CA951319A - Piperazinylalkyl-quinazolone-(4) derivatives, process for their production and pharmaceutical products containing them - Google Patents
Piperazinylalkyl-quinazolone-(4) derivatives, process for their production and pharmaceutical products containing themInfo
- Publication number
- CA951319A CA951319A CA114,709,A CA114709A CA951319A CA 951319 A CA951319 A CA 951319A CA 114709 A CA114709 A CA 114709A CA 951319 A CA951319 A CA 951319A
- Authority
- CA
- Canada
- Prior art keywords
- piperazinylalkyl
- quinazolone
- derivatives
- production
- products containing
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19702027645 DE2027645A1 (de) | 1970-06-05 | 1970-06-05 | Piperazinylalkyl chinazolon (4) den vate, Verfahren zu deren Herstellung und sie enthaltende Arzneimittel |
Publications (1)
Publication Number | Publication Date |
---|---|
CA951319A true CA951319A (en) | 1974-07-16 |
Family
ID=5773104
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA114,709,A Expired CA951319A (en) | 1970-06-05 | 1971-06-03 | Piperazinylalkyl-quinazolone-(4) derivatives, process for their production and pharmaceutical products containing them |
Country Status (10)
Country | Link |
---|---|
US (1) | US3984555A (sl) |
AT (3) | AT318615B (sl) |
BE (1) | BE768137A (sl) |
CA (1) | CA951319A (sl) |
CH (3) | CH569732A5 (sl) |
DE (1) | DE2027645A1 (sl) |
FR (1) | FR2100726B1 (sl) |
GB (1) | GB1331522A (sl) |
LU (1) | LU63267A1 (sl) |
NL (1) | NL7107695A (sl) |
Families Citing this family (32)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4287341A (en) * | 1979-11-01 | 1981-09-01 | Pfizer Inc. | Alkoxy-substituted-6-chloro-quinazoline-2,4-diones |
US6723727B1 (en) * | 1996-12-20 | 2004-04-20 | Hoechst Aktiengesellschaft | Substituted purine derivatives, processes for their preparation, their use, and compositions comprising them |
DE69842109D1 (de) * | 1997-08-21 | 2011-03-10 | Shiseido Co Ltd | Chinazolin-4-on Derivate, deren Herstellung und deren Verwendung als Haarwuchsmittel oder in äusserlich anzuwendenden Hautpflegemitteln |
US6436919B1 (en) | 1999-10-01 | 2002-08-20 | Theravance Inc. | Local anesthetic compounds |
US6667300B2 (en) | 2000-04-25 | 2003-12-23 | Icos Corporation | Inhibitors of human phosphatidylinositol 3-kinase delta |
ATE502941T1 (de) * | 2000-04-25 | 2011-04-15 | Icos Corp | Hemmer der menschlichen phosphatidyl-inositol-3- kinase delta |
AUPR201600A0 (en) * | 2000-12-11 | 2001-01-11 | Fujisawa Pharmaceutical Co., Ltd. | Quinazolinone derivative |
EP2116248A1 (en) | 2001-09-05 | 2009-11-11 | Minerva Biotechnologies Corporation | Compositions and Methods of Treatment of Cancer |
WO2003020280A2 (en) * | 2001-09-05 | 2003-03-13 | Minerva Biotechnologies Corporation | Compositions and use thereof in the treatment of cancer |
JP2005511581A (ja) | 2001-11-07 | 2005-04-28 | メルク エンド カムパニー インコーポレーテッド | 有糸分裂キネシン阻害剤 |
AUPS019702A0 (en) * | 2002-01-29 | 2002-02-21 | Fujisawa Pharmaceutical Co., Ltd. | Condensed heterocyclic compounds |
US20040048853A1 (en) * | 2002-08-21 | 2004-03-11 | Gustave Bergnes | Compounds, compositions, and methods |
EP1558260A4 (en) * | 2002-11-04 | 2006-10-25 | Nps Pharma Inc | CHINAZOLINONE COMPOUNDS AS CALCILYTIC |
WO2004111014A1 (en) * | 2003-06-06 | 2004-12-23 | Vertex Pharmaceuticals Incorporated | Pyrimidine derivatives as modulators of atp-binding cassette transporters |
