CA3164650A1 - Compound and composition as pdgf receptor kinase inhibitor - Google Patents

Compound and composition as pdgf receptor kinase inhibitor

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Publication number
CA3164650A1
CA3164650A1 CA3164650A CA3164650A CA3164650A1 CA 3164650 A1 CA3164650 A1 CA 3164650A1 CA 3164650 A CA3164650 A CA 3164650A CA 3164650 A CA3164650 A CA 3164650A CA 3164650 A1 CA3164650 A1 CA 3164650A1
Authority
CA
Canada
Prior art keywords
hydroxycyclohexyl
methyl
carboxamide
pyridin
amino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CA3164650A
Other languages
English (en)
French (fr)
Inventor
Junshi ASADA
Yoshinari Haruta
Hiroyuki YAKUSHIJI
Toru Tanaka
Kazuya Kuramoto
Keiji KOSUGI
Chiaki FUCHIKAMI
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Nippon Shinyaku Co Ltd
Original Assignee
Nippon Shinyaku Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nippon Shinyaku Co Ltd filed Critical Nippon Shinyaku Co Ltd
Publication of CA3164650A1 publication Critical patent/CA3164650A1/en
Pending legal-status Critical Current

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    • A61K31/00—Medicinal preparations containing organic active ingredients
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/421—1,3-Oxazoles, e.g. pemoline, trimethadione
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