SG11201408619WA - Saxagliptin salts - Google Patents
Saxagliptin saltsInfo
- Publication number
- SG11201408619WA SG11201408619WA SG11201408619WA SG11201408619WA SG11201408619WA SG 11201408619W A SG11201408619W A SG 11201408619WA SG 11201408619W A SG11201408619W A SG 11201408619WA SG 11201408619W A SG11201408619W A SG 11201408619WA SG 11201408619W A SG11201408619W A SG 11201408619WA
- Authority
- SG
- Singapore
- Prior art keywords
- saxagliptin
- international
- delhi
- singh
- del
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Diabetes (AREA)
- General Chemical & Material Sciences (AREA)
- Emergency Medicine (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Endocrinology (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
(12) INTERNATIONAL APPLICATION PUBLISHED UNDER THE PATENT COOPERATION TREATY (PCT) (19) World Intellectual Property Organization International Bureau (43) International Publication Date 9 January 2014 (09.01.2014) WIPOIPCT (10) International Publication Number WO 2014/006569 A2 (51) International Patent Classification: C07D 209/52 (2006.01) (21) International Application Number: PCT/IB2013/055429 2 July 2013 (02.07.2013) (22) International Filing Date: (25) Filing Language: English (26) Publication Language: English (30) Priority Data: 2061/DEL/2012 2 July 2012 (02.07.2012) IN 3917/DEL/2012 19 December 2012 (19.12.2012) IN (71) Applicant: RANBAXY LABORATORIES LIMITED [IN/IN]; Head Office: 12th Floor, Devika Tower, 06 Nehru Place, New Delhi, Delhi 110019 (IN). (72) Inventors: ARYAN, Ram, Chander; 1066, Sector-A, Pocket-A, Vasant Kunj, New Delhi, Delhi 110070 (IN). SINGH, Ashwani, Kumar; Opposite Post Office, Main Road, Khemganj, Sirsaganj, Firozabad, Uttar Pradesh 205151 (IN). SHARMA, Amit; House No. 108/B-l, Mod el Town, Pinjore, Panchkula, Haryana 134102 (IN). RATHORE, Ramendra, Singh; House No. 4/1, Mohalla, Chobdaran, Farrukhabad, Uttar Pradesh 209625 (IN). (81) Designated States (unless otherwise indicated, for every kind of national protection available)'. AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW. (84) Designated States (unless otherwise indicated, for every kind of regional protection available)'. ARIPO (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, UG, ZM, ZW), Eurasian (AM, AZ, BY, KG, KZ, RU, TJ, TM), European (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR), OAPI (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG). Published: — without international search report and to be republished upon receipt of that report (Rule 48.2(g)) CJ as o o o CJ (54) Title: SAXAGLIPTIN SALTS (57) Abstract: The present invention provides saxagliptin bisulphate, saxagliptin acetate, saxagliptin oxalate, saxagliptin bicarbon ate, and saxagliptin carbonate, their polymorphic forms, processes for their preparation, and pharmaceutical compositions thereof.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN2061DE2012 | 2012-07-02 | ||
IN3917DE2012 | 2012-12-19 | ||
PCT/IB2013/055429 WO2014006569A2 (en) | 2012-07-02 | 2013-07-02 | Saxagliptin salts |
Publications (1)
Publication Number | Publication Date |
---|---|
SG11201408619WA true SG11201408619WA (en) | 2015-01-29 |
Family
ID=54193750
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SG11201408619WA SG11201408619WA (en) | 2012-07-02 | 2013-07-02 | Saxagliptin salts |
Country Status (5)
Country | Link |
---|---|
EP (1) | EP2867206A2 (en) |
AU (1) | AU2013285078A1 (en) |
CA (1) | CA2879824A1 (en) |
SG (1) | SG11201408619WA (en) |
WO (1) | WO2014006569A2 (en) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2013175297A1 (en) | 2012-05-24 | 2013-11-28 | Apotex Pharmachem India Pvt. Ltd | Salts of saxagliptin with organic acids |
WO2015166466A1 (en) * | 2014-05-01 | 2015-11-05 | Sun Pharmaceutical Industries Limited | Crystalline form of saxagliptin acetate |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6395767B2 (en) * | 2000-03-10 | 2002-05-28 | Bristol-Myers Squibb Company | Cyclopropyl-fused pyrrolidine-based inhibitors of dipeptidyl peptidase IV and method |
US7420079B2 (en) | 2002-12-09 | 2008-09-02 | Bristol-Myers Squibb Company | Methods and compounds for producing dipeptidyl peptidase IV inhibitors and intermediates thereof |
TW200538122A (en) | 2004-03-31 | 2005-12-01 | Bristol Myers Squibb Co | Process for preparing a dipeptidyl peptidase Ⅳ inhibitor and intermediates employed therein |
US7741082B2 (en) | 2004-04-14 | 2010-06-22 | Bristol-Myers Squibb Company | Process for preparing dipeptidyl peptidase IV inhibitors and intermediates therefor |
US7214702B2 (en) | 2004-05-25 | 2007-05-08 | Bristol-Myers Squibb Company | Process for producing a dipeptidyl peptidase IV inhibitor |
PE20090696A1 (en) * | 2007-04-20 | 2009-06-20 | Bristol Myers Squibb Co | CRYSTALLINE FORMS OF SAXAGLIPTIN AND PROCESSES FOR PREPARING THEM |
CN102459170B (en) | 2009-04-09 | 2014-07-23 | 桑多斯股份公司 | Crystal forms of saxagliptin |
EP2601175A1 (en) | 2010-08-06 | 2013-06-12 | Sandoz AG | A novel crystalline compound comprising saxagliptin and phosphoric acid |
WO2012017029A1 (en) * | 2010-08-06 | 2012-02-09 | Sandoz Ag | Novel salts of saxagrliptin with organic di-acids |
US8410288B2 (en) | 2010-10-04 | 2013-04-02 | Teva Pharmaceutical Industries Ltd. | Polymorphs of Saxagliptin hydrochloride and processes for preparing them |
CN102086172A (en) * | 2011-01-13 | 2011-06-08 | 廖国超 | Medicinal salts of saxagliptin and preparation methods of medicinal salts |
-
2013
- 2013-07-02 SG SG11201408619WA patent/SG11201408619WA/en unknown
- 2013-07-02 EP EP13762566.1A patent/EP2867206A2/en not_active Withdrawn
- 2013-07-02 AU AU2013285078A patent/AU2013285078A1/en not_active Abandoned
- 2013-07-02 CA CA2879824A patent/CA2879824A1/en not_active Abandoned
- 2013-07-02 WO PCT/IB2013/055429 patent/WO2014006569A2/en active Application Filing
Also Published As
Publication number | Publication date |
---|---|
WO2014006569A2 (en) | 2014-01-09 |
EP2867206A2 (en) | 2015-05-06 |
CA2879824A1 (en) | 2014-01-09 |
AU2013285078A1 (en) | 2015-01-29 |
WO2014006569A3 (en) | 2014-03-06 |
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