DK131152B - Analogifremgangsmåde til fremstilling af 4-acyloxy-3-(3-isoxazolocarbamyl)-2H-1,2-benzothiazin-1,1-dioxider. - Google Patents

Analogifremgangsmåde til fremstilling af 4-acyloxy-3-(3-isoxazolocarbamyl)-2H-1,2-benzothiazin-1,1-dioxider.

Info

Publication number
DK131152B
DK131152B DK310172AA DK310172A DK131152B DK 131152 B DK131152 B DK 131152B DK 310172A A DK310172A A DK 310172AA DK 310172 A DK310172 A DK 310172A DK 131152 B DK131152 B DK 131152B
Authority
DK
Denmark
Prior art keywords
isoxazolocarbamyl
benzothiazine
dioxides
acyloxy
preparation
Prior art date
Application number
DK310172AA
Other languages
English (en)
Other versions
DK131152C (da
Inventor
H Zinnes
M L Schwartz
J Shavel
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of DK131152B publication Critical patent/DK131152B/da
Application granted granted Critical
Publication of DK131152C publication Critical patent/DK131152C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
DK310172AA 1971-06-22 1972-06-21 Analogifremgangsmåde til fremstilling af 4-acyloxy-3-(3-isoxazolocarbamyl)-2H-1,2-benzothiazin-1,1-dioxider. DK131152B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US15560571A 1971-06-22 1971-06-22

Publications (2)

Publication Number Publication Date
DK131152B true DK131152B (da) 1975-06-02
DK131152C DK131152C (da) 1975-11-03

Family

ID=22556087

Family Applications (1)

Application Number Title Priority Date Filing Date
DK310172AA DK131152B (da) 1971-06-22 1972-06-21 Analogifremgangsmåde til fremstilling af 4-acyloxy-3-(3-isoxazolocarbamyl)-2H-1,2-benzothiazin-1,1-dioxider.

Country Status (6)

Country Link
US (1) US3704298A (da)
JP (1) JPS5144953B1 (da)
CA (1) CA962678A (da)
DK (1) DK131152B (da)
FR (1) FR2143146B1 (da)
GB (1) GB1340289A (da)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3787324A (en) * 1971-03-01 1974-01-22 Warner Lambert Co 4-hydroxy-3-(3-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,dioxides and process for their production
US3957772A (en) * 1975-05-21 1976-05-18 Warner-Lambert Company Process for the preparation of 4-hydroxy-3-(5-methyl-3-isoxazolylcarbamoyl)-2-methyl-2h-1,2-benzothiazine 1,1-dioxide
US4474955A (en) * 1981-06-17 1984-10-02 Vincenzo Iannella Process for preparing 4-hydroxy-2-methyl-2H-1,2-benzothiazine-3-[N-(2-pyridinyl)carboxamide]-1,1-dioxide, and its phosphoric ester
JPS60184077A (ja) * 1984-02-23 1985-09-19 フアイザー・インコーポレーテツド 抗炎症性オキシム前駆薬
US4604458A (en) * 1984-07-31 1986-08-05 The Hilton-Davis Chemical Co. 3-substituted carbonyloxy-7-disubstituted amino-10-substituted carbonylphenothiazines
US4604461A (en) * 1984-07-31 1986-08-05 The Hilton-Davis Chemical Co. 5-substituted-9-disubstituted amino-12-substituted carbonylbenzo[a]phenoxazines
US4610982A (en) * 1985-06-03 1986-09-09 Pfizer Inc. Anti-inflammatory benzo- and thieno-1,2-thiazine-3-carboxamide 1,1-dioxide derivatives, compositions, and method of use therefor
US20090221703A1 (en) 2006-07-09 2009-09-03 Chongxi Yu High penetration composition and uses thereof
US20090238763A1 (en) 2006-07-09 2009-09-24 Chongxi Yu High penetration compositions and uses thereof
CN101522692A (zh) * 2006-10-11 2009-09-02 于崇曦 具有快速皮肤穿透速度的带正电荷的水溶性的昔康及其相关化合物的前药
KR20180049144A (ko) * 2007-06-04 2018-05-10 테크필즈 인크 매우 높은 피부 및 막 침투율을 가지는 비스테로이드성 소염제(ｎｓａｉａ) 약물전구체 및 이들의 새로운 의약적 용도
JP2012511027A (ja) 2008-12-04 2012-05-17 チョンシー ユー 高透過性組成物およびその用途

Also Published As

Publication number Publication date
CA962678A (en) 1975-02-11
FR2143146A1 (da) 1973-02-02
DE2227742B2 (da) 1975-07-03
JPS5144953B1 (da) 1976-12-01
DE2227742A1 (de) 1972-12-28
FR2143146B1 (da) 1976-03-05
GB1340289A (en) 1973-12-12
DK131152C (da) 1975-11-03
US3704298A (en) 1972-11-28

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Legal Events

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PBP Patent lapsed