CA959841A - Isothiocyano-benzazole derivatives and processes for the production thereof - Google Patents

Isothiocyano-benzazole derivatives and processes for the production thereof

Info

Publication number
CA959841A
CA959841A CA025,922A CA25922A CA959841A CA 959841 A CA959841 A CA 959841A CA 25922 A CA25922 A CA 25922A CA 959841 A CA959841 A CA 959841A
Authority
CA
Canada
Prior art keywords
isothiocyano
processes
production
benzazole derivatives
benzazole
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA025,922A
Other languages
English (en)
Inventor
Alfred Margot
Paul Brenneisen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Individual
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Application granted granted Critical
Publication of CA959841A publication Critical patent/CA959841A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/56—Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/08—Radicals containing only hydrogen and carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/10—Radicals substituted by halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/12—Radicals substituted by oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/14—Radicals substituted by nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/16—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/18—Benzimidazoles; Hydrogenated benzimidazoles with aryl radicals directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/56—Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D263/57—Aryl or substituted aryl radicals
CA025,922A 1967-07-26 1968-07-25 Isothiocyano-benzazole derivatives and processes for the production thereof Expired CA959841A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH1062867A CH542853A (de) 1967-07-26 1967-07-26 Verfahren zur Herstellung neuer Isothiocyano-benzazol-Derivate

Publications (1)

Publication Number Publication Date
CA959841A true CA959841A (en) 1974-12-24

Family

ID=4365199

Family Applications (1)

Application Number Title Priority Date Filing Date
CA025,922A Expired CA959841A (en) 1967-07-26 1968-07-25 Isothiocyano-benzazole derivatives and processes for the production thereof

Country Status (14)

Country Link
US (1) US3586670A (de)
JP (1) JPS4843602B1 (de)
BE (1) BE718548A (de)
CA (1) CA959841A (de)
CH (1) CH542853A (de)
DE (1) DE1770981A1 (de)
DK (1) DK137988B (de)
ES (2) ES356463A1 (de)
FR (1) FR1587072A (de)
GB (1) GB1238867A (de)
IE (1) IE32210B1 (de)
IL (1) IL30429A (de)
NL (1) NL161059C (de)
OA (1) OA02865A (de)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3933841A (en) * 1971-05-24 1976-01-20 Ciba-Geigy Corporation 2-Phenoxy, -phenylthio-, and -phenyl-amino-benzoxazoles having an isothiocyano substituent
US3894037A (en) * 1971-05-24 1975-07-08 Ciba Geigy Corp Certain isothiocyanobenzimidazoles
BE792402A (fr) * 1971-12-07 1973-06-07 Ciba Geigy Composes heterocycliques azotes et medicaments anthelminthiqueset antimicrobiens qui en contiennent
US3934017A (en) * 1971-12-07 1976-01-20 Ciba-Geigy Corporation Anthelmintic composition and method utilizing isothiocyanobenzazoles active ingredients
US3983130A (en) * 1972-06-02 1976-09-28 E. R. Squibb & Sons, Inc. Anthelmintic isothiocyanobenzoxazoles
US3853894A (en) * 1972-06-02 1974-12-10 Squibb & Sons Inc Isothiocyanobenzimidazoles
US3985755A (en) * 1972-06-02 1976-10-12 E. R. Squibb & Sons, Inc. Pyridine containing isothiocyanobenzoxazoles
FR2162489A1 (en) * 1972-12-08 1973-07-20 Ciba Geigy Ag Isocyanato-benzoxazoles-benzothiazoles and benimidazoles - as anthelmintics and antimicrobials
US4046906A (en) * 1973-04-21 1977-09-06 Hoechst Aktiengesellschaft Salts of alkyl 2-benzimidazole-carbamate
US3864350A (en) * 1974-03-18 1975-02-04 Squibb & Sons Inc Pridyl-1H-benzimidazole N-oxides
DE2640730C2 (de) * 1976-09-10 1983-08-25 Hoechst Ag, 6230 Frankfurt Benzoxazolyloxy- und Benzothiazolyloxy-phenoxy-Verbindungen und diese enthaltende herbizide Mittel
CA1125768A (en) * 1978-10-31 1982-06-15 Hoffmann-La Roche Limited Benzoxazole derivatives
US5089592A (en) * 1988-06-09 1992-02-18 The Dow Chemical Company Biscyclobutarene monomer comprising two cyclobutarene moieties bridged by a divalent radical comprising at least one benzothiazole or benzimidazole linkage
US5104960A (en) * 1989-02-22 1992-04-14 The Dow Chemical Company Nucleophilic displacement method for synthesis of non-rigid PBZ polymers
US5216110A (en) * 1989-02-22 1993-06-01 The Dow Chemical Company Monomers useful in nucleophilic displacement synthesis of polybenzazole polymers
US5194562A (en) * 1989-02-22 1993-03-16 The Dow Chemical Company Nucleophilic displacement method for synthesis of non-rigid PBZ polymers
GB9312853D0 (en) * 1993-06-22 1993-08-04 Euro Celtique Sa Chemical compounds
US5591776A (en) * 1994-06-24 1997-01-07 Euro-Celtique, S.A. Pheynl or benzyl-substituted rolipram-based compounds for and method of inhibiting phosphodiesterase IV
US5922751A (en) * 1994-06-24 1999-07-13 Euro-Celtique, S.A. Aryl pyrazole compound for inhibiting phosphodiesterase IV and methods of using same
US5496826A (en) * 1994-09-02 1996-03-05 Bristol-Myers Squibb Company Pharmaceutical methods of using heterocyclic derivatives of N-phenylamides
US6372770B1 (en) 1994-10-12 2002-04-16 Euro-Celtique, S.A. Benzoxazoles
ATE248153T1 (de) * 1994-10-12 2003-09-15 Euro Celtique Sa Neue benzoxazole
DE69531555T2 (de) * 1994-12-13 2004-06-17 Euroceltique S.A. Dreifachsubstituierte thioxanthine
EP0814809B1 (de) * 1994-12-13 2003-08-13 Euroceltique S.A. Arylthioxanthine
US6025361A (en) * 1994-12-13 2000-02-15 Euro-Celtique, S.A. Trisubstituted thioxanthines
US6166041A (en) * 1995-10-11 2000-12-26 Euro-Celtique, S.A. 2-heteroaryl and 2-heterocyclic benzoxazoles as PDE IV inhibitors for the treatment of asthma
US6075016A (en) * 1996-04-10 2000-06-13 Euro-Celtique S.A. 6,5-fused aromatic ring systems having enhanced phosphodiesterase IV inhibitory activity
DE69727199T2 (de) * 1996-12-09 2004-11-18 Pfizer Inc. Benzimidazol-Verbindungen

