B1 (OSRAM) 1976-12-01
US3704298A (en) 1972-11-28
GB1340289A (en) 1973-12-12
DE2227742A1 (de) 1972-12-28
DK131152C (OSRAM) 1975-11-03
DE2227742B2 (OSRAM) 1975-07-03
DK131152B (da) 1975-06-02
FR2143146A1 (OSRAM) 1973-02-02

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