CA2836827C - Alpha amino acid ester-drug conjugates hydrolysable by carboxylesterases - Google Patents
Alpha amino acid ester-drug conjugates hydrolysable by carboxylesterases Download PDFInfo
- Publication number
- CA2836827C CA2836827C CA2836827A CA2836827A CA2836827C CA 2836827 C CA2836827 C CA 2836827C CA 2836827 A CA2836827 A CA 2836827A CA 2836827 A CA2836827 A CA 2836827A CA 2836827 C CA2836827 C CA 2836827C
- Authority
- CA
- Canada
- Prior art keywords
- amino acid
- inhibitor
- ester
- conjugate
- acid ester
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
Links
Landscapes
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
- Enzymes And Modification Thereof (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0509226A GB0509226D0 (en) | 2005-05-05 | 2005-05-05 | Enzyme and receptor modulation |
| GB0509226.7 | 2005-05-05 | ||
| US68054205P | 2005-05-13 | 2005-05-13 | |
| US60/680,542 | 2005-05-13 | ||
| CA2607020A CA2607020C (en) | 2005-05-05 | 2006-05-04 | Alpha amino acid ester-drug conjugates hydrolysable by carboxylesterases |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2607020A Division CA2607020C (en) | 2005-05-05 | 2006-05-04 | Alpha amino acid ester-drug conjugates hydrolysable by carboxylesterases |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CA2836827A1 CA2836827A1 (en) | 2006-11-09 |
| CA2836827C true CA2836827C (en) | 2016-05-03 |
Family
ID=34685158
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2836827A Active CA2836827C (en) | 2005-05-05 | 2006-05-04 | Alpha amino acid ester-drug conjugates hydrolysable by carboxylesterases |
Country Status (10)
| Country | Link |
|---|---|
| CN (1) | CN101171039B (pt) |
| CA (1) | CA2836827C (pt) |
| DK (1) | DK1877098T3 (pt) |
| ES (2) | ES2415244T3 (pt) |
| GB (1) | GB0509226D0 (pt) |
| NZ (1) | NZ561710A (pt) |
| PT (1) | PT1877098E (pt) |
| SG (1) | SG2014007512A (pt) |
| SI (1) | SI1877098T1 (pt) |
| ZA (1) | ZA200708283B (pt) |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1231919B1 (en) * | 1999-09-08 | 2015-09-30 | Sloan-Kettering Institute For Cancer Research | Derivatives of 1-amino-1-(hetero)arylaminocarbonyl-6-hydroxyaminocarbonylhexane useful in the treatment of tumors |
| JP2007509082A (ja) * | 2003-10-22 | 2007-04-12 | アルピダ エー／エス | ペプチドデホルミラーゼ阻害剤としてのベンゾイミダゾール誘導体類およびそれらの使用 |
-
2005
- 2005-05-05 GB GB0509226A patent/GB0509226D0/en not_active Ceased
-
2006
- 2006-05-04 ES ES06727008T patent/ES2415244T3/es active Active
- 2006-05-04 SG SG2014007512A patent/SG2014007512A/en unknown
- 2006-05-04 ES ES08075300.7T patent/ES2577433T3/es active Active
- 2006-05-04 CN CN200680014981.9A patent/CN101171039B/zh not_active Expired - Fee Related
- 2006-05-04 PT PT06727008T patent/PT1877098E/pt unknown
- 2006-05-04 CA CA2836827A patent/CA2836827C/en active Active
- 2006-05-04 NZ NZ561710A patent/NZ561710A/en not_active IP Right Cessation
- 2006-05-04 DK DK06727008.2T patent/DK1877098T3/da active
- 2006-05-04 SI SI200631620T patent/SI1877098T1/sl unknown
-
2007
- 2007-09-27 ZA ZA200708283A patent/ZA200708283B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| PT1877098E (pt) | 2013-07-31 |
| GB0509226D0 (en) | 2005-06-15 |
| NZ561710A (en) | 2010-08-27 |
| CN101171039B (zh) | 2013-01-23 |
| SG2014007512A (en) | 2014-03-28 |
| SI1877098T1 (sl) | 2013-08-30 |
| CN101171039A (zh) | 2008-04-30 |
| DK1877098T3 (da) | 2013-07-08 |
| ZA200708283B (en) | 2008-10-29 |
| ES2415244T3 (es) | 2013-07-24 |
| ES2577433T3 (es) | 2016-07-14 |
| CA2836827A1 (en) | 2006-11-09 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EEER | Examination request |
Effective date: 20131217 |