CA3004028C - Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives - Google Patents

Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives Download PDF

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Publication number
CA3004028C
CA3004028C CA3004028A CA3004028A CA3004028C CA 3004028 C CA3004028 C CA 3004028C CA 3004028 A CA3004028 A CA 3004028A CA 3004028 A CA3004028 A CA 3004028A CA 3004028 C CA3004028 C CA 3004028C
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Canada
Prior art keywords
balsalazide
administration
food
subject
asa
Prior art date
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Active
Application number
CA3004028A
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English (en)
French (fr)
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CA3004028A1 (en
Inventor
Lorin Johnson
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Salix Pharmaceuticals Inc
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Salix Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
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Publication of CA3004028A1 publication Critical patent/CA3004028A1/en
Application granted granted Critical
Publication of CA3004028C publication Critical patent/CA3004028C/en
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Anticipated expiration legal-status Critical

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/60—Salicylic acid; Derivatives thereof
    • A61K31/606—Salicylic acid; Derivatives thereof having amino groups
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/63—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
    • A61K31/635—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide having a heterocyclic ring, e.g. sulfadiazine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/655—Azo (—N=N—), diazo (=N2), azoxy (>N—O—N< or N(=O)—N<), azido (—N3) or diazoamino (—N=N—N<) compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
CA3004028A 2006-11-03 2007-03-23 Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives Active CA3004028C (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US11/592,854 2006-11-03
US11/592,854 US8921344B2 (en) 2006-11-03 2006-11-03 Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives
CA2668441A CA2668441C (en) 2006-11-03 2007-03-23 Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
CA2668441A Division CA2668441C (en) 2006-11-03 2007-03-23 Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives

Publications (2)

Publication Number Publication Date
CA3004028A1 CA3004028A1 (en) 2008-05-29
CA3004028C true CA3004028C (en) 2021-07-13

Family

ID=38263983

Family Applications (2)

Application Number Title Priority Date Filing Date
CA2668441A Active CA2668441C (en) 2006-11-03 2007-03-23 Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives
CA3004028A Active CA3004028C (en) 2006-11-03 2007-03-23 Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives

Family Applications Before (1)

Application Number Title Priority Date Filing Date
CA2668441A Active CA2668441C (en) 2006-11-03 2007-03-23 Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives

Country Status (12)

Country Link
US (1) US8921344B2 (enExample)
EP (1) EP2096912B1 (enExample)
JP (2) JP6067203B2 (enExample)
KR (2) KR20090118906A (enExample)
CN (1) CN101610670A (enExample)
AU (1) AU2007322362B2 (enExample)
BR (1) BRPI0717859A2 (enExample)
CA (2) CA2668441C (enExample)
DK (1) DK2096912T3 (enExample)
IL (1) IL198513B (enExample)
MX (1) MX2009004826A (enExample)
WO (1) WO2008063211A2 (enExample)

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CA2359812C (en) 2000-11-20 2004-02-10 The Procter & Gamble Company Pharmaceutical dosage form with multiple coatings for reduced impact of coating fractures
HUE029189T2 (en) 2004-02-06 2017-02-28 Pharmatel (R&D) Pty Ltd As Trustee For The Pharmatel (R & D) Trust The use of aminosalicylates in diarrhea prodominant irritable bowel syndrome
US8497258B2 (en) 2005-11-12 2013-07-30 The Regents Of The University Of California Viscous budesonide for the treatment of inflammatory diseases of the gastrointestinal tract
US7541384B2 (en) 2007-06-08 2009-06-02 Axcan Pharma Inc. Mesalamine suppository
US8436051B2 (en) 2007-06-08 2013-05-07 Aptalis Pharma Canada Inc. Mesalamine suppository
US8217083B2 (en) * 2007-06-08 2012-07-10 Aptalis Pharma Canada Inc. Mesalamine suppository
ITMI20071965A1 (it) * 2007-10-11 2009-04-12 Domenico Russo Composizione farmaceutica comprendente sucralfato e mesalazina
WO2010040021A1 (en) * 2008-10-03 2010-04-08 Salix Pharmaceuticals, Ltd. Compositions and methods for the treatment of bowel diseases with granulated mesalamine
US20120111756A1 (en) * 2008-12-17 2012-05-10 Altheus Therapeutics, Inc. Enema formulations
WO2010144865A2 (en) 2009-06-12 2010-12-16 Meritage Pharma, Inc. Methods for treating gastrointestinal disorders
EP2563117B1 (en) * 2010-04-26 2018-02-21 Salix Pharmaceuticals, Ltd. Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives for the treatment of males
JP6008866B2 (ja) * 2010-12-03 2016-10-19 オレキシジェン・セラピューティクス・インコーポレーテッド ナルトレキソン療法における薬物バイオアベイラビリティの増加
CN103483220B (zh) * 2013-06-09 2015-06-17 陕西新药技术开发中心 一种化合物及其制备方法和抗溃疡性结肠炎用途
CN103333084B (zh) * 2013-06-09 2015-01-07 陕西新药技术开发中心 3,3’-偶氮双[6-(丁酰氧基)苯甲酸]及其制备方法和应用
CN104706582A (zh) * 2013-12-12 2015-06-17 四川健能制药有限公司 含有美沙拉秦的药物组合物
US10100005B1 (en) * 2017-11-17 2018-10-16 Eclipse Therapeutics, LLC Mesalazine derivatives
JP2020090456A (ja) * 2018-12-05 2020-06-11 日本化薬株式会社 エルロチニブを有効成分とする医薬錠剤

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Also Published As

Publication number Publication date
AU2007322362B2 (en) 2013-06-20
JP6067203B2 (ja) 2017-01-25
JP2013032395A (ja) 2013-02-14
CA2668441C (en) 2018-06-12
BRPI0717859A2 (pt) 2013-01-22
IL198513B (en) 2018-05-31
AU2007322362A1 (en) 2008-05-29
CA3004028A1 (en) 2008-05-29
KR20090118906A (ko) 2009-11-18
IL198513A0 (en) 2010-02-17
WO2008063211A2 (en) 2008-05-29
EP2096912A2 (en) 2009-09-09
EP2096912A4 (en) 2010-01-06
KR20140098863A (ko) 2014-08-08
US20070167416A1 (en) 2007-07-19
CN101610670A (zh) 2009-12-23
WO2008063211A3 (en) 2008-11-20
MX2009004826A (es) 2009-07-17
JP2010509326A (ja) 2010-03-25
DK2096912T3 (en) 2018-08-27
US8921344B2 (en) 2014-12-30
CA2668441A1 (en) 2008-05-29
EP2096912B1 (en) 2018-05-30

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Effective date: 20181102