CA3116533A1 - Methodes de traitement de la nephropathie chronique au moyen de la dapagliflozine - Google Patents
Methodes de traitement de la nephropathie chronique au moyen de la dapagliflozine Download PDFInfo
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- CA3116533A1 CA3116533A1 CA3116533A CA3116533A CA3116533A1 CA 3116533 A1 CA3116533 A1 CA 3116533A1 CA 3116533 A CA3116533 A CA 3116533A CA 3116533 A CA3116533 A CA 3116533A CA 3116533 A1 CA3116533 A1 CA 3116533A1
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- 229960001288 triamterene Drugs 0.000 description 1
- 229960004813 trichlormethiazide Drugs 0.000 description 1
- LMJSLTNSBFUCMU-UHFFFAOYSA-N trichlormethiazide Chemical compound C1=C(Cl)C(S(=O)(=O)N)=CC2=C1NC(C(Cl)Cl)NS2(=O)=O LMJSLTNSBFUCMU-UHFFFAOYSA-N 0.000 description 1
- 229960001641 troglitazone Drugs 0.000 description 1
- GXPHKUHSUJUWKP-UHFFFAOYSA-N troglitazone Chemical compound C1CC=2C(C)=C(O)C(C)=C(C)C=2OC1(C)COC(C=C1)=CC=C1CC1SC(=O)NC1=O GXPHKUHSUJUWKP-UHFFFAOYSA-N 0.000 description 1
- GXPHKUHSUJUWKP-NTKDMRAZSA-N troglitazone Natural products C([C@@]1(OC=2C(C)=C(C(=C(C)C=2CC1)O)C)C)OC(C=C1)=CC=C1C[C@H]1SC(=O)NC1=O GXPHKUHSUJUWKP-NTKDMRAZSA-N 0.000 description 1
- 229940116269 uric acid Drugs 0.000 description 1
- 230000002485 urinary effect Effects 0.000 description 1
- 230000002792 vascular Effects 0.000 description 1
- 208000019553 vascular disease Diseases 0.000 description 1
- 230000002861 ventricular Effects 0.000 description 1
- 229960001722 verapamil Drugs 0.000 description 1
- 238000012795 verification Methods 0.000 description 1
- 229960001254 vildagliptin Drugs 0.000 description 1
- SYOKIDBDQMKNDQ-XWTIBIIYSA-N vildagliptin Chemical compound C1C(O)(C2)CC(C3)CC1CC32NCC(=O)N1CCC[C@H]1C#N SYOKIDBDQMKNDQ-XWTIBIIYSA-N 0.000 description 1
- 230000009278 visceral effect Effects 0.000 description 1
- 229940015903 xigduo Drugs 0.000 description 1
- 229960002769 zofenopril Drugs 0.000 description 1
- IAIDUHCBNLFXEF-MNEFBYGVSA-N zofenopril Chemical compound C([C@@H](C)C(=O)N1[C@@H](C[C@@H](C1)SC=1C=CC=CC=1)C(O)=O)SC(=O)C1=CC=CC=C1 IAIDUHCBNLFXEF-MNEFBYGVSA-N 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7004—Monosaccharides having only carbon, hydrogen and oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
- A61K31/351—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom not condensed with another ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7028—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
- A61K31/7034—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/401—Proline; Derivatives thereof, e.g. captopril
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Molecular Biology (AREA)
- Urology & Nephrology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (15)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202063057139P | 2020-07-27 | 2020-07-27 | |
| US63/057,139 | 2020-07-27 | ||
| US202063070869P | 2020-08-27 | 2020-08-27 | |
| US63/070,869 | 2020-08-27 | ||
| US202063082524P | 2020-09-24 | 2020-09-24 | |
| US63/082,524 | 2020-09-24 | ||
| US202063093961P | 2020-10-20 | 2020-10-20 | |
| US63/093,961 | 2020-10-20 | ||
