CA2879824A1 - Sels de saxagliptine - Google Patents

Sels de saxagliptine Download PDF

Info

Publication number
CA2879824A1
CA2879824A1 CA2879824A CA2879824A CA2879824A1 CA 2879824 A1 CA2879824 A1 CA 2879824A1 CA 2879824 A CA2879824 A CA 2879824A CA 2879824 A CA2879824 A CA 2879824A CA 2879824 A1 CA2879824 A1 CA 2879824A1
Authority
CA
Canada
Prior art keywords
saxagliptin
acetate
process according
bicarbonate
bisulphate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA2879824A
Other languages
English (en)
Inventor
Ram Chander Aryan
Ashwani Kumar Singh
Amit Sharma
Ramendra Singh Rathore
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Ranbaxy Laboratories Ltd
Original Assignee
Ranbaxy Laboratories Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ranbaxy Laboratories Ltd filed Critical Ranbaxy Laboratories Ltd
Publication of CA2879824A1 publication Critical patent/CA2879824A1/fr
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • General Chemical & Material Sciences (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
CA2879824A 2012-07-02 2013-07-02 Sels de saxagliptine Abandoned CA2879824A1 (fr)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
IN2061DE2012 2012-07-02
IN2061/DEL/2012 2012-07-02
IN3917DE2012 2012-12-19
IN3917/DEL/2012 2012-12-19
PCT/IB2013/055429 WO2014006569A2 (fr) 2012-07-02 2013-07-02 Sels de saxagliptine

Publications (1)

Publication Number Publication Date
CA2879824A1 true CA2879824A1 (fr) 2014-01-09

Family

ID=54193750

Family Applications (1)

Application Number Title Priority Date Filing Date
CA2879824A Abandoned CA2879824A1 (fr) 2012-07-02 2013-07-02 Sels de saxagliptine

Country Status (5)

Country Link
EP (1) EP2867206A2 (fr)
AU (1) AU2013285078A1 (fr)
CA (1) CA2879824A1 (fr)
SG (1) SG11201408619WA (fr)
WO (1) WO2014006569A2 (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013175297A1 (fr) 2012-05-24 2013-11-28 Apotex Pharmachem India Pvt. Ltd Sels de saxagliptine avec des acides organiques
WO2015166466A1 (fr) * 2014-05-01 2015-11-05 Sun Pharmaceutical Industries Limited Forme cristalline d'acétate de saxagliptine

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6395767B2 (en) * 2000-03-10 2002-05-28 Bristol-Myers Squibb Company Cyclopropyl-fused pyrrolidine-based inhibitors of dipeptidyl peptidase IV and method
US7420079B2 (en) 2002-12-09 2008-09-02 Bristol-Myers Squibb Company Methods and compounds for producing dipeptidyl peptidase IV inhibitors and intermediates thereof
TW200538122A (en) 2004-03-31 2005-12-01 Bristol Myers Squibb Co Process for preparing a dipeptidyl peptidase Ⅳ inhibitor and intermediates employed therein
US7741082B2 (en) 2004-04-14 2010-06-22 Bristol-Myers Squibb Company Process for preparing dipeptidyl peptidase IV inhibitors and intermediates therefor
US7214702B2 (en) 2004-05-25 2007-05-08 Bristol-Myers Squibb Company Process for producing a dipeptidyl peptidase IV inhibitor
PE20090696A1 (es) * 2007-04-20 2009-06-20 Bristol Myers Squibb Co Formas cristalinas de saxagliptina y procesos para preparar las mismas
WO2010115974A1 (fr) 2009-04-09 2010-10-14 Sandoz Ag Formes cristallines de la saxagliptine
WO2012017029A1 (fr) * 2010-08-06 2012-02-09 Sandoz Ag Nouveaux sels de saxagliptine comportant des diacides organiques
WO2012017028A1 (fr) 2010-08-06 2012-02-09 Sandoz Ag Nouveau composé cristallin comprenant de la saxagliptine et de l'acide phosphorique
US8410288B2 (en) 2010-10-04 2013-04-02 Teva Pharmaceutical Industries Ltd. Polymorphs of Saxagliptin hydrochloride and processes for preparing them
CN102086172A (zh) * 2011-01-13 2011-06-08 廖国超 沙格列汀的药用盐及其制备方法

Also Published As

Publication number Publication date
SG11201408619WA (en) 2015-01-29
WO2014006569A2 (fr) 2014-01-09
EP2867206A2 (fr) 2015-05-06
AU2013285078A1 (en) 2015-01-29
WO2014006569A3 (fr) 2014-03-06

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Legal Events

Date Code Title Description
EEER Examination request

Effective date: 20141223

FZDE Dead

Effective date: 20170517