CA2905570A1 - Salts, co-crystals, and polymorphs of an anxiolytic compound - Google Patents
Salts, co-crystals, and polymorphs of an anxiolytic compound Download PDFInfo
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- CA2905570A1 CA2905570A1 CA2905570A CA2905570A CA2905570A1 CA 2905570 A1 CA2905570 A1 CA 2905570A1 CA 2905570 A CA2905570 A CA 2905570A CA 2905570 A CA2905570 A CA 2905570A CA 2905570 A1 CA2905570 A1 CA 2905570A1
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
-
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P25/04—Centrally acting analgesics, e.g. opioids
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C55/00—Saturated compounds having more than one carboxyl group bound to acyclic carbon atoms
- C07C55/02—Dicarboxylic acids
- C07C55/10—Succinic acid
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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- Rheumatology (AREA)
- Hospice & Palliative Care (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361798926P | 2013-03-15 | 2013-03-15 | |
| US61/798,926 | 2013-03-15 | ||
| PCT/AU2014/000272 WO2014138812A1 (en) | 2013-03-15 | 2014-03-14 | Salts, co-crystals, and polymorphs of an anxiolytic compound |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2905570A1 true CA2905570A1 (en) | 2014-09-18 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2905570A Abandoned CA2905570A1 (en) | 2013-03-15 | 2014-03-14 | Salts, co-crystals, and polymorphs of an anxiolytic compound |
Country Status (9)
| Country | Link |
|---|---|
| US (2) | US9745296B2 (https=) |
| EP (1) | EP2970247A4 (https=) |
| JP (1) | JP2016510768A (https=) |
| CN (1) | CN105492440A (https=) |
| AU (2) | AU2014231722B2 (https=) |
| CA (1) | CA2905570A1 (https=) |
| HK (1) | HK1220191A1 (https=) |
| MX (1) | MX2015013059A (https=) |
| WO (1) | WO2014138812A1 (https=) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN112964689A (zh) * | 2015-12-15 | 2021-06-15 | 诺威量测设备股份有限公司 | 测量图案化结构的一个或多个特征时使用的方法和系统 |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6688434B2 (en) | 2002-02-22 | 2004-02-10 | Ecolab Inc. | Conveyor and lubricating apparatus, lubricant dispensing device, and method for applying lubricant to conveyor |
| CN105541701A (zh) * | 2015-12-11 | 2016-05-04 | 吉林大学珠海学院 | 以顺丁烯二酸为前驱体的去铁酮药物共晶及其制备方法 |
| WO2019109150A1 (en) * | 2017-12-07 | 2019-06-13 | Bionomics Limited | Methods of treating agitation |
| US20210393621A1 (en) | 2018-10-26 | 2021-12-23 | The Research Foundation For The State University Of New York | Combination serotonin specific reuptake inhibitor and serotonin 1a receptor partial agonist for reducing l-dopa-induced dyskinesia |
| CA3149182A1 (en) * | 2019-09-23 | 2021-04-01 | Bionomics Limited | Therapeutic formulations and uses thereof |
| AU2023201463A1 (en) * | 2023-03-08 | 2024-09-26 | Bionomics Limited | Method of treating social anxiety disorder |
| CN121646412A (zh) * | 2023-08-08 | 2026-03-10 | 株式会社明治 | 昼夜节律的调整 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2535803A1 (en) * | 2003-08-21 | 2005-03-03 | Transoral Pharmaceuticals, Inc. | Compositions for delivering 5-ht agonists across the oral mucosa and methods of use thereof |
| NZ576036A (en) * | 2006-10-16 | 2010-10-29 | Bionomics Ltd | Naphthyridine containing compounds for treating anxiety disorders |
| DE102006060598A1 (de) * | 2006-12-21 | 2008-06-26 | Merck Patent Gmbh | Tetrahydrobenzoisoxazole |
| GB0706044D0 (en) * | 2007-03-28 | 2007-05-09 | Syngenta Ltd | C0-Crystals |
| CN104230936A (zh) * | 2009-12-03 | 2014-12-24 | 阿斯利康(瑞典)有限公司 | 三唑并[4,5-d]嘧啶血小板聚集抑制剂的共晶体 |
| US20140051701A1 (en) * | 2011-03-02 | 2014-02-20 | Bionomics Limited | Methods of treating a disease or condition of the central nervous system |
| EP2707367B1 (en) * | 2011-05-12 | 2019-10-09 | Bionomics Limited | Methods for preparing naphthyridines |
| AU2013204159B2 (en) * | 2013-03-15 | 2015-05-07 | Bionomics Limited | A Crystalline Form of an Anxiolytic Compound |
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2014
- 2014-03-14 MX MX2015013059A patent/MX2015013059A/es unknown
- 2014-03-14 EP EP14765186.3A patent/EP2970247A4/en not_active Withdrawn
- 2014-03-14 CA CA2905570A patent/CA2905570A1/en not_active Abandoned
- 2014-03-14 US US14/776,643 patent/US9745296B2/en active Active
- 2014-03-14 JP JP2015561831A patent/JP2016510768A/ja active Pending
- 2014-03-14 WO PCT/AU2014/000272 patent/WO2014138812A1/en not_active Ceased
- 2014-03-14 HK HK16108260.8A patent/HK1220191A1/zh unknown
- 2014-03-14 AU AU2014231722A patent/AU2014231722B2/en active Active
- 2014-03-14 CN CN201480028564.4A patent/CN105492440A/zh active Pending
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2017
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- 2017-08-25 US US15/687,274 patent/US10266529B2/en active Active
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN112964689A (zh) * | 2015-12-15 | 2021-06-15 | 诺威量测设备股份有限公司 | 测量图案化结构的一个或多个特征时使用的方法和系统 |
Also Published As
| Publication number | Publication date |
|---|---|
| EP2970247A1 (en) | 2016-01-20 |
| AU2017201916A1 (en) | 2017-04-13 |
| AU2017201916B2 (en) | 2018-09-27 |
| EP2970247A4 (en) | 2016-08-10 |
| US10266529B2 (en) | 2019-04-23 |
| US20170362230A1 (en) | 2017-12-21 |
| AU2014231722B2 (en) | 2016-12-22 |
| AU2014231722A1 (en) | 2015-09-24 |
| MX2015013059A (es) | 2016-08-05 |
| JP2016510768A (ja) | 2016-04-11 |
| WO2014138812A1 (en) | 2014-09-18 |
| HK1220191A1 (zh) | 2017-04-28 |
| CN105492440A (zh) | 2016-04-13 |
| US20160185770A1 (en) | 2016-06-30 |
| US9745296B2 (en) | 2017-08-29 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EEER | Examination request |
Effective date: 20190220 |
|
| FZDE | Discontinued |
Effective date: 20210831 |