US20050054614A1 (en) * | 2003-08-14 | 2005-03-10 | Diacovo Thomas G. | Methods of inhibiting leukocyte accumulation |
WO2005016348A1 (en) * | 2003-08-14 | 2005-02-24 | Icos Corporation | Method of inhibiting immune responses stimulated by an endogenous factor |
US7932260B2 (en) | 2004-05-13 | 2011-04-26 | Icos Corporation | Quinazolinones as inhibitors of human phosphatidylinositol 3-kinase delta |
EP1755609A1 (en) * | 2004-05-25 | 2007-02-28 | Icos Corporation | Methods for treating and/or preventing aberrant proliferation of hematopoietic cells |
EP1885356A2 (en) * | 2005-02-17 | 2008-02-13 | Icos Corporation | Phosphoinositide 3-kinase inhibitors for inhibiting leukocyte accumulation |
US8349850B2 (en) * | 2006-03-28 | 2013-01-08 | Atir Holding S.A. | Heterocyclic compounds and uses thereof in the treatment of sexual disorders |
US9492449B2 (en) | 2008-11-13 | 2016-11-15 | Gilead Calistoga Llc | Therapies for hematologic malignancies |
ES2674719T3 (es) | 2008-11-13 | 2018-07-03 | Gilead Calistoga Llc | Terapias para neoplasias hematológicas |
EP2411391A1 (en) | 2009-03-24 | 2012-02-01 | Gilead Calistoga LLC | Atropisomers of2-purinyl-3-tolyl-quinazolinone derivatives and methods of use |
CN102458410A (zh) * | 2009-04-20 | 2012-05-16 | 吉联亚·卡利斯托加有限责任公司 | 治疗实体瘤的方法 |
CN102647987A (zh) | 2009-07-21 | 2012-08-22 | 吉里德卡利斯托加公司 | 使用pi3k抑制剂治疗肝脏障碍 |
BRPI1003506B1 (pt) | 2010-09-24 | 2019-12-03 | Ache Int Bvi Ltd | composto alquil-piperazino-fenil-4(3h)quinazolinonas e uso do composto alquil-piperazino-fenil-4(3h)quinazolinonas associado aos receptores serotoninérgicos 5-ht1a e 5-ht2a |
CA2832822A1 (en) * | 2011-04-10 | 2012-10-18 | Atir Holding S.A. | Heterocyclic compounds and uses thereof in the treatment of sexual disorders |
AR090253A1 (es) | 2012-03-05 | 2014-10-29 | Gilead Calistoga Llc | Formas polimorficas de (s)-2-(1-(9h-purin-6-ilamino)propil)-5-fluor-3-fenilquinazolin-4(3h)-ona |
ES2595240T3 (es) | 2012-07-09 | 2016-12-28 | Lupin Limited | Derivados de tetrahidroquinazolinona como inhibidores de PARP |
MX2016008259A (es) | 2013-12-20 | 2016-10-13 | Gilead Calistoga Llc | Metodo de proceso para inhibidores de fosfatidilinositol 3-cinasa. |
US9708327B2 (en) | 2013-12-20 | 2017-07-18 | Gilead Calistoga Llc | Polymorphic forms of a hydrochloride salt of (S)-2-(1-(9H-purin-6-ylamino)propyl)-5-fluoro-3-phenylquinazolin-4(3H)-one |
SG11201609877XA (en) | 2014-06-13 | 2016-12-29 | Gilead Sciences Inc | Phosphatidylinositol 3-kinase inhibitors |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE1249281B (sl) * | 1963-05-18 |
-
1970
- 1970-06-05 DE DE19702027645 patent/DE2027645A1/de active Pending
-
1971
- 1971-05-28 US US05/148,100 patent/US3984555A/en not_active Expired - Lifetime
- 1971-06-01 AT AT470571A patent/AT318615B/de not_active IP Right Cessation
- 1971-06-01 AT AT244273A patent/AT317899B/de not_active IP Right Cessation
- 1971-06-01 AT AT244173A patent/AT318628B/de not_active IP Right Cessation
- 1971-06-02 CH CH450174A patent/CH569732A5/xx not_active IP Right Cessation
- 1971-06-02 CH CH450074A patent/CH558374A/xx not_active IP Right Cessation
- 1971-06-02 CH CH802071A patent/CH557829A/xx not_active IP Right Cessation
- 1971-06-02 LU LU63267D patent/LU63267A1/xx unknown