Also Published As

Publication number Publication date
OA02865A (fr) 1970-12-15
JPS4843602B1 (de) 1973-12-19
IE32210L (en) 1969-01-26
IL30429A (en) 1973-06-29
US3586670A (en) 1971-06-22
GB1238867A (de) 1971-07-14
BE718548A (de) 1969-01-27
DK137988C (de) 1978-11-06
ES356462A1 (es) 1970-01-16
DE1770981A1 (de) 1972-01-13
NL161059B (nl) 1979-08-15
NL161059C (nl) 1980-01-15
CH542853A (de) 1973-10-15
DK137988B (da) 1978-06-19
FR1587072A (de) 1970-03-13
IL30429A0 (en) 1968-09-26
NL6810558A (de) 1969-01-28
ES356463A1 (es) 1970-01-16
IE32210B1 (en) 1973-05-16

Similar Documents

Publication Publication Date Title
CA959841A (en) Isothiocyano-benzazole derivatives and processes for the production thereof
CA952106A (en) Benzodiazepine derivatives and process for the manufacture thereof
CA959835A (en) Benzodiazepine derivatives and process for the manufacture thereof
CA949558A (en) Benzodiazepine derivatives and process for the manufacture thereof
CA948628A (en) Benzodiazepine derivatives and process for the manufacture thereof
CA969935A (en) Dibenzocycloheptene derivatives and process for the manufacture thereof
AU423811B2 (en) Bornane-methylamines and processes for the production thereof
CA751437A (en) Dihalogeno-amino-benzylamine derivatives and processes for their production
AU3143367A (en) Bornane-methylamines and processes for the production thereof
AU424523B2 (en) N-sulphonyl-2-phenyl-ethylamine derivatives and processes for their manufacture
CA949559A (en) Diphenylmethylenepyrrolidine derivatives and processes for preparing the same
CA752405A (en) Aminoisoxazoles and process for the manufacture thereof
CA756609A (en) Azapentanols and process for the manufacture thereof
CA759993A (en) Polyeneketones and process for the manufacture thereof
CA759392A (en) Photographic products and processes for the production thereof
CA760504A (en) Stable polyacetaldehydes and improved process for the production thereof
AU423465B2 (en) 5-benzylpyrimidine derivatives and process for the preparation thereof
AU421068B2 (en) Dibenzocycloheptene derivatives and process for the manufacture thereof
CA758122A (en) Phenylalanine derivatives and process for the manufacture thereof
AU2881167A (en) N-sulphonyl-2-phenyl-ethylamine derivatives and processes for their manufacture
CA754607A (en) Hydrazine derivatives and process for the manufacture thereof
AU421298B2 (en) 2-sulphonamidopyrimidine derivatives and process for their manufacture
AU283160B2 (en) Dibenzocyloheptene derivatives and their production
CA770133A (en) Benzodiazepin a derivatives and process for the manufacture thereof
CA768162A (en) Benzodiazepine derivatives and process for the manufacture thereof