CA3006999A1 - Gastric retentive devices - Google Patents
Gastric retentive devices Download PDFInfo
- Publication number
- CA3006999A1 CA3006999A1 CA3006999A CA3006999A CA3006999A1 CA 3006999 A1 CA3006999 A1 CA 3006999A1 CA 3006999 A CA3006999 A CA 3006999A CA 3006999 A CA3006999 A CA 3006999A CA 3006999 A1 CA3006999 A1 CA 3006999A1
- Authority
- CA
- Canada
- Prior art keywords
- hours
- enteric polymer
- hpmcas
- subject
- coating
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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- 238000000034 method Methods 0.000 claims abstract description 51
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- 239000003814 drug Substances 0.000 claims description 44
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- MLKXDPUZXIRXEP-MFOYZWKCSA-N sulindac Chemical compound CC1=C(CC(O)=O)C2=CC(F)=CC=C2\C1=C/C1=CC=C(S(C)=O)C=C1 MLKXDPUZXIRXEP-MFOYZWKCSA-N 0.000 description 1
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Classifications
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- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
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- A61M31/002—Devices for releasing a drug at a continuous and controlled rate for a prolonged period of time
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- A—HUMAN NECESSITIES
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- B29K2105/00—Condition, form or state of moulded material or of the material to be shaped
- B29K2105/0005—Condition, form or state of moulded material or of the material to be shaped containing compounding ingredients
- B29K2105/0035—Medical or pharmaceutical agents
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- B—PERFORMING OPERATIONS; TRANSPORTING
- B29—WORKING OF PLASTICS; WORKING OF SUBSTANCES IN A PLASTIC STATE IN GENERAL
- B29K—INDEXING SCHEME ASSOCIATED WITH SUBCLASSES B29B, B29C OR B29D, RELATING TO MOULDING MATERIALS OR TO MATERIALS FOR MOULDS, REINFORCEMENTS, FILLERS OR PREFORMED PARTS, e.g. INSERTS
- B29K2105/00—Condition, form or state of moulded material or of the material to be shaped
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- B—PERFORMING OPERATIONS; TRANSPORTING
- B29—WORKING OF PLASTICS; WORKING OF SUBSTANCES IN A PLASTIC STATE IN GENERAL
- B29K—INDEXING SCHEME ASSOCIATED WITH SUBCLASSES B29B, B29C OR B29D, RELATING TO MOULDING MATERIALS OR TO MATERIALS FOR MOULDS, REINFORCEMENTS, FILLERS OR PREFORMED PARTS, e.g. INSERTS
- B29K2105/00—Condition, form or state of moulded material or of the material to be shaped
- B29K2105/0094—Condition, form or state of moulded material or of the material to be shaped having particular viscosity
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Inorganic Chemistry (AREA)
- Nutrition Science (AREA)
- Hematology (AREA)
- Physiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Biomedical Technology (AREA)
- Anesthesiology (AREA)
- Mechanical Engineering (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Manufacturing & Machinery (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201562261752P | 2015-12-01 | 2015-12-01 | |
| US62/261,752 | 2015-12-01 | ||
| PCT/US2016/064439 WO2017096054A1 (en) | 2015-12-01 | 2016-12-01 | Gastric retentive devices |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA3006999A1 true CA3006999A1 (en) | 2017-06-08 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA3006999A Abandoned CA3006999A1 (en) | 2015-12-01 | 2016-12-01 | Gastric retentive devices |
Country Status (8)
| Country | Link |
|---|---|
| US (2) | US11147766B2 (enExample) |
| EP (1) | EP3383365A1 (enExample) |
| JP (1) | JP2018536007A (enExample) |
| CN (1) | CN108601724A (enExample) |
| AU (1) | AU2016365321A1 (enExample) |
| CA (1) | CA3006999A1 (enExample) |
| IL (1) | IL259584A (enExample) |
| WO (1) | WO2017096054A1 (enExample) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN106535878B (zh) * | 2014-06-02 | 2022-11-01 | 科莱西奥生物科技有限公司 | 可张开的胃内滞留剂型 |
| CN118975972A (zh) | 2015-10-23 | 2024-11-19 | 林德拉治疗公司 | 用于治疗剂缓释的胃驻留系统及其使用方法 |
| EP3383365A1 (en) * | 2015-12-01 | 2018-10-10 | Clexio Biosciences Ltd. | Gastric retentive devices |