| US202063119711P | 2020-12-01 | 2020-12-01 | |
| US63/119,711 | 2020-12-01 | ||
| US202163152445P | 2021-02-23 | 2021-02-23 | |
| US63/152,445 | 2021-02-23 | ||
| US202163161629P | 2021-03-16 | 2021-03-16 | |
| US63/161,629 | 2021-03-16 | ||
| PCT/EP2021/058727 WO2022022865A1 (fr) | 2020-07-27 | 2021-04-01 | Procédés de traitement d'une maladie rénale chronique avec de la dapagliflozine |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA3116533A1 true CA3116533A1 (fr) | 2022-01-27 |
Family
ID=79551924
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA3116533A Pending CA3116533A1 (fr) | 2020-07-27 | 2021-04-01 | Methodes de traitement de la nephropathie chronique au moyen de la dapagliflozine |
Country Status (13)
| Country | Link |
|---|---|
| EP (1) | EP4188389A1 (fr) |
| JP (1) | JP2023536009A (fr) |
| KR (2) | KR20220097854A (fr) |
| CN (3) | CN116392472A (fr) |
| AU (2) | AU2021202643B2 (fr) |
| BR (1) | BR112021008094A2 (fr) |
| CA (1) | CA3116533A1 (fr) |
| CR (1) | CR20210222A (fr) |
| DO (1) | DOP2021000083A (fr) |
| IL (2) | IL311682A (fr) |
| JO (1) | JOP20210087A1 (fr) |
| MX (1) | MX2021005191A (fr) |
| PE (1) | PE20231306A1 (fr) |
-
2021
- 2021-04-01 BR BR112021008094A patent/BR112021008094A2/pt unknown
- 2021-04-01 CN CN202310547700.1A patent/CN116392472A/zh active Pending
- 2021-04-01 KR KR1020217013222A patent/KR20220097854A/ko not_active IP Right Cessation
- 2021-04-01 MX MX2021005191A patent/MX2021005191A/es unknown
- 2021-04-01 PE PE2021000657A patent/PE20231306A1/es unknown
- 2021-04-01 CA CA3116533A patent/CA3116533A1/fr active Pending
- 2021-04-01 JP JP2021523830A patent/JP2023536009A/ja active Pending
- 2021-04-01 CN CN202210071080.4A patent/CN114209689B/zh active Active
- 2021-04-01 AU AU2021202643A patent/AU2021202643B2/en active Active
- 2021-04-01 CN CN202180001003.5A patent/CN114630682A/zh active Pending
- 2021-04-01 CR CR20210222A patent/CR20210222A/es unknown
- 2021-04-01 KR KR1020237034971A patent/KR20230149329A/ko active Search and Examination
- 2021-04-01 IL IL311682A patent/IL311682A/en unknown
- 2021-04-01 JO JOP/2021/0087A patent/JOP20210087A1/ar unknown
- 2021-04-01 EP EP21716724.6A patent/EP4188389A1/fr active Pending
- 2021-04-26 IL IL282665A patent/IL282665A/en unknown
- 2021-05-03 DO DO2021000083A patent/DOP2021000083A/es unknown
-
2023
- 2023-04-24 AU AU2023202490A patent/AU2023202490A1/en active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| IL282665A (en) | 2021-12-01 |
| KR20230149329A (ko) | 2023-10-26 |
| AU2021202643A1 (en) | 2022-02-10 |
| BR112021008094A2 (pt) | 2022-02-22 |
| CN116392472A (zh) | 2023-07-07 |
| CN114209689B (zh) | 2023-02-17 |
| KR20220097854A (ko) | 2022-07-08 |
| CN114209689A (zh) | 2022-03-22 |
| CN114630682A (zh) | 2022-06-14 |
| MX2021005191A (es) | 2022-04-18 |
| DOP2021000083A (es) | 2022-04-18 |
| AU2023202490A1 (en) | 2023-05-11 |
| EP4188389A1 (fr) | 2023-06-07 |
| CR20210222A (es) | 2022-08-29 |
| JP2023536009A (ja) | 2023-08-23 |
| PE20231306A1 (es) | 2023-08-24 |
| JOP20210087A1 (ar) | 2023-01-30 |
| AU2021202643B2 (en) | 2023-02-02 |
| IL311682A (en) | 2024-05-01 |
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