- 1971-06-03 GB GB1880371*[A patent/GB1331522A/en not_active Expired
- 1971-06-03 CA CA114,709,A patent/CA951319A/en not_active Expired
- 1971-06-04 FR FR7120368A patent/FR2100726B1/fr not_active Expired
- 1971-06-04 BE BE768137A patent/BE768137A/xx unknown
- 1971-06-04 NL NL7107695A patent/NL7107695A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
AT318628B (de) | 1974-11-11 |
AT318615B (de) | 1974-11-11 |
FR2100726B1 (sl) | 1975-10-10 |
NL7107695A (sl) | 1971-12-07 |
AT317899B (de) | 1974-09-25 |
GB1331522A (en) | 1973-09-26 |
CH558374A (de) | 1975-01-31 |
FR2100726A1 (sl) | 1972-03-24 |
US3984555A (en) | 1976-10-05 |
CH569732A5 (sl) | 1975-11-28 |
CH557829A (de) | 1975-01-15 |
LU63267A1 (sl) | 1972-08-23 |
DE2027645A1 (de) | 1971-12-09 |
BE768137A (fr) | 1971-12-06 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CA951319A (en) | Piperazinylalkyl-quinazolone-(4) derivatives, process for their production and pharmaceutical products containing them | |
CA923898A (en) | Process for the preparation of new phenyl-imidazolyl-alkanyl derivatives and products thereby produced | |
CA1008620A (en) | Process and apparatus for making pile-surfaced products | |
CA935025A (en) | Poultry product and process for producing same | |
AU471079B2 (en) | 5, 9, 13-prostatrienoic acid derivatives and process for their preparation | |
CA986140A (en) | 3,4-dihydroxy-benzylalcohol derivatives and process for preparing same | |
AU2207570A (en) | Pyridinesulfonic acids, process for their manufacture and pharmaceutical preparations containing them | |
CA971152A (en) | Product and process | |
IL36917A (en) | Dibenzothiepinopyrrole derivatives,their production and pharmaceutical compositions containing them | |
GB1407529A (en) | 1,2-dihydroindene-2-spiro-2-piperazine derivatives and process for production thereof | |
CA942304A (en) | Nitrofuryl-amidine derivatives and process for their preparation | |
CA963472A (en) | Cycloalkano-quinolone derivatives and process for their preparation | |
IL37888A (en) | 3-phenyl-2-alkoxycarbonylaminophenyl-6(7)alkoxycarbonylamino-4-quinazolone derivatives,their production and pharmaceutical compositions containing them | |
AU469309B2 (en) | Nitrofurane derivatives and process for production thereof | |
CA842787A (en) | Decomposition products of .delta.4,20,22-bufatrienolides and process for their separation | |
AU452006B2 (en) | 3 guanidinoalkyl thiphenes, process for their manufacture and pharmaceutical preparations containing them | |
AU425975B2 (en) | Novel 3, 4-dihydroxy-benzylalcohol derivatives and process for preparing same | |
CA840886A (en) | Process for preparing structural elements and product thereof | |
AU434713B2 (en) | Pharmaceutical preparatins containing glucose compounds, glucose derivatives and process for their manufacture | |
AU2749571A (en) | 3 guanidinoalkyl thiphenes, process for their manufacture and pharmaceutical preparations containing them | |
CA859756A (en) | Naphthyridene derivatives and processes for their production | |
AU475269B2 (en) | Process for preparing 1,2,4,5-tetrahydro-3h, 3-benzazepines and products obtained thereby | |
CA832484A (en) | Substituted 1-phenoxy-3-alkylamino-propanoles(2) and process for their production | |
CA845073A (en) | Process for preparing cereal product | |
CA848916A (en) | Process for preparing cereal product |