| BR112018011636B1 (pt) | 2015-12-08 | 2024-03-12 | Lyndra Therapeutics, Inc | Sistema de residência gástrico para liberação sustentada de um agente terapêutico |
| CN119925721A (zh) | 2016-05-27 | 2025-05-06 | 林德拉治疗公司 | 用于胃驻留系统的材料结构 |
| CN110022861B (zh) | 2016-09-30 | 2024-06-28 | 林德拉治疗公司 | 用于金刚烷类药物缓释的胃驻留系统 |
| AU2018279853B2 (en) | 2017-06-09 | 2024-07-04 | Lyndra Therapeutics, Inc. | Gastric residence systems with release rate-modulating films |
| WO2020230089A1 (en) | 2019-05-14 | 2020-11-19 | Clexio Biosciences Ltd. | Treatment of nocturnal symptoms and morning akinesia in subjects with parkinson's disease |
| WO2022195476A1 (en) | 2021-03-15 | 2022-09-22 | Clexio Biosciences Ltd. | Gastroretentive devices for assessment of intragastric conditions |
| IL320492A (en) | 2022-10-25 | 2025-06-01 | Veradermics Incorporated | Compositions and methods of use for modified release minoxidil |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU449029B2 (en) | 1969-08-28 | 1974-04-17 | Commonwealth Scientific And Industrial Research Organisation | Device for administration to ruminants |
| US4735804A (en) | 1985-05-10 | 1988-04-05 | Merck & Co., Inc. | Drug delivery device which can be retained in the stomach for a controlled period of time |
| US4767627A (en) | 1985-05-29 | 1988-08-30 | Merck & Co., Inc. | Drug delivery device which can be retained in the stomach for a controlled period of time |
| US5002772A (en) * | 1988-05-31 | 1991-03-26 | Pfizer Inc. | Gastric retention system for controlled drug release |
| IL133196A0 (en) * | 1999-11-29 | 2001-03-19 | Yissum Res Dev Co | Gastroretentive controlled release pharmaceutical dosage forms |
| CA2613178A1 (en) | 2005-07-15 | 2007-01-25 | Kissei Pharmaceutical Co., Ltd. | Sustained release preparation |
| EP1945189A4 (en) * | 2005-11-03 | 2012-08-15 | Sun Pharmaceutical Ind Ltd | CONTROLLED RELEASE COATED TABLETS CHARACTERIZED BY PROLONGED GASTRIC RETENTION |
| US8298574B2 (en) | 2006-01-18 | 2012-10-30 | Intec Pharma Ltd. | Method and apparatus for forming delivery devices for oral intake of an agent |
| ES2606395T3 (es) * | 2008-04-18 | 2017-03-23 | Intec Pharma Ltd. | Administración de fármacos gastrorretentivos para carbidopa/levodopa |
| JP2012500230A (ja) | 2008-08-18 | 2012-01-05 | 北京天衡▲薬▼物研究院 | 胃内滞留薬物放出システム及びその製造方法と使用 |
| US20110066175A1 (en) * | 2009-05-07 | 2011-03-17 | Rainbow Medical Ltd. | Gastric anchor |
| CN106535878B (zh) * | 2014-06-02 | 2022-11-01 | 科莱西奥生物科技有限公司 | 可张开的胃内滞留剂型 |
| JP6666858B2 (ja) * | 2014-06-11 | 2020-03-18 | マサチューセッツ インスティテュート オブ テクノロジー | 滞留構造体および関連方法 |
| EP3383365A1 (en) * | 2015-12-01 | 2018-10-10 | Clexio Biosciences Ltd. | Gastric retentive devices |
| JP2018537201A (ja) * | 2015-12-02 | 2018-12-20 | クレキシオ バイオサイエンシーズ エルティーディー． | 胃保持型投与形態を調整する装置および方法 |
| IL266377B2 (en) * | 2016-12-02 | 2023-10-01 | Clexio Biosciences Ltd | Gastric residence system |
-
2016
- 2016-12-01 EP EP16820048.3A patent/EP3383365A1/en not_active Withdrawn
- 2016-12-01 WO PCT/US2016/064439 patent/WO2017096054A1/en not_active Ceased
- 2016-12-01 CA CA3006999A patent/CA3006999A1/en not_active Abandoned
- 2016-12-01 AU AU2016365321A patent/AU2016365321A1/en not_active Abandoned
- 2016-12-01 JP JP2018529014A patent/JP2018536007A/ja active Pending
- 2016-12-01 CN CN201680070026.0A patent/CN108601724A/zh active Pending
- 2016-12-01 US US15/780,420 patent/US11147766B2/en active Active
-
2018
- 2018-05-24 IL IL259584A patent/IL259584A/en unknown
-
2021
- 2021-09-20 US US17/479,131 patent/US20220008334A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| AU2016365321A1 (en) | 2018-06-21 |
| WO2017096054A1 (en) | 2017-06-08 |
| EP3383365A1 (en) | 2018-10-10 |
| US20220008334A1 (en) | 2022-01-13 |
| WO2017096054A9 (en) | 2017-09-08 |
| JP2018536007A (ja) | 2018-12-06 |
| US20180369138A1 (en) | 2018-12-27 |
| US11147766B2 (en) | 2021-10-19 |
| CN108601724A (zh) | 2018-09-28 |
| IL259584A (en) | 2018-07-31 |
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| FZDE | Discontinued |
Effective date: 20220601 |
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| FZDE | Discontinued |
Effective date: 20220601 |