CA3074923A1 - Novel salts - Google Patents
Novel salts Download PDFInfo
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- CA3074923A1 CA3074923A1 CA3074923A CA3074923A CA3074923A1 CA 3074923 A1 CA3074923 A1 CA 3074923A1 CA 3074923 A CA3074923 A CA 3074923A CA 3074923 A CA3074923 A CA 3074923A CA 3074923 A1 CA3074923 A1 CA 3074923A1
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- Prior art keywords
- compound
- methyl
- disorder
- salt
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- 239000003053 toxin Substances 0.000 description 1
- 231100000765 toxin Toxicity 0.000 description 1
- 108700012359 toxins Proteins 0.000 description 1
- 239000000196 tragacanth Substances 0.000 description 1
- 235000010487 tragacanth Nutrition 0.000 description 1
- 229940116362 tragacanth Drugs 0.000 description 1
- 230000001052 transient effect Effects 0.000 description 1
- 201000005142 transvestism Diseases 0.000 description 1
- 229960003741 tranylcypromine Drugs 0.000 description 1
- 230000008733 trauma Effects 0.000 description 1
- 230000009529 traumatic brain injury Effects 0.000 description 1
- 229960003991 trazodone Drugs 0.000 description 1
- PHLBKPHSAVXXEF-UHFFFAOYSA-N trazodone Chemical compound ClC1=CC=CC(N2CCN(CCCN3C(N4C=CC=CC4=N3)=O)CC2)=C1 PHLBKPHSAVXXEF-UHFFFAOYSA-N 0.000 description 1
- JOFWLTCLBGQGBO-UHFFFAOYSA-N triazolam Chemical compound C12=CC(Cl)=CC=C2N2C(C)=NN=C2CN=C1C1=CC=CC=C1Cl JOFWLTCLBGQGBO-UHFFFAOYSA-N 0.000 description 1
- 229960003386 triazolam Drugs 0.000 description 1
- QORWJWZARLRLPR-UHFFFAOYSA-H tricalcium bis(phosphate) Chemical compound [Ca+2].[Ca+2].[Ca+2].[O-]P([O-])([O-])=O.[O-]P([O-])([O-])=O QORWJWZARLRLPR-UHFFFAOYSA-H 0.000 description 1
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- ZEWQUBUPAILYHI-UHFFFAOYSA-N trifluoperazine Chemical compound C1CN(C)CCN1CCCN1C2=CC(C(F)(F)F)=CC=C2SC2=CC=CC=C21 ZEWQUBUPAILYHI-UHFFFAOYSA-N 0.000 description 1
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- 230000001960 triggered effect Effects 0.000 description 1
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- LNPDTQAFDNKSHK-UHFFFAOYSA-N valdecoxib Chemical compound CC=1ON=C(C=2C=CC=CC=2)C=1C1=CC=C(S(N)(=O)=O)C=C1 LNPDTQAFDNKSHK-UHFFFAOYSA-N 0.000 description 1
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- HUNXMJYCHXQEGX-UHFFFAOYSA-N zaleplon Chemical compound CCN(C(C)=O)C1=CC=CC(C=2N3N=CC(=C3N=CC=2)C#N)=C1 HUNXMJYCHXQEGX-UHFFFAOYSA-N 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/10—Spiro-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Neurosurgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201762564744P | 2017-09-28 | 2017-09-28 | |
| US62/564,744 | 2017-09-28 | ||
| PCT/US2018/053520 WO2019067961A1 (en) | 2017-09-28 | 2018-09-28 | NEW SALTS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA3074923A1 true CA3074923A1 (en) | 2019-04-04 |
Family
ID=65902742
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA3074923A Withdrawn CA3074923A1 (en) | 2017-09-28 | 2018-09-28 | Novel salts |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US20200255438A1 (enExample) |
| EP (1) | EP3687533A4 (enExample) |
| JP (1) | JP2020536070A (enExample) |
| KR (1) | KR20200060404A (enExample) |
| CN (1) | CN111343978A (enExample) |
| AU (2) | AU2018338884A1 (enExample) |
| BR (1) | BR112020005992A2 (enExample) |
| CA (1) | CA3074923A1 (enExample) |
| EA (1) | EA202090853A1 (enExample) |
| IL (1) | IL273520A (enExample) |
| MA (1) | MA50669A (enExample) |
| MX (1) | MX2020003741A (enExample) |
| SG (1) | SG11202002200UA (enExample) |
| WO (1) | WO2019067961A1 (enExample) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA3077088A1 (en) | 2017-10-10 | 2019-04-18 | Biogen Inc. | Process for preparing spiro derivatives |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2789711C (en) * | 2010-02-17 | 2014-08-05 | Amgen Inc. | Aryl carboxamide derivatives as sodium channel inhibitors for treatment of pain |
| EA201491990A1 (ru) * | 2012-05-03 | 2015-02-27 | Новартис Аг | L-малатная соль 2,7-диазаспиро[4.5]дец-7-иловых производных и их кристаллические формы в качестве агонистов грелиновых рецепторов |
| GB201209015D0 (en) * | 2012-05-22 | 2012-07-04 | Convergence Pharmaceuticals | Novel compounds |
-
2018
- 2018-09-28 MX MX2020003741A patent/MX2020003741A/es unknown
- 2018-09-28 EP EP18861356.6A patent/EP3687533A4/en not_active Withdrawn
- 2018-09-28 MA MA050669A patent/MA50669A/fr unknown
- 2018-09-28 EA EA202090853A patent/EA202090853A1/ru unknown
- 2018-09-28 WO PCT/US2018/053520 patent/WO2019067961A1/en not_active Ceased
- 2018-09-28 US US16/651,577 patent/US20200255438A1/en not_active Abandoned
- 2018-09-28 JP JP2020518078A patent/JP2020536070A/ja not_active Withdrawn
- 2018-09-28 SG SG11202002200UA patent/SG11202002200UA/en unknown
- 2018-09-28 CA CA3074923A patent/CA3074923A1/en not_active Withdrawn
- 2018-09-28 BR BR112020005992-7A patent/BR112020005992A2/pt not_active Application Discontinuation
- 2018-09-28 AU AU2018338884A patent/AU2018338884A1/en not_active Abandoned
- 2018-09-28 CN CN201880063113.2A patent/CN111343978A/zh not_active Withdrawn
- 2018-09-28 KR KR1020207009445A patent/KR20200060404A/ko not_active Withdrawn
-
2020
- 2020-03-23 IL IL273520A patent/IL273520A/en unknown
-
2023
- 2023-04-13 AU AU2023202293A patent/AU2023202293A1/en not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| AU2023202293A1 (en) | 2023-05-11 |
| EP3687533A4 (en) | 2021-01-20 |
| JP2020536070A (ja) | 2020-12-10 |
| MA50669A (fr) | 2020-08-05 |
| AU2018338884A1 (en) | 2020-04-16 |
| IL273520A (en) | 2020-05-31 |
| KR20200060404A (ko) | 2020-05-29 |
| SG11202002200UA (en) | 2020-04-29 |
| MX2020003741A (es) | 2021-01-08 |
| BR112020005992A2 (pt) | 2020-09-29 |
| US20200255438A1 (en) | 2020-08-13 |
| EA202090853A1 (ru) | 2020-08-27 |
| CN111343978A (zh) | 2020-06-26 |
| WO2019067961A1 (en) | 2019-04-04 |
| EP3687533A1 (en) | 2020-08-05 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AZWI | Withdrawn application |
Effective date: 20230